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Bioorganic and Medicinal Chemistry Letters

Volumn 26, Issue 8, 2016, Pages 2092-2097

Derivatization of agelastatin A leading to bioactive analogs and a trifunctional probe

(11) Jouanneau, Morgan a McClary, Brandon c Reyes, Jeremy Chris P b,f Chen, Rong d Chen, Yuling d Plunkett, William d Cheng, Xin e Milinichik, Andrew Z e Albone, Earl F e Liu, Jun O c Romo, Daniel a

a BAYLOR UNIVERSITY (United States)

b TEXAS A AND M UNIVERSITY (United States)

c JOHNS HOPKINS UNIVERSITY SCHOOL OF MEDICINE (United States)

d UNIVERSITY OF TEXAS (United States)

e Morphotek Inc (United States)

f DOW CHEMICAL COMPANY (United States)

Author keywords

Agelastatin A; Diazirine; Photoaffinity probe; Pyrrole aminoimidazole alkaloid; Structure activity relationship

Indexed keywords

AGELASTATIN A; ALKALOID; ALKALOID DERIVATIVE; ALKYNE; AMIDE; ANTINEOPLASTIC AGENT; BENZENE DERIVATIVE; PYRROLE DERIVATIVE; UNCLASSIFIED DRUG; MOLECULAR PROBE; OXAZOLIDINONE DERIVATIVE;

ACYLATION; ALKYNYLATION; ANTINEOPLASTIC ACTIVITY; ARTICLE; ARYLATION; CANCER CELL LINE; CHLORINATION; CHRONIC LYMPHATIC LEUKEMIA; DERIVATIZATION; DRUG POTENCY; DRUG SYNTHESIS; FEMALE; HELA CELL LINE; HUMAN; HUMAN CELL; IC50; METHYLATION; OSTEOSARCOMA CELL LINE; OVARIAN CANCER CELL LINE; QUANTITATIVE ANALYSIS; SQUAMOUS CELL CARCINOMA CELL LINE; STRUCTURE ACTIVITY RELATION; T-CELL LEUKEMIA CELL LINE; CELL PROLIFERATION; CHEMICAL STRUCTURE; CHEMISTRY; DOSE RESPONSE; DRUG EFFECTS; DRUG SCREENING; MOLECULAR PROBE; PHARMACOLOGY; SYNTHESIS; TUMOR CELL LINE;

ALKALOIDS; ANTINEOPLASTIC AGENTS, PHYTOGENIC; CELL LINE, TUMOR; CELL PROLIFERATION; DOSE-RESPONSE RELATIONSHIP, DRUG; DRUG SCREENING ASSAYS, ANTITUMOR; HUMANS; MOLECULAR PROBES; MOLECULAR STRUCTURE; OXAZOLIDINONES; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 84959459130 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2016.02.051 Document Type: Article

Times cited : (20)

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