Synthesis, characterization and antimicrobial activity of thiazole, benzothiazole and pyrimidine derivatives bearing sydnone moieties

Pharmaceutical Chemistry Journal

Volumn 45, Issue 12, 2012, Pages 725-731

  Asundaria, S T ^a   Patel, K C ^a  

^a VEER NARMAD SOUTH GUJARAT UNIVERSITY   (India)

Author keywords

Antimicrobial activity; Benzothiazole; Pyrimidine; Sulfonamide; Sydnone; Thiazole

Indexed keywords

3 (4 CHLOROPHENYL) 4 [[(2,5 DICHLOROPHENYL) 6 (4 METHOXYPHENYL)PYRIMIDIN 2 YL]SULFAMOYL]SYDNONE; 3 (4 CHLOROPHENYL) 4 [[4 (3 METHOXYPHENYL) 6 (4 METHOXYPHENYL)PYRIMIDIN 2 YL]SULFAMOYL]SYDNONE; 3 (4 CHLOROPHENYL) 4 [[4 (4 CHLOROPHENYL) 6 (4 METHOXYPHENYL)PYRIMIDIN 2 YL]SULFAMOYL]SYDNONE; 3 (4 CHLOROPHENYL) 4 [[4 (4 FLUOROPHENYL) 6 (4 METHOXYPHENYL)PYRIMIDIN 2 YL]SULFAMOYL]SYDNONE; 3 (4 CHLOROPHENYL) 4 [[4 (4 METHOXYPHENYL) 6 (3 NITROPHENYL)PYRIMIDIN 2 YL]SULFAMOYL]SYDNONE; 3 (4 CHLOROPHENYL) 4 [[4 (4 METHOXYPHENYL) 6 (4 NITROPHENYL)PYRIMIDIN 2 YL]SULFAMOYL]SYDNONE; 3 (4 CHLOROPHENYL) 4 [[4 (4 METHOXYPHENYL) 6 PHENYLPYRIMIDIN 2 YL]SULFAMOYL]SYDNONE; 4 [(4, 6 DINITRO 1,3 BENZOTHIAZOL 2 YL)SULFAMOYL] 3 (4 CHLOROPHENYL)SYDNONE; 4 [(5 METHYL 1,3 BENZOTHIAZOL 2 YL]SULFAMOYL] 3 (4 CHLOROPHENYL)SYDNONE; 4 [(6 BROMO 1,3 BENZOTHIAZOL 2 YL)SULFAMOYL] 3 (4 CHLOROPHENYL)SYDNONE; 4 [(6 CHLORO 1,3 BENZOTHIAZOL 2 YL)SULFAMOYL] 3 (4 CHLOROPHENYL)SYDNONE; 4 [(6 FLUORO 1,3 BENZOTHIAZOL 2 YL)SULFAMOYL] 3 (4 CHLOROPHENYL)SYDNONE; 4 [(6 METHOXY 1,3 BENZOTHIAZOL 2 YL)SULFAMOYL] 3 (4 CHLOROPHENYL)SYDNONE; 4 [(6 METHYL 1,3 BENZOTHIAZOL 2 YL)SULFAMOYL] 3 (4 CHLOROPHENYL)SYDNONE; 4 [(NITRO 1,3 BENZOTHIAZOL 2 YL)SULFAMOYL] 3 (4 CHLOROPHENYL)SYDNONE; 4 [[4 (2,4 DICHLOROPHENYL) 1,3 THIAZOL 2 YL]SULFAMOYL]3 (4 CHLOROPHENYL)SYDNONE; 4 [[4 (4 BROMOPHENYL) 6 (4 PYRIMIDIN 2 YL]SULFAMOYL] 3 (4 CHLOROPHENYL)SYDNONE; 4 [[4 (4 CHLOROPHENYL) 1,3 THIAZOL 2 YL]SULFAMOYL]3 (4 CHLOROPHENYL)SYDNONE; 4 [[4 (4 FLUOROPHENYL) 1,3 THIAZOL 2 YL]SULFAMOYL]3 (4 CHLOROPHENYL)SYDNONE; 4 [[4 (4 METHOXYPHENYL) 1,3 THIAZOL 2 YL]SULFAMOYL]3 (4 CHLOROPHENYL)SYDNONE; 4 [[4 (4 METHYLPHENYL) 1,3 THIAZOL 2 YL]SULFAMOYL]3 (4 CHLOROPHENYL)SYDNONE; 4 [[4 (5 CHLORO 2,4 DIFLUOROPHENYL) 1,3 THIAZOL 2 YL]SULFAMOYL]3 (4 CHLOROPHENYL)SYDNONE; 4 [[4,6 BIS(4 METHOXYPHENYL)PYRIMIDIN 2 YL]SULFAMOYL] 3 (4 CHLOROPHENYL)SYDNONE; 4 [[6 (TRIFLUOROMETHYL) 1,3 BENZOTHIAZOL 2 YL]SULFAMOYL] 3 (4 CHLOROPHENYL)SYDNONE; BENZOTHIAZOLE DERIVATIVE; CARBONYL DERIVATIVE; CIPROFLOXACIN; PYRIMIDINE DERIVATIVE; THIAZOLE DERIVATIVE; UNCLASSIFIED DRUG;

ABSORPTION; ANTIMICROBIAL ACTIVITY; ARTICLE; BACTERIAL STRAIN; DRUG SYNTHESIS; IRRADIATION; MINIMUM INHIBITORY CONCENTRATION; NONHUMAN; PROTON NUCLEAR MAGNETIC RESONANCE;

EID: 85027927846     PISSN: 0091150X     EISSN: 15739031     Source Type: Journal    
DOI: 10.1007/s11094-012-0712-5     Document Type: Article

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