New class of methyl tetrazole based hybrid of (Z)-5-benzylidene-2- (piperazin-1-yl)thiazol-4(%H)-one as potent antitubercular agents

Bioorganic and Medicinal Chemistry Letters

Volumn 24, Issue 17, 2014, Pages 4166-4170

  Chauhan, Kuldeep ^a   Sharma, Moni ^a   Trivedi, Priyanka ^a   Chaturvedi, Vinita ^a   Chauhan, Prem M S ^a  

^a CENTRAL DRUG RESEARCH INSTITUTE   (India)

Author keywords

Cytotoxicity; Mycobacterium tuberculosis; Rhodanine; Tetrazole

Indexed keywords

ETHAMBUTOL; ISONIAZID; PIPERAZINE DERIVATIVE; PYRAZINAMIDE; RHODANINE; TETRAZOLE DERIVATIVE; THIAZOLONE PIPERAZINE TETRAZOLE DERIVATIVE; TUBERCULOSTATIC AGENT; UNCLASSIFIED DRUG; THIAZOLE DERIVATIVE;

ANIMAL CELL; ANTIBACTERIAL ACTIVITY; ARTICLE; BONE MARROW DERIVED MACROPHAGE; CONTROLLED STUDY; CYTOTOXICITY; DRUG POTENCY; DRUG SYNTHESIS; IN VITRO STUDY; MINIMUM INHIBITORY CONCENTRATION; MOUSE; MYCOBACTERIUM TUBERCULOSIS; NONHUMAN; STRUCTURE ACTIVITY RELATION; VERO CELL LINE; ANIMAL; CHEMICAL STRUCTURE; CHEMISTRY; CHLOROCEBUS AETHIOPS; CLASSIFICATION; DOSE RESPONSE; DRUG EFFECTS; MICROBIAL SENSITIVITY TEST; SYNTHESIS;

MYCOBACTERIUM TUBERCULOSIS;

ANIMALS; ANTITUBERCULAR AGENTS; CERCOPITHECUS AETHIOPS; DOSE-RESPONSE RELATIONSHIP, DRUG; MICROBIAL SENSITIVITY TESTS; MOLECULAR STRUCTURE; MYCOBACTERIUM TUBERCULOSIS; STRUCTURE-ACTIVITY RELATIONSHIP; TETRAZOLES; THIAZOLES; VERO CELLS;

EID: 84906935718     PISSN: 0960894X     EISSN: 14643405     Source Type: Journal    
DOI: 10.1016/j.bmcl.2014.07.061     Document Type: Article

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