메뉴 건너뛰기




Volumn 114, Issue , 2018, Pages 346-355

Alginate as a potential diphase solid dispersion carrier with enhanced drug dissolution and improved storage stability

Author keywords

Alginate; Hansen solubility parameter; Miscibility; Raman mapping; Solid dispersion; Stability

Indexed keywords

ALGINIC ACID; DRUG CARRIER; INDOMETACIN; MEVINOLIN; GLUCURONIC ACID; HEXURONIC ACID;

EID: 85040017295     PISSN: 09280987     EISSN: 18790720     Source Type: Journal    
DOI: 10.1016/j.ejps.2017.12.028     Document Type: Article
Times cited : (41)

References (30)
  • 1
    • 84947255835 scopus 로고    scopus 로고
    • Sodium alginate as a potential carrier in solid dispersion formulations to enhance dissolution rate and apparent water solubility of BCS II drugs
    • Borba, Amarante P.A., Pinotti, M., Maduro de Campos, C.E., Pezzini, B.R., Stulzer, H.K., Sodium alginate as a potential carrier in solid dispersion formulations to enhance dissolution rate and apparent water solubility of BCS II drugs. Carbohydr. Polym. 137 (2016), 350–359.
    • (2016) Carbohydr. Polym. , vol.137 , pp. 350-359
    • Borba, A.P.A.1    Pinotti, M.2    Maduro de Campos, C.E.3    Pezzini, B.R.4    Stulzer, H.K.5
  • 2
    • 0037074108 scopus 로고    scopus 로고
    • The mechanisms of drug release from solid dispersions in water-soluble polymers
    • Craig, D.Q.M., The mechanisms of drug release from solid dispersions in water-soluble polymers. Int. J. Pharm. 231:2002 (2002), 131–144.
    • (2002) Int. J. Pharm. , vol.231 , Issue.2002 , pp. 131-144
    • Craig, D.Q.M.1
  • 3
    • 84875522078 scopus 로고    scopus 로고
    • Smart porous microparticles based on gelatin/sodium alginate polyelectrolyte complex
    • Devi, N., Kakati, D.K., Smart porous microparticles based on gelatin/sodium alginate polyelectrolyte complex. J. Food Eng. 117 (2013), 193–204.
    • (2013) J. Food Eng. , vol.117 , pp. 193-204
    • Devi, N.1    Kakati, D.K.2
  • 4
    • 34547864243 scopus 로고    scopus 로고
    • Drug delivery strategies for poorly water-soluble drugs
    • Fahr, A., Liu, X., Drug delivery strategies for poorly water-soluble drugs. Expert Opin. Drug Deliv. 4 (2007), 403–416.
    • (2007) Expert Opin. Drug Deliv. , vol.4 , pp. 403-416
    • Fahr, A.1    Liu, X.2
  • 5
    • 64649100465 scopus 로고    scopus 로고
    • Hydroxypropyl methylcellulose acetate succinate-based spray-dried dispersions: an overview
    • Friesen, D.T., Shanker, R., Crew, M., Smithey, D.T., Curatolo, W.J., Nightingale, J.A.S., Hydroxypropyl methylcellulose acetate succinate-based spray-dried dispersions: an overview. Mol. Pharm. 5 (2008), 1003–1019.
    • (2008) Mol. Pharm. , vol.5 , pp. 1003-1019
    • Friesen, D.T.1    Shanker, R.2    Crew, M.3    Smithey, D.T.4    Curatolo, W.J.5    Nightingale, J.A.S.6
  • 6
    • 33746474818 scopus 로고    scopus 로고
    • Polyionic hydrocolloids for the intestinal delivery of protein drugs: alginate and chitosan - a review
    • George, M., Abraham, T.E., Polyionic hydrocolloids for the intestinal delivery of protein drugs: alginate and chitosan - a review. J. Control. Release 114 (2006), 1–14.
    • (2006) J. Control. Release , vol.114 , pp. 1-14
    • George, M.1    Abraham, T.E.2
  • 7
    • 85019846697 scopus 로고    scopus 로고
    • Exploration of alginates as potential stabilizers of nanosuspension
    • Guan, J., Zhang, Y., Liu, Q., Zhang, X., Chokshi, R., Mao, S., Exploration of alginates as potential stabilizers of nanosuspension. AAPS PharmSciTech 18 (2017), 3172–3181.
    • (2017) AAPS PharmSciTech , vol.18 , pp. 3172-3181
    • Guan, J.1    Zhang, Y.2    Liu, Q.3    Zhang, X.4    Chokshi, R.5    Mao, S.6
  • 8
    • 28444461830 scopus 로고    scopus 로고
    • Drug nanocrystals of poorly soluble drugs produced by high pressure homogenisation
