메뉴 건너뛰기




Volumn 34, Issue 4, 2014, Pages 1737-1742

Multidrug resistance reversing activity of newly developed phenothiazines on P-glycoprotein (ABCB1)-related resistance of mouse T-lymphoma cells

Author keywords

ABCB1; ATP binding cassette protein B1; Ethidium bromide; Mouse T lymphoma cell lines; Multidrug resistance; P glycoprotein; Phenothiazines; Rhodamine 123; Thioridazine; Verapamil

Indexed keywords

ETHIDIUM BROMIDE; PHENOTHIAZINE DERIVATIVE; RHODAMINE 123; THIORIDAZINE; VERAPAMIL; ANTINEOPLASTIC AGENT; MULTIDRUG RESISTANCE PROTEIN; PHENOTHIAZINE;

EID: 84902265726     PISSN: 02507005     EISSN: 17917530     Source Type: Journal    
DOI: None     Document Type: Article
Times cited : (16)

References (20)
  • 1
    • 0030801767 scopus 로고    scopus 로고
    • The potential management of resistant infections with non-antibiotics
    • Kristiansen JE and Amaral L: The potential management of resistant infections with non-antibiotics. J Antimicrob Chemother 40: 319-327, 1997.
    • (1997) J Antimicrob Chemother , vol.40 , pp. 319-327
    • Kristiansen, J.E.1    Amaral, L.2
  • 3
    • 0026525237 scopus 로고
    • Antiplasmid activity of phenothiazines, benzo[a]phenothiazines and benz[c]acridines
    • Motohashi N, Sakagami H, Kurihara T, Csuri K and Molnar J: Antiplasmid activity of phenothiazines, benzo[a]phenothiazines and benz[c]acridines. Anticancer Res 12(1): 135-139, 1992.
    • (1992) Anticancer Res , vol.12 , Issue.1 , pp. 135-139
    • Motohashi, N.1    Sakagami, H.2    Kurihara, T.3    Csuri, K.4    Molnar, J.5
  • 7
    • 79958257266 scopus 로고    scopus 로고
    • Recent progress in biological activities of synthesized phenothiazines
    • Pluta K, Morak-Mlodawska B and Jeleñ M: Recent progress in biological activities of synthesized phenothiazines. Eur J Med Chem 46(8): 3179-3189, 2011.
    • (2011) Eur J Med Chem , vol.46 , Issue.8 , pp. 3179-3189
    • Pluta, K.1    Morak-Mlodawska, B.2    Jeleñ, M.3
  • 8
    • 79851507774 scopus 로고    scopus 로고
    • Phenothiazine: The seven lives of pharmacology's first lead structure
    • Ohlow MJ and Moosmann B: Phenothiazine: The seven lives of pharmacology's first lead structure. Drug Discov Today 16(3-4): 119-131, 2011.
    • (2011) Drug Discov Today , vol.16 , Issue.3-4 , pp. 119-131
    • Ohlow, M.J.1    Moosmann, B.2
  • 9
    • 79960639569 scopus 로고    scopus 로고
    • Evaluation of 40 new phenothiazine derivatives for activity against intrinsic efflux pump systems of reference Escherichia coli, Salmonella Enteritidis, Enterococcus faecalis and Staphylococcus aureus strains
    • Takács D, Cerca P, Martins A, Riedl Z, Hajós G, Molnár J, Viveiros M, Couto I and Amaral L: Evaluation of 40 new phenothiazine derivatives for activity against intrinsic efflux pump systems of reference Escherichia coli, Salmonella Enteritidis, Enterococcus faecalis and Staphylococcus aureus strains. In Vivo 25(5): 719-724, 2011.
    • (2011) In Vivo , vol.25 , Issue.5 , pp. 719-724
    • Takács, D.1    Cerca, P.2    Martins, A.3    Riedl, Z.4    Hajós, G.5    Molnár, J.6    Viveiros, M.7    Couto, I.8    Amaral, L.9
  • 10
    • 73949118463 scopus 로고    scopus 로고
    • Reversing agents for ATP-binding cassette drug transporters
    • Lee CH: Reversing agents for ATP-binding cassette drug transporters. Methods Mol Biol 596: 325-340, 2010.
    • (2010) Methods Mol Biol , vol.596 , pp. 325-340
    • Lee, C.H.1
  • 12
    • 84878579770 scopus 로고    scopus 로고
    • Synthesis and pharmacological investigation of new 2-amino-N -hydroxyalkylphenothiazines exhibiting marked MDR-inhibitory effect
    • Takács D, Bombicz P, Egyed O, Drahos L, Jemnitz K, Visy J, Molnár J, Riedl Z and Hajós G: Synthesis and pharmacological investigation of new 2-amino-N -hydroxyalkylphenothiazines exhibiting marked MDR-inhibitory effect. Bioorg Med Chem 21: 3760-3779, 2013.
