Evaluation of gum mastic (Pistacia lentiscus) as a microencapsulating and matrix forming material for sustained drug release

Asian Journal of Pharmaceutical Sciences

Volumn 12, Issue 5, 2017, Pages 424-432

  Morkhade, Dinesh M ^a  

^a RTM NAGPUR UNIVERSITY   (India)

Author keywords

Diclofenac sodium; Diltiazem hydrochloride; Gum mastic; Matrix tablets; Microparticles; Sustained release

Indexed keywords

DICLOFENAC; DILTIAZEM; MASTIC; OIL;

ARTICLE; CONTROLLED STUDY; DRUG GRANULATION; EVAPORATION; MATRIX TABLET; MELTING POINT; MICROENCAPSULATION; PARTICLE SIZE; PHYSICAL CHEMISTRY; PISTACIA LENTISCUS; SUSTAINED DRUG RELEASE; WETTABILITY;

EID: 85019718869     PISSN: 18180876     EISSN: 2221285X     Source Type: Journal    
DOI: 10.1016/j.ajps.2017.05.002     Document Type: Article

References (37)

1. Bharadwaj, T.R., Kanwar, M., Lal, R., et al. Natural gums and modified gums as sustained-release carriers. Drug Dev Ind Pharm 26 (2000), 1025–1038.
2. Morkhade, D.M., Fulzele, S.V., Satturwar, P.M., et al. Gum copal and gum damar: novel matrix forming materials for sustained drug delivery. Ind J Pharm Sci 68 (2006), 53–58.
3. Morkhade, D.M., Nande, V.S., Barabde, U.V., et al. PEGylated rosin derivatives: novel microencapsulating materials for sustained drug delivery. AAPS PharmSciTech 8:2 (2007), E1–E9 Article 47.
4. Morkhade, D.M., Joshi, S.B., Evaluation of gum damar as a novel microencapsulating material for ibuprofen and diltiazem hydrochloride. Ind J Pharm Sci 69:2 (2007), 263–268.
5. Nande, V.S., Barabde, U.V., Morkhade, D.M., et al. Synthesis and characterization of PEGylated derivatives of rosin for sustained drug delivery. React Funct Polym 66:11 (2006), 1373–1383.
6. Morkhade, D.M., Nande, V.S., Barabde, U.V., et al. A comparative study of aqueous and organic-based films and coatings of PEGylated rosin derivative. Drug Dev Ind Pharm 34:1 (2008), 24–32.
7. Nande, V.S., Barabde, U.V., Morkhade, D.M., et al. Investigation of PEGylated derivatives of rosin as sustained release film formers. AAPS PharmSciTech 9:1 (2008), 105–111.
8. Rovolvy, Mastic (plant resin). Available from: https://www.revolvy.com/main/index.php?s=Mastic%20(plant%20resin)&item_type=topic, 2017 [Accessed 22 March 2017].
9. Henriette's Herbal Homepage, The British Pharmaceutical Codex 1911. Available from: http://www.henriettes-herb.com/eclectic/bpc1911/pistacia.html, 2017 [Accessed 22 March 2017].
10. Coppen, J.J.W., Gums, resins and latexes of plant origin. Available from: http://www.fao.org/3/a-v9236e.pdf, 2017 [Accessed 22 March 2017].
11. Scrubis, B., Markakis, P., Zabik, M.J., Essential oil of mastic gum. Int Flav Food Additiv 6:6 (1975), 349–356.
12. Al-Said, M.S., Ageel, A.M., Parmar, N.S., et al. Evaluation of mastic, a crude drug obtained from Pistacia lentiscus for gastric and duodenal anti-ulcer activity. J Ethnopharmacol 15:3 (1986), 271–278.
13. Marone, P., Bono, L., Leone, E., et al. Bactericidal activity of Pistacia lentiscus mastic gum against Helicobacter pylori. J Chemother 13:6 (2001), 611–614.
14. Wallis, T.E., Resins, gum-resins, oleo-resins. Wallis, T.E., (eds.) Text book of Pharmacognosy, 1985, CBS Publisher and Distributors, India, 483–572.
15. Sampson, F.J., Thin film coating for tablets and the like and method of coating. US Patent, 1964 US3149039.
16. Panagopoulou, A., Georgarakis, M., Effect of compression and diluent on drug release from mastix matrix tablets. A statistical analysis. Drug Dev Ind Pharm 16:4 (2008), 637–649.
17. Assimopoulou, A.N., Papageorgiou, V.P., Kiparissides, C., Synthesis and release studies of shikonin-containing microcapsules prepared by the solvent evaporation method. J Microencapsul 20:5 (2003), 581–596.
