Preparation of N-aryl-5r-hydroxymethyl-2-oxazolidinones from N-aryl carbamates: N-phenyl-(5R)-hydroxymethyl-2-oxazolidinone: [2-Oxazolidinone, 5-(Hydroxymethyl)-3-phenyl-, (5R)-]

Organic Syntheses

Volumn 81, Issue , 2005, Pages 112-120

  Manninen, Peter R ^a,b   Brickner, Steven J ^c   Darwish, Ossama ^d   Miller, Marvin J ^d  

^a Medicinal Chemistry Research   (United States)

^b ELI LILLY AND COMPANY   (United States)

^c PFIZER GLOBAL RESEARCH AND DEVELOPMENT   (United States)

^d NONE

Author keywords

[No Author keywords available]

Indexed keywords

EID: 85027843197     PISSN: 00786209     EISSN: 16000730     Source Type: Book Series    
DOI: 10.15227/orgsyn.081.0112     Document Type: Article

References (7)

1. Gregory, W. A.; Brittelli, D. R.; Wang, C. L. J.; Wounola, M. A.; McRipley, R. J.; Eustice D. C.; Eberly, V. S.; Bartholomew, P. T.; Slee, A. M.; Forbes, M. J. Med. Chem. 1989, 32, 1673.
2. Herweh, J. E.; Kauffman, W. J.; Tetrahedron Lett. 1971, 12, 809.
3. Brickner, S. J.; Hutchinson, D. K.; Barbachyn, M. R.; Manninen P. R.; Ulanowicz, D. A.; Garmon, S. A.; Grega, K. C.; Hendges, S. K.; Toops, D. S.; Ford. C. W.; Zurenko, G. E. J. Med. Chem. 1996, 39, 673.
4. Manninen, P. R.; Little, H. A.; Brickner, S. J.; Division of Organic Chemistry, American Chemical Society, 212th ACS National Meeting, Orlando, FL, August, 1996.
5. Citations that have used this method: Barbachyn, M. R.; Hutchinson, D. K.; Brickner, S. J.; Cynamon, M. H.; Kilburn, J. O.; Klemens, S. P.; Glickman, E. S.; Grega, K. C.; Hendges, S. K.; Toops, D. S.; Ford. C. W.; Zurenko, G. E. J. Med. Chem. 1996, 39, 680.;
6. Genin, M. J.; Allwine, D. A.; Anderson, D. J.; Barbachyn, M. R.; Emmert, D. E.; Garmon, S. A.; Graber, D. R.; Grega, K. C.; Hester, J. B.; Hutchinson, D. K.; Morris, J.; Reischer, R. J.; Ford. C. W.; Zurenko, G. E.; Hamel, J. C.; Schaadt, R. D.; Stapert, D.; Yagi, B. H. J. Med. Chem. 2000, 43, 953.;
7. Tucker, J. A.; Allwine, D. A.; Grega, K. C.; Barbachyn, M. R.; Klock, J. L.; Adamski, J. L.; Brickner, S. J.; Hutchinson, D. K.; Ford. C. W.; Zurenko, G. E.; Conradi, R. A.; Burton, P. S.; Jensen, R. M. J. Med. Chem. 1998, 41, 3727.