Buccal films of prednisolone with enhanced bioavailability

Drug Delivery

Volumn 23, Issue 2, 2016, Pages 471-478

  Kumria, Rachna ^a   Nair, Anroop B ^b   Goomber, Garima ^c   Gupta, Sumeet ^c  

^a Swift School of Pharmacy   (India)

^b KING FAISAL UNIVERSITY   (Saudi Arabia)

^c MAHARISHI MARKANDESHWAR DEEMED TO BE UNIVERSITY   (India)

Author keywords

Buccal; drug release; mucoadhesive; permeation; pharmacokinetics; prednisolone

Indexed keywords

CARBOMER; CARBOPOL 940; EUDRAGIT; HYDROXYL GROUP; METHYLCELLULOSE; POLYMER; PREDNISOLONE; PROPANE; ACRYLIC ACID RESIN; DRUG CARRIER; DRUG DOSAGE FORM; GLUCOCORTICOID; HYDROXYPROPYLMETHYLCELLULOSE; HYPROMELLOSE 2208 (100 MPA.S); POLYMETHACRYLIC ACID DERIVATIVE; WATER;

ANIMAL EXPERIMENT; ANIMAL TISSUE; AREA UNDER THE CURVE; ARTICLE; CHEEK MUCOSA; CONTROLLED DRUG RELEASE; CONTROLLED STUDY; DRUG ABSORPTION; DRUG BIOAVAILABILITY; DRUG DELIVERY SYSTEM; DRUG FORMULATION; DRUG PENETRATION; DRUG SOLUBILITY; HUMAN; HUMAN EXPERIMENT; HYDRATION; MALE; MAXIMUM PLASMA CONCENTRATION; MUCOADHESION; MUCOADHESIVE STRENGTH; NONHUMAN; NORMAL HUMAN; PH; PIG; PRIORITY JOURNAL; QUALITY CONTROL; RAT; STEADY STATE; STRENGTH; SWELLING BEHAVIOR; VISCOSITY; ADHESION; ANIMAL; BIOAVAILABILITY; BUCCAL DRUG ADMINISTRATION; CHEMISTRY; COMPARATIVE STUDY; DRUG DOSAGE FORM; FEASIBILITY STUDY; GASTROINTESTINAL ABSORPTION; METABOLISM; MOUTH MUCOSA; ORAL DRUG ADMINISTRATION; PERMEABILITY; PHARMACEUTICS; PROCEDURES; SOLUBILITY; SPRAGUE DAWLEY RAT;

ACRYLIC RESINS; ADHESIVENESS; ADMINISTRATION, BUCCAL; ADMINISTRATION, ORAL; ANIMALS; BIOLOGICAL AVAILABILITY; DOSAGE FORMS; DRUG CARRIERS; DRUG COMPOUNDING; FEASIBILITY STUDIES; GLUCOCORTICOIDS; HYPROMELLOSE DERIVATIVES; MALE; MOUTH MUCOSA; ORAL MUCOSAL ABSORPTION; PERMEABILITY; POLYMETHACRYLIC ACIDS; PREDNISOLONE; RATS, SPRAGUE-DAWLEY; SOLUBILITY; SWINE; TECHNOLOGY, PHARMACEUTICAL; WATER;

EID: 84954357831     PISSN: 10717544     EISSN: 15210464     Source Type: Journal    
DOI: 10.3109/10717544.2014.920058     Document Type: Article

References (30)