    • Keck, C.M., Muller, R.H., Drug nanocrystals of poorly soluble drugs produced by high pressure homogenisation. Eur. J. Pharm. Biopharm. 62 (2006), 3–16.
    • (2006) Eur. J. Pharm. Biopharm. , vol.62 , pp. 3-16
    • Keck, C.M.1    Muller, R.H.2
  • 9
    • 84919921268 scopus 로고    scopus 로고
    • Pharmaceutical particle technologies: an approach to improve drug solubility, dissolution and bioavailability
    • Khadka, P., Ro, J., Kim, H., Kim, I., Kim, J.T., Kim, H., Cho, J.M., Yun, G., Lee, J., Pharmaceutical particle technologies: an approach to improve drug solubility, dissolution and bioavailability. Asian J. Pharm. Sci. 9 (2014), 304–316.
    • (2014) Asian J. Pharm. Sci. , vol.9 , pp. 304-316
    • Khadka, P.1    Ro, J.2    Kim, H.3    Kim, I.4    Kim, J.T.5    Kim, H.6    Cho, J.M.7    Yun, G.8    Lee, J.9
  • 11
    • 84877820916 scopus 로고    scopus 로고
    • Drug release characteristics from chitosan-alginate matrix tablets based on the theory of self-assembled film
    • Li, L., Wang, L.L., Shao, Y., Ni, R., Zhang, T.T., Mao, S.R., Drug release characteristics from chitosan-alginate matrix tablets based on the theory of self-assembled film. Int. J. Pharm. 450 (2013), 197–207.
    • (2013) Int. J. Pharm. , vol.450 , pp. 197-207
    • Li, L.1    Wang, L.L.2    Shao, Y.3    Ni, R.4    Zhang, T.T.5    Mao, S.R.6
  • 12
    • 31144464449 scopus 로고    scopus 로고
    • Evaluation of sodium alginate as drug release modifier in matrix tablets
    • Liew, C.V., Chan, L.W., Ching, A.L., Heng, P.W.S., Evaluation of sodium alginate as drug release modifier in matrix tablets. Int. J. Pharm. 309 (2006), 25–37.
    • (2006) Int. J. Pharm. , vol.309 , pp. 25-37
    • Liew, C.V.1    Chan, L.W.2    Ching, A.L.3    Heng, P.W.S.4
  • 13
    • 6444234760 scopus 로고    scopus 로고
    • The role of the medicinal chemist in drug discovery - then and now
    • Lombardino, J.G., Lowe, J.A., The role of the medicinal chemist in drug discovery - then and now. Nat. Rev. Drug Discov. 3 (2004), 853–862.
    • (2004) Nat. Rev. Drug Discov. , vol.3 , pp. 853-862
    • Lombardino, J.G.1    Lowe, J.A.2
  • 14
    • 33749442356 scopus 로고    scopus 로고
    • Theoretical and practical approaches for prediction of drug-polymer miscibility and solubility
    • Marsac, P.J., Shamblin, S.L., Taylor, L.S., Theoretical and practical approaches for prediction of drug-polymer miscibility and solubility. Pharm. Res. 23 (2006), 2417–2426.
    • (2006) Pharm. Res. , vol.23 , pp. 2417-2426
    • Marsac, P.J.1    Shamblin, S.L.2    Taylor, L.S.3
  • 15
    • 0032756138 scopus 로고    scopus 로고
    • Physical properties of solid molecular dispersions of indomethacin with poly(vinylpyrrolidone) and poly(vinylpyrrolidone-co-vinyl-acetate) in relation to indomethacin crystallization
    • Matsumoto, T., Zografi, G., Physical properties of solid molecular dispersions of indomethacin with poly(vinylpyrrolidone) and poly(vinylpyrrolidone-co-vinyl-acetate) in relation to indomethacin crystallization. Pharm. Res. 16 (1999), 1722–1728.
    • (1999) Pharm. Res. , vol.16 , pp. 1722-1728
    • Matsumoto, T.1    Zografi, G.2
  • 16
    • 84963854435 scopus 로고    scopus 로고
    • Effect of water on molecular mobility and physical stability of amorphous pharmaceuticals
    • Mehta, M., Kothari, K., Ragoonanan, V., Suryanarayanan, R., Effect of water on molecular mobility and physical stability of amorphous pharmaceuticals. Mol. Pharm. 13 (2016), 1339–1346.
    • (2016) Mol. Pharm. , vol.13 , pp. 1339-1346
    • Mehta, M.1    Kothari, K.2    Ragoonanan, V.3    Suryanarayanan, R.4
  • 17
    • 84977642034 scopus 로고    scopus 로고
    • Solid microcrystalline dispersion films as a new strategy to improve the dissolution rate of poorly water soluble drugs: a case study using olanzapine
    • de Mohac, L.M., Pina, M.D., Raimi-Abraham, B.T., Solid microcrystalline dispersion films as a new strategy to improve the dissolution rate of poorly water soluble drugs: a case study using olanzapine. Int. J. Pharm. 508 (2016), 42–50.
    • (2016) Int. J. Pharm. , vol.508 , pp. 42-50
    • de Mohac, L.M.1    Pina, M.D.2    Raimi-Abraham, B.T.3
  • 18
    • 84898026386 scopus 로고    scopus 로고
    • Evaluation of tadalafil nanosuspensions and their PEG solid dispersion matrices for enhancing its dissolution properties
    • Obeidat, W.M., Sallam, A.A., Evaluation of tadalafil nanosuspensions and their PEG solid dispersion matrices for enhancing its dissolution properties. AAPS PharmSciTech 15 (2014), 364–374.
    • (2014) AAPS PharmSciTech , vol.15 , pp. 364-374
    • Obeidat, W.M.1    Sallam, A.A.2
  • 19
    • 77949844000 scopus 로고    scopus 로고
    • Formulation design and photochemical studies on nanocrystal solid dispersion of curcumin with improved oral bioavailability
    • Onoue, S., Takahashi, H., Kawabata, Y., Seto, Y., Hatanaka, J., Timmermann, B., Yamada, S., Formulation design and photochemical studies on nanocrystal solid dispersion of curcumin with improved oral bioavailability. J. Pharm. Sci. 99 (2010), 1871–1881.
    • (2010) J. Pharm. Sci. , vol.99 , pp. 1871-1881
    • Onoue, S.1    Takahashi, H.2    Kawabata, Y.3    Seto, Y.4    Hatanaka, J.5    Timmermann, B.6    Yamada, S.7
  • 20
    • 84960110225 scopus 로고    scopus 로고
    • Characterization of solid dispersion of itraconazole prepared by solubilization in concentrated aqueous solutions of weak organic acids and drying
    • Parikh, T., Sandhu, H.K., Talele, T.T., Serajuddin, A.T.M., Characterization of solid dispersion of itraconazole prepared by solubilization in concentrated aqueous solutions of weak organic acids and drying. Pharm. Res. 33 (2016), 1456–1471.
    • (2016) Pharm. Res. , vol.33 , pp. 1456-1471
    • Parikh, T.1    Sandhu, H.K.2    Talele, T.T.3    Serajuddin, A.T.M.4
  • 21
    • 84965078970 scopus 로고    scopus 로고
    • Hot melt extruded Aprepitant-Soluplus solid dispersion: preformulation considerations, stability and in vitro study
    • Penumetcha, S.S., Gutta, L.N., Dhanala, H., Yamili, S., Challa, S., Rudraraju, S., Rudraraju, V., Hot melt extruded Aprepitant-Soluplus solid dispersion: preformulation considerations, stability and in vitro study. Drug Dev. Ind. Pharm. 42 (2016), 1609–1620.
    • (2016) Drug Dev. Ind. Pharm. , vol.42 , pp. 1609-1620
    • Penumetcha, S.S.1    Gutta, L.N.2    Dhanala, H.3    Yamili, S.4    Challa, S.5    Rudraraju, S.6    Rudraraju, V.7
  • 22
    • 79961026635 scopus 로고    scopus 로고
    • Thermal and microbial degradation of alginate-based superabsorbent polymer
    • Phang, Y.N., Chee, S.Y., Lee, C.O., Teh, Y.L., Thermal and microbial degradation of alginate-based superabsorbent polymer. Polym. Degrad. Stab. 96 (2011), 1653–1661.
    • (2011) Polym. Degrad. Stab. , vol.96 , pp. 1653-1661
    • Phang, Y.N.1    Chee, S.Y.2    Lee, C.O.3    Teh, Y.L.4
  • 23
    • 77953296607 scopus 로고    scopus 로고
    • Drug-polymer solubility and miscibility: stability consideration and practical challenges in amorphous solid dispersion development
    • Qian, F., Huang, J., Hussain, M.A., Drug-polymer solubility and miscibility: stability consideration and practical challenges in amorphous solid dispersion development. J. Pharm. Sci. 99 (2010), 2941–2947.
    • (2010) J. Pharm. Sci. , vol.99 , pp. 2941-2947
    • Qian, F.1    Huang, J.2    Hussain, M.A.3
  • 24
    • 84946606953 scopus 로고    scopus 로고
    • Development and characterization of amorphous nanofiber drug dispersions prepared using pressurized gyration
