Synthesis and antibacterial evaluation of series of novel tri-substituted-s-triazine derivatives

Medicinal Chemistry Research

Volumn 20, Issue 9, 2011, Pages 1603-1610

  Singh, Udaya Pratap ^a   Singh, Ramendra Kumar ^b   Bhat, Hans Raj ^a   Subhashchandra, Yadav Pankajkumar ^a   Kumar, Vikas ^a   Kumawat, Mukesh Kumar ^c   Gahtori, Prashant ^d  

^a SAM HIGGINBOTTOM UNIVERSITY OF AGRICULTURE   (India)

^b UNIVERSITY OF ALLAHABAD   (India)

^c NIMS UNIVERSITY   (India)

^d Devsthali Vidyapeeth College of Pharmacy   (India)

Author keywords

Amines; Antibacterial; MIC; S triazines

Indexed keywords

TRIAZINE DERIVATIVE;

ANTIBACTERIAL ACTIVITY; BACILLUS CEREUS; BACILLUS SUBTILIS; CONFERENCE PAPER; CONTROLLED STUDY; DRUG STRUCTURE; DRUG SYNTHESIS; ESCHERICHIA COLI; IN VITRO STUDY; KLEBSIELLA PNEUMONIAE; MINIMUM INHIBITORY CONCENTRATION; NONHUMAN; PHYSICAL CHEMISTRY; PSEUDOMONAS AERUGINOSA; STAPHYLOCOCCUS AUREUS;

EID: 85028095214     PISSN: 10542523     EISSN: 15548120     Source Type: Journal    
DOI: 10.1007/s00044-010-9446-7     Document Type: Conference Paper

References (11)

1. Bharti SK, Nath G, Tilak R, Singh SK (2010) Synthesis, anti-bacterial and anti-fungal activities of some novel Schiff bases containing 2,4-disubstituted thiazole ring. Eur J Med Chem 45:651-660
2. Devasia RA, Jones TF, Ward J, Stafford L, Hardin H, Bopp C, Beatty M, Mintz E, Schaffner W (2006) Endemically acquired foodborne outbreak of enterotoxin-producing Escherichia coli serotype O169:H41. Am J Med 119:168.e7-168.e10
3. Garaj V, Puccetti L, Fasolis G, Jean-Yves Winum, Jean-Louis M, Scozzafava A, Vullo D, Innocentia A, Supurana CT (2005) Carbonic anhydrase inhibitors: Novel sulfonamides incorporating 1,3,5-triazine moieties as inhibitors of the cytosolic and tumourassociated carbonic anhydrase isozymes I, II and IX. Bioorg Med Chem Lett 15:3102-3108 (Pubitemid 40755204)
4. Khalil AM, Berghot MA, Gouda MA (2009) Synthesis and antibacterial activity of some new thiazole and thiophene derivatives. Eur J Med Chem 44:4434-4440
5. Klenke B, Barrett MP, Brun R, Gilbert IH (2003) Antiplasmodial activity of a series of 1,3,5-triazine-substituted polyamines. J Antimicrob Chemother 52:290-293 (Pubitemid 36986894)
6. Mandal S, Bérubé G, Asselin E, Mohammad I, Richardson VJ, Gupta A, Pramanik SK, Williams AL, Mandal SK (2007) A novel series of potent cytotoxic agents targeting G2/M phase of the cell cycle and demonstrating cell killing by apoptosis in human breast cancer cells. Bioorg Med Chem Lett 17: 4955-4960 (Pubitemid 47187684)
7. National Committee for Clinical Laboratory Standards (1982) Standard methods for dilution antimicrobial susceptibility test for bacteria which grows aerobically. NCCLS, Villanova, p. 242
8. Projan SJ, Bradford PA (2007) Late stage antibacterial drugs in the clinical pipeline. Curr Opin Microbiol 10:441-446 (Pubitemid 350052689)
9. Qadri F, Svennerholm AM, Faruque ASG, Sack RB (2005) Enterotoxigenic Escherichia coli in developing countries: Epidemiology, microbiology, clinical features, treatment, and prevention. Clin Microbiol Rev 18:465-483 (Pubitemid 40995112)
10. Sharma P, Rane N, Gurram VK (2004) Synthesis and QSAR studies of pyrimido[4,5-d]pyrimidine-2,5-dione derivatives as potential antimicrobial agents. Bioorg Med Chem Lett 14:4185-4190 (Pubitemid 38916932)
11. Srinivas K, Srinivas U, Bhanuprakash K, Harakishore K, Murthy USN, Rao VJ (2006) Synthesis and antibacterial activity of various substituted s-triazines. Eur J Med Chem 41:1240-1246 (Pubitemid 44666218)