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Chemical Communications

Volumn 51, Issue 56, 2015, Pages 11174-11177

A systematic approach to diverse, lead-like scaffolds from α,α-disubstituted amino acids

(5) Foley, Daniel J a Doveston, Richard G a Churcher, Ian b Nelson, Adam a Marsden, Stephen P a

a UNIVERSITY OF LEEDS (United Kingdom)

b GLAXOSMITHKLINE (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

ALKENE DERIVATIVE; ALLYL COMPOUND; AMINE; AMINO ACID DERIVATIVE; CARBOXYLIC ACID; HYDANTOIN DERIVATIVE; INDOLIZIDINE DERIVATIVE; LACTAM DERIVATIVE; LEAD; MOLECULAR SCAFFOLD; NUCLEOPHILE; PIPERAZINEDIONE; AMINO ACID; AZABICYCLO DERIVATIVE; AZEPINE DERIVATIVE; PYRIDINE DERIVATIVE;

ALKYLATION; ALLYLATION; ARTICLE; CHEMICAL PARAMETERS; CHEMICAL REACTION; CHEMICAL STRUCTURE; CYCLIZATION; DRUG DEVELOPMENT; LIPOPHILICITY; MOLECULAR LIBRARY; MOLECULAR SIZE; NUCLEOPHILICITY; SYNTHESIS; CHEMISTRY;

AMINO ACIDS; AZABICYCLO COMPOUNDS; AZEPINES; MOLECULAR STRUCTURE; PYRIDINES;

EID: 84933566830 PISSN: 13597345 EISSN: 1364548X Source Type: Journal
DOI: 10.1039/c5cc03002a Document Type: Article

Times cited : (55)

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