18. Assimopoulou, A.N., Papageorgiou, V.P., Preparation and release studies of alkannin-containing microcapsules. J Microencapsul 21:2 (2004), 161–173.
19. Georgarakis, M., Groning, R., Henzler, P., Microencapsulation of potassium chloride with mastic. Pharmazie 42:7 (1987), 455–456.
20. Nouh, A.T., Abd El-Gawad, A.H., Guda, T.K., Formulation and bioavailability of controlled release salbutamol sulphate tablets using natural additives. Drug Discov Ther 4:2 (2010), 85–92.
21. Nouh, A.T., Abd El-Gawad, A.H., Guda, T.K., Stability, bioavailability, and ulcerative activity of diclofenac sodium-mastic controlled release tablets. Drug Discov Ther 4:2 (2010), 93–99.
22. Deshpande, R.D., Gowda, D.V., Mahammed, N., Design of Pistacia lentiscus (mastic gum) controlled release spheroids and investigating the influence of roll compaction. Ind crops prod 44 (2013), 603–610.
23. Drugs.com, Diclofenac. Available at: https://www.drugs.com/pro/diclofenac.html, 2017 [Accessed 22 March 2017].
24. EMC, Diltiazem hydrochloride tablets 60 mg. Available at: http://www.medicines.org.uk/emc/medicine/23945/SPC/diltiazem%20hydrochloride%20tablets%2060 mg/, 2017 [Accessed 22 March 2017].
25. Bhatia, M.S., Deshmukh, R., Choudhari, P., et al. Chemical modification of pectins, characterization and evaluation for drug delivery. Sci Pharm 76 (2008), 775–784.
26. Costa, P., Lobo, J.M.S., Modeling and comparison of dissolution profiles. Eur J Pharm Sci 13 (2000), 123–133.
27. McGee, J.P., Singh, M., Li, X.M., et al. The encapsulation of a model protein in poly (D, L-lactide-co-glycolide) microparticles of various sizes; an evaluation of process reproducibility. J Microencapsul 14 (1997), 197–210.
28. Lin, Y.H., Vasavada, R.C., Studies on microencapsulation of 5-flurouracil with poly (ortho ester) polymers. J Microencapsul 17 (2000), 1–11.
29. Rippie, E.G., Mixing. Lachman, L., Liberman, H.A., Kanig, J., (eds.) The theory and practice of industrial pharmacy, 1990, Varghese publication house, Bombay, 3–20.
30. Yan, C., Resau, J.H., Hewetson, J., et al. Characterization and morphological analysis of protein loaded poly (lactide-co-glycolide) microparticles prepared by water-in-oil-in water emulsion technique. J Control Rel 32 (1994), 231–241.
31. Ghaderi, R., Struesson, C., Carlfors, J., Effect of preparative parameters on the characteristics of poly (D, L-lactide-co-glycolide) microspheres made by the double emulsion method. Int J Pharm 141 (1996), 205–216.
32. Narayani, R., Rao, K.P., Controlled release of anticancer drug methotrexate from biodegradable gelatin microspheres. J Microencapsul 11 (1994), 69–77.
33. Sansdrap, P., Moes, A.J., In vitro evaluation of the hydrolytic dehydration of dispersed and aggregated poly (D, L-lactide-co-glycolide) microspheres. J Control Rel 43 (1997), 47–58.
34. Bezemer, J.M., Radersma, R., Grijpma, D.W., et al. Microspheres for protein delivery prepared from amphiphilic multiblock copolymer 2. Modulation of release rate. J Control Rel 7 (2000), 249–260.
35. Janjikhel, R.K., Adeyeye, C.M., Stereospecific formulation and characterization of ibuprofen microspheres. J Microencapsul 14 (1997), 409–426.
36. Nokhodchi, A., Farid, D., Microencapsulation of paracetamol by various emulsion techniques using cellulose acetate phthalate. Pharm Tech 2 (2002), 54–60.
37. Yang, Y.Y., Chung, T.S., Bai, X.L., et al. Effect of preparation conditions on morphology and release profiles of biodegradable polymeric microspheres containing protein fabricated by double emulsion method. Chem Eng Sci 55 (2000), 2223–2236.