The selective adenosine A(2A) receptor antagonist SCH 58261 discriminates between two different binding sites for [3H]-CGS 21680 in the rat brain

Naunyn-Schmiedeberg's Archives of Pharmacology

Volumn 354, Issue 4, 1996, Pages 539-541

  Lindström, Karin ^a   Ongini, Ennio ^b   Fredholm, Bertil B ^a  

^a KAROLINSKA INSTITUTE   (Sweden)

^b San Raffaele Science Park   (Italy)

Author keywords

Adenosine receptors; Autoradiography hippocampus; Cortex; Striatum

Indexed keywords

2 [4 (2 CARBOXYETHYL)PHENETHYLAMINO]ADENOSINE 5' (N ETHYLCARBOXAMIDE); 5 AMINO 2 (2 FURYL) 7 (2 PHENYLETHYL)PYRAZOLO[4,3 E][1,2,4]TRIAZOLO[1,5 C]PYRIMIDINE; ADENOSINE A2 RECEPTOR; ADENOSINE A2 RECEPTOR ANTAGONIST; ADENOSINE; ADENOSINE RECEPTOR; DRUG DERIVATIVE; PHENETHYLAMINE DERIVATIVE; PYRIMIDINE DERIVATIVE; TRIAZOLE DERIVATIVE; TRITIUM;

ANIMAL TISSUE; ARTICLE; AUTORADIOGRAPHY; BINDING SITE; BRAIN CORTEX; BRAIN REGION; CONTROLLED STUDY; CORPUS STRIATUM; DRUG RECEPTOR BINDING; NONHUMAN; QUANTITATIVE ASSAY; RAT; ANIMAL; BINDING COMPETITION; BRAIN; DRUG ANTAGONISM; DRUG POTENTIATION; HIPPOCAMPUS; METABOLISM; PROTEIN BINDING;

ADENOSINE; ANIMALS; AUTORADIOGRAPHY; BINDING, COMPETITIVE; BRAIN; CEREBRAL CORTEX; CORPUS STRIATUM; HIPPOCAMPUS; PHENETHYLAMINES; PROTEIN BINDING; PYRIMIDINES; RATS; RECEPTORS, PURINERGIC P1; TRIAZOLES; TRITIUM;

EID: 0029658870     PISSN: 00281298     EISSN: None     Source Type: Journal    
DOI: 10.1007/BF00168448     Document Type: Article

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