Allosteric regulation of G protein-coupled receptor activity by phospholipids

Nature Chemical Biology

Volumn 12, Issue 1, 2016, Pages 35-39

  Dawaliby, Rosie ^a   Trubbia, Cataldo ^a   Delporte, Cédric ^a   Masureel, Matthieu ^b   Van Antwerpen, Pierre ^a   Kobilka, Brian K ^b   Govaerts, Cédric ^a  

^a UNIVERSITÉ LIBRE DE BRUXELLES   (Belgium)

^b STANFORD UNIVERSITY SCHOOL OF MEDICINE   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

BETA 2 ADRENERGIC RECEPTOR; G PROTEIN COUPLED RECEPTOR; GUANINE NUCLEOTIDE BINDING PROTEIN; HIGH DENSITY LIPOPROTEIN; ISOPRENALINE; PHOSPHATIDYLCHOLINE; PHOSPHATIDYLETHANOLAMINE; PHOSPHATIDYLGLYCEROL; PHOSPHATIDYLINOSITOL; PHOSPHATIDYLSERINE; PHOSPHOLIPID; BETA 2 ADRENERGIC RECEPTOR BLOCKING AGENT; BETA 2 ADRENERGIC RECEPTOR STIMULATING AGENT; LIPID BILAYER;

ALLOSTERISM; ARTICLE; BINDING AFFINITY; CONTROLLED STUDY; HEK293 CELL LINE; HUMAN; HUMAN CELL; IC50; LIGAND BINDING; LIPID COMPOSITION; LIPID MEMBRANE; PRIORITY JOURNAL; PROTEIN CONFORMATION; PROTEIN LIPID INTERACTION; ANIMAL; CELL MEMBRANE; CHEMISTRY; GENETICS; LIPID BILAYER; METABOLISM; SPECTROFLUOROMETRY; SPODOPTERA;

ADRENERGIC BETA-2 RECEPTOR AGONISTS; ADRENERGIC BETA-2 RECEPTOR ANTAGONISTS; ALLOSTERIC REGULATION; ANIMALS; CELL MEMBRANE; HUMANS; LIPID BILAYERS; PHOSPHOLIPIDS; RECEPTORS, ADRENERGIC, BETA-2; RECEPTORS, G-PROTEIN-COUPLED; SPECTROMETRY, FLUORESCENCE; SPODOPTERA;

EID: 84951907601     PISSN: 15524450     EISSN: 15524469     Source Type: Journal    
DOI: 10.1038/nchembio.1960     Document Type: Article

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