Effect of operating parameters on PVP/tadalafil solid dispersions prepared using supercritical anti-solvent process

Journal of Supercritical Fluids

Volumn 90, Issue , 2014, Pages 126-133

  Park, Junsung ^a,b   Cho, Wonkyung ^a,b   Kang, Han ^a   Lee, Benjamin Byung Jun ^a   Kim, Taek Sun ^a   Hwang, Sung Joo ^a  

^a Yonsei University   (South Korea)

^b Chungnam National University   (South Korea)

Author keywords

Box Behnken design; Operation parameter; Solid dispersion; Supercritical anti solvent process; Tadalafil

Indexed keywords

CRYSTALLINITY; DISPERSIONS; DISSOLUTION; SOLVENTS;

BOX-BEHNKEN DESIGN; OPERATION PARAMETERS; SOLID DISPERSION; SUