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Volumn 6, Issue 6, 2015, Pages 1024-1029

Discovery of a series of 2-(pyridinyl)pyrimidines as potent antagonists of GPR40

(18) Waring, Michael J a Baker, David J a Bennett, Stuart N L a Dossetter, Alexander G a Fenwick, Mark a Garcia, Rob a Georgsson, Jennie a Groombridge, Sam D a Loxham, Susan a MacFaul, Philip A a Maskill, Katie G a Morgan, David a Morrell, Jenny a Pointon, Helen a Robb, Graeme R a Smith, David M a Stokes, Stephen a Wilkinson, Gary a

a ASTRAZENECA (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

2 (PYRIDINYL)PYRIMIDINE DERIVATIVE; ANTIDIABETIC AGENT; G PROTEIN COUPLED RECEPTOR 40; G PROTEIN COUPLED RECEPTOR 40 AGONIST; INSULIN; RECEPTOR BLOCKING AGENT; UNCLASSIFIED DRUG;

ARTICLE; DRUG MECHANISM; DRUG POTENCY; DRUG RECEPTOR BINDING; DRUG RESEARCH; DRUG SCREENING; DRUG STRUCTURE; DRUG SYNTHESIS; HUMAN; IN VIVO STUDY; INSULIN RELEASE; LIPOPHILICITY; NON INSULIN DEPENDENT DIABETES MELLITUS; NONHUMAN; PHYSICAL CHEMISTRY; PRIORITY JOURNAL; RECEPTOR BLOCKING; STRUCTURE ACTIVITY RELATION;

EID: 84935859525 PISSN: 20402503 EISSN: 20402511 Source Type: Journal
DOI: 10.1039/c5md00037h Document Type: Article

Times cited : (13)

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