Synthesis of the tritium labeled SCH 58261, a new non-xanthine A(2A) adenosine receptor antagonist

Journal of Labelled Compounds and Radiopharmaceuticals

Volumn 38, Issue 8, 1996, Pages 725-732

  Baraldi, Pier Giovanni ^a   Cacciari, Barbara ^a   Dionisotti, Silvio ^b   Egan, Judith ^c   Spalluto, Giampiero ^a   Zocchi, Cristina ^b  

^a UNIVERSITY OF FERRARA   (Italy)

^b Faculty of Medicine   (Italy)

^c DUPONT COMPANY   (United States)

Author keywords

3H SCH 58261; A(2A) adenosine receptors; A(2A) receptor antagonists; Adenosine receptors; Binding assay

Indexed keywords

AIR PURIFICATION; AROMATIC COMPOUNDS;

% REDUCTIONS; 3H-SCH 58261; A(2A) ADENOSINE RECEPTOR; A(2A) RECEPTOR ANTAGONIST; ADENOSINE RECEPTOR; BINDING ASSAYS; RADIOCHEMICAL PURITY; RECEPTOR ANTAGONISTS; TRITIUM GAS;

TRITIUM;

5 AMINO 2 (2 FURYL) 7 (2 PHENYLETHYL)PYRAZOLO[4,3 E][1,2,4]TRIAZOLO[1,5 C]PYRIMIDINE; ADENOSINE RECEPTOR BLOCKING AGENT; TRITIUM;

ANIMAL EXPERIMENT; ANIMAL TISSUE; ARTICLE; CONTROLLED STUDY; CORPUS STRIATUM; DRUG BINDING; DRUG SYNTHESIS; ISOTOPE LABELING; RAT;

ANIMALIA; TRITIUM;

EID: 0029900723     PISSN: 03624803     EISSN: None     Source Type: Journal    
DOI: 10.1002/(SICI)1099-1344(199608)38:8<725::AID-JLCR885>3.0.CO;2-G     Document Type: Article

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