    • Raimi-Abraham, B.T., Mahalingam, S., Davies, P.J., Edirisinghe, M., Craig, D.Q.M., Development and characterization of amorphous nanofiber drug dispersions prepared using pressurized gyration. Mol. Pharm. 12 (2015), 3851–3861.
    • (2015) Mol. Pharm. , vol.12 , pp. 3851-3861
    • Raimi-Abraham, B.T.1    Mahalingam, S.2    Davies, P.J.3    Edirisinghe, M.4    Craig, D.Q.M.5
  • 25
    • 84951775551 scopus 로고    scopus 로고
    • Alginate biomaterial for the treatment of myocardial infarction: progress, translational strategies, and clinical outlook from ocean algae to patient bedside
    • Ruvinov, E., Cohen, S., Alginate biomaterial for the treatment of myocardial infarction: progress, translational strategies, and clinical outlook from ocean algae to patient bedside. Adv. Drug Deliv. Rev. 96 (2016), 54–76.
    • (2016) Adv. Drug Deliv. Rev. , vol.96 , pp. 54-76
    • Ruvinov, E.1    Cohen, S.2
  • 26
    • 84872130842 scopus 로고    scopus 로고
    • Hot melt extrusion (HME) for amorphous solid dispersions: predictive tools for processing and impact of drug-polymer interactions on supersaturation
    • Sarode, A.L., Sandhu, H., Shah, N., Malick, W., Zia, H., Hot melt extrusion (HME) for amorphous solid dispersions: predictive tools for processing and impact of drug-polymer interactions on supersaturation. Eur. J. Pharm. Sci. 48 (2013), 371–384.
    • (2013) Eur. J. Pharm. Sci. , vol.48 , pp. 371-384
    • Sarode, A.L.1    Sandhu, H.2    Shah, N.3    Malick, W.4    Zia, H.5
  • 27
    • 84984677936 scopus 로고    scopus 로고
    • Exploring the effect of hydrophilic and hydrophobic structure of grafted polymeric micelles on drug loading
    • Shi, C., Sun, Y., Wu, H., Zhu, C., Wei, G., Li, J., Chan, T., Ouyang, D., Mao, S., Exploring the effect of hydrophilic and hydrophobic structure of grafted polymeric micelles on drug loading. Int. J. Pharm. 512 (2016), 282–291.
    • (2016) Int. J. Pharm. , vol.512 , pp. 282-291
    • Shi, C.1    Sun, Y.2    Wu, H.3    Zhu, C.4    Wei, G.5    Li, J.6    Chan, T.7    Ouyang, D.8    Mao, S.9
  • 28
    • 84922682137 scopus 로고    scopus 로고
    • Preparation, characterization and in vitro/vivo evaluation of tectorigenin solid dispersion with improved dissolution and bioavailability
    • Shuai, S.P., Yue, S.L., Huang, Q.T., Wang, W., Yang, J.Y., Lan, K., Ye, L.M., Preparation, characterization and in vitro/vivo evaluation of tectorigenin solid dispersion with improved dissolution and bioavailability. Eur. J. Drug Metab. Pharmacokinet. 41 (2016), 413–422.
    • (2016) Eur. J. Drug Metab. Pharmacokinet. , vol.41 , pp. 413-422
    • Shuai, S.P.1    Yue, S.L.2    Huang, Q.T.3    Wang, W.4    Yang, J.Y.5    Lan, K.6    Ye, L.M.7
  • 29
    • 85010941395 scopus 로고    scopus 로고
    • Properties of Polymers: Their Correlation with Chemical Structure; their Numerical Estimation and Prediction from Additive Group Contributions
    • Elsevier
    • Van Krevelen, D.W., Te Nijenhuis, K., Properties of Polymers: Their Correlation with Chemical Structure; their Numerical Estimation and Prediction from Additive Group Contributions. 2009, Elsevier.
    • (2009)
    • Van Krevelen, D.W.1    Te Nijenhuis, K.2
  • 30
    • 84940521136 scopus 로고    scopus 로고
    • Physical stability of solid dispersions with respect to thermodynamic solubility of tadalafil in PVP-VA
    • Wlodarski, K., Sawicki, W., Kozyra, A., Tajber, L., Physical stability of solid dispersions with respect to thermodynamic solubility of tadalafil in PVP-VA. Eur. J. Pharm. Biopharm. 96 (2015), 237–246.
    • (2015) Eur. J. Pharm. Biopharm. , vol.96 , pp. 237-246
    • Wlodarski, K.1    Sawicki, W.2    Kozyra, A.3    Tajber, L.4


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.