    • (2013) Bioorg Med Chem , vol.21 , pp. 3760-3779
    • Takács, D.1    Bombicz, P.2    Egyed, O.3    Drahos, L.4    Jemnitz, K.5    Visy, J.6    Molnár, J.7    Riedl, Z.8    Hajós, G.9
  • 14
    • 0013508682 scopus 로고
    • A retrovirus carrying an MDR1 cDNA confers multidrug resistance and polarized expression of P-glycoprotein in MDCK cells
    • Pastan I, Gottesman, MM, Ueda K, Lovelace E, Rutherford AV and Willingham MC: A retrovirus carrying an MDR1 cDNA confers multidrug resistance and polarized expression of P-glycoprotein in MDCK cells. Proc Natl Acad Sci USA 85: 4486-4490, 1988.
    • (1988) Proc Natl Acad Sci USA , vol.85 , pp. 4486-4490
    • Pastan, I.1    Gottesman, M.M.2    Ueda, K.3    Lovelace, E.4    Rutherford, A.V.5    Willingham, M.C.6
  • 15
    • 0025861828 scopus 로고
    • Multidrug resistance after retroviral transfer of the human MDR1 gene correlates with P-glycoprotein density in the plasma membrane and is not affected by cytotoxic selection
    • Choi K, Frommel TO, Stern RK, Perez CF, Kriegler M, Tsuruo T and Roninson IB: Multidrug resistance after retroviral transfer of the human MDR1 gene correlates with P-glycoprotein density in the plasma membrane and is not affected by cytotoxic selection. Proc Natl Acad Sci USA 88: 7386-7390, 1991.
    • (1991) Proc Natl Acad Sci USA , vol.88 , pp. 7386-7390
    • Choi, K.1    Frommel, T.O.2    Stern, R.K.3    Perez, C.F.4    Kriegler, M.5    Tsuruo, T.6    Roninson, I.B.7
  • 16
    • 32144459525 scopus 로고    scopus 로고
    • Reversal of multidrug resistance of cancer cells in vitro: Modification of drug resistance by selected carotenoids
    • Gyemant N, Tanaka M, Molnar P, Deli J, Mandoky L and Molnar J: Reversal of multidrug resistance of cancer cells in vitro: modification of drug resistance by selected carotenoids. Anticancer Res 26: 367-374, 2006.
    • (2006) Anticancer Res , vol.26 , pp. 367-374
    • Gyemant, N.1    Tanaka, M.2    Molnar, P.3    Deli, J.4    Mandoky, L.5    Molnar, J.6
  • 17
    • 0030035535 scopus 로고    scopus 로고
    • Effects of steroids and verapamil on P-glycoprotein ATPase activity: Progesterone, desoxycorticosterone, corticosterone and verapamil are mutually non-exclusive modulators
    • Orlowski S, Mir LM, Belehradek J Jr. and Garrigos M: Effects of steroids and verapamil on P-glycoprotein ATPase activity: Progesterone, desoxycorticosterone, corticosterone and verapamil are mutually non-exclusive modulators. Biochem J 317(Pt 2): 515-522, 1996.
    • (1996) Biochem J , vol.317 , pp. 515-522
    • Orlowski, S.1    Mir, L.M.2    Belehradek, J.3    Garrigos, M.4
  • 19
    • 0031922586 scopus 로고    scopus 로고
    • The primary in vitro anticancer activity of 'half-mustard type' phenothiazines in NCI's revised anticancer screening paradigm
    • Wuonola MA, Palfreyman MG, Motohashi N, Kawase M, Gabay S, Gupta RR and Molnár J: The primary in vitro anticancer activity of 'half-mustard type' phenothiazines in NCI's revised anticancer screening paradigm. Anticancer Res 18: 337-348, 1998.
    • (1998) Anticancer Res , vol.18 , pp. 337-348
    • Wuonola, M.A.1    Palfreyman, M.G.2    Motohashi, N.3    Kawase, M.4    Gabay, S.5    Gupta, R.R.6    Molnár, J.7
  • 20
    • 44849117020 scopus 로고    scopus 로고
    • Multidrug resistance reverting activity and antitumor profile of new phenothiazine derivatives
    • Bisi A, Meli M, Gobbi S, Rampa A, Tolomeo M and Dusonchet L: Multidrug resistance reverting activity and antitumor profile of new phenothiazine derivatives. Bioorg Med Chem 16: 6474-6482, 2008.
    • (2008) Bioorg Med Chem , vol.16 , pp. 6474-6482
    • Bisi, A.1    Meli, M.2    Gobbi, S.3    Rampa, A.4    Tolomeo, M.5    Dusonchet, L.6


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.