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Volumn 58, Issue 3, 2015, Pages 1281-1297

Fragment-based drug discovery of 2-thiazolidinones as BRD4 inhibitors: 2. Structure-based optimization

Author keywords

[No Author keywords available]

Indexed keywords

1 (3 BROMO 4 METHYL 5 NITROPHENYL)ETHANONE; 2 AMINO N CYCLOPENTYL 5 (2 OXO 2,3 DIHYDROTHIAZOL 4 YL)BENZENESULFONAMIDE; 2 CHLORO N CYCLOPENTYL 5 (2 OXO 2,3 DIHYDROTHIAZOL 4 YL)BENZENESULFONAMIDE; 3 (2 BROMOACETYL) N CYCLOPENTYLBENZENESULFONAMIDE; 3 (2 OXO 2,3 DIHYDROTHIAZOL 4 YL) N (TETRAHYDROFURAN 3 YL)BENZENESULFONAMIDE; 3 (2 OXO 2,3 DIHYDROTHIAZOL 4 YL) N [(TETRAHYDROFURAN 2 YL)METHYL]BENZENESULFONAMIDE; 3 (2 OXO 2,3 DIHYDROTHIAZOL 4 YL) N [2 (THIOPHEN 2 YL)ETHYL]BENZENESULFONAMIDE; 5 (2 BROMOACETYL) N CYCLOPENTYL 2 METHYLBENZENESULFONAMIDE; 5 (2 BROMOACETYL) N CYCLOPENTYL 2 NITROBENZENESULFONAMIDE; 5 ACETYL 2 METHYLBENZENE 1 SULFONYL CHLORIDE; 5 ACETYL 2 NITROBENZENE 1 SULFONYL CHLORIDE; 5 ACETYL N CYCLOPENTYL 2 METHYLBENZENESULFONAMIDE; 5 ACETYL N CYCLOPENTYL 2 NITROBENZENESULFONAMIDE; ANTINEOPLASTIC AGENT; BENZENESULFONAMIDE DERIVATIVE; BROMODOMAIN INHIBITOR; MYC PROTEIN; N (4 AMINOPHENYL) 3 (2 OXO 2,3 DIHYDROTHIAZOL 4 YL) BENZENESULFONAMIDE; N (4 METHOXYPHENYL) 3 (2 OXO 2,3 DIHYDROTHIAZOL 4 YL)BENZENESULFONAMIDE; N (5 ACETYL 2 NITROPHENYL)ACETAMIDE; N (ISOXAZOL 3 YL) 3 (2 OXO 2,3 DIHYDROTHIAZOL 4 YL) BENZENESULFONAMIDE; N BENZYL 3 (2 OXO 2,3 DIHYDROTHIAZOL 4 YL)BENZENESULFONAMIDE; N CYCLOHEXYL 3 (2 OXO 2,3 DIHYDROTHIAZOL 4 YL) BENZENESULFONAMIDE; N CYCLOPENTYL 2 FLUORO 5 (2 OXO 2,3 DIHYDROTHIAZOL 4 YL)BENZENESULFONAMIDE; N CYCLOPENTYL 2 METHOXY 5 (2 OXO 2,3 DIHYDROTHIAZOL 4 YL)BENZENESULFONAMIDE; N CYCLOPENTYL 2 METHYL 5 (2 OXO 2,3 DIHYDROTHIAZOL 4 YL)BENZENESULFONAMIDE; N CYCLOPENTYL 2 NITRO 5 (2 OXO 2,3 DIHYDROTHIAZOL 4 YL)BENZENESULFONAMIDE; N CYCLOPENTYL 3 (2 OXO 2,3 DIHYDROTHIAZOL 4 YL) BENZENESULFONAMIDE; N CYCLOPROPYL 3 (2 OXO 2,3 DIHYDROTHIAZOL 4 YL)BENZENESULFONAMIDE; UNCLASSIFIED DRUG; UNINDEXED DRUG; BRD4 PROTEIN, HUMAN; NUCLEAR PROTEIN; THIAZOLIDINE DERIVATIVE; TRANSCRIPTION FACTOR;

EID: 84922822753     PISSN: 00222623     EISSN: 15204804     Source Type: Journal    
DOI: 10.1021/jm501504k     Document Type: Article
Times cited : (49)

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* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.