1. Adhikari SN, Nayak BS, Nayak AK, Mohanty B. (2010). Formulation and evaluation of buccal patches for delivery of atenolol. AAPS PharmSciTech 11: 1038-44
2. Bergrem H, Grøttum P, Rugstad HE. (1983). Pharmacokinetics and protein binding of prednisolone after oral and intravenous administration. Eur J ClinPharmacol 24: 415-19
3. Boateng JS, Matthews KH, Auffret AD, et al. (2009). In vitro drug release studies of polymeric freeze-dried wafers and solvent-cast films using paracetamol as a model soluble drug. Int J Pharm 378: 66-72
4. Di Colo G, Baggiani A, Zambito Y, et al. (2006). A new hydrogel for the extended and complete prednisolone release in the GI tract. Int J Pharm 310: 154-61
5. Disanto AR, Desante KA. (1975). Bioavailability and pharmacokinetics of prednisone in humans. J Pharm Sci 64: 109-12
6. Dixit RP, Puthli SP. (2009). Oral strip technology: overview and future potential. J Control Release 139: 94-107
7. Giovino C, Ayensu I, Tetteh J, Boateng JS. (2013). An integrated buccal system combining chitosan films impregnated with peptide loaded PEG-b-PLA nanoparticles. Colloids Surf B Biointerfaces 112: 9-15
8. Jones E, Ojewole E, Pillay V, et al. (2013). Monolayeredmultipolymeric buccal films with drug and polymers of opposing solubilities for ARV therapy: physico-mechanical evaluation and molecular mechanics modelling. Int J Pharm 455: 197-212
9. Kamath KR, Park K. (1994). Surface modification of polymeric biomaterials by albumin grafting using h-irradiation. J Appl Biomater 5: 163-73
10. Kumria R, Gupta V, Bansal S, et al. (2013). Oral buccoadhesive films of ondansetron: development and evaluation. Int J Pharm Investig 3: 112-8
11. Kumria R, Nair AB, Al-Dhubiab BE. (2014). Loratidine buccal films for allergic rhinitis: development and evaluation. Drug Dev Ind Pharm 40: 625-31
12. Lobatto ME, Fayad ZA, Silvera S, et al. (2010). Multimodal clinical imaging to longitudinally assess a nanomedical anti-inflammatory treatment in experimental atherosclerosis. Mol Pharm 7: 2020-9
13. Meher JG, Tarai M, Yadav NP, et al. (2013). Development and characterization of cellulose-polymethacrylate mucoadhesive film for buccal delivery of carvedilol. Carbohydr Polym 96: 172-80
14. Metselaar JM, Wauben MH, Wagenaar-Hilbers JP, et al. (2003). Complete remission of experimental arthritis by joint targeting of glucocorticoids with long-circulating liposomes. Arthritis Rheum 48: 2059-66
15. Mohammadi-Samani S, Bahri-Najafi R, Yousefi G. (2005). Formulation and in vitro evaluation of prednisolone buccoadhesive tablets. Farmaco 60: 339-44
16. Morales JO, McConville JT. (2011). Manufacture and characterization of mucoadhesive buccal films. Eur J Pharm Biopharm 77: 187-99
17. Nair A, Gupta R, Vasanti S. (2007). In vitro controlled release of alfuzosin hydrochloride using HPMC-based matrix tablets and its comparison with marketed product. Pharm Dev Technol 12: 621-5
18. Nair A, Reddy C, Jacob S. (2009). Delivery of a classical antihypertensive agent through the skin by chemical enhancers and iontophoresis. Skin Res Technol 15: 187-94
19. Nair AB, Kumria R, Harsha S, et al. (2013). In vitro techniques to evaluate buccal films. J Control Release 166: 10-21
20. Nishimura M, Matsuura K, Tsukioka T, et al. (2009). In vitro and in vivo characteristics of prochlorperazine oral disintegrating film. Int J Pharm 368: 98-102
21. Okamoto H, Taguchi H, Iida K, Danjo K. (2001). Development of polymer film dosage forms of lidocaine for buccal administration. I. Penetration rate and release rate. J Control Release 77: 253-60
22. Park HS, Lee JY, Cho SH, et al. (2002). Colon delivery of prednisolone based on chitosan coated polysaccharide tablets. Arch Pharm Res 25: 964-8
23. Patel VF, Liu F, Brown MB. (2011). Advances in oral transmucosal drug delivery. J Control Release 153: 106-16
24. Perioli L, Ambrogi V, Angelici F, et al. (2004). Development of mucoadhesive patches for buccal administration of ibuprofen. J Control Release 99: 73-82
25. Ritthidej GC, Phaechamud T, Koizumi T. (2002). Moist heat treatment on physicochemical change of chitosan salt films. Int J Pharm 232: 11-22
26. Satishbabu BK, Srinivasan BP. (2008). Preparation and evaluation of bucoadhesive films of atenolol. Indian J Pharm Sci 70: 175-9
27. Semalty M, Semalty A, Kumar G. (2008). Formulation and characterization of mucoadhesive buccal films of glipizide. Indian J Pharm Sci 70: 43-8
28. Shimoda H, Taniguchi K, Nishimura M, et al. (2009). Preparation of a fast dissolving oral thin film containing dexamethasone: a possible application to antiemesis during cancer chemotherapy. Eur J Pharm Biopharm 73: 361-5
29. Wong CF, Yuen KH, Peh KK. (1999). Formulation and evaluation of controlled release Eudragit buccal patches. Int J Pharm 178: 11-22
30. Yehia SA, El-Gazayerly ON, Basalious EB. (2009). Fluconazole mucoadhesive buccal films: in vitro/in vivo performance. Curr Drug Deliv 6: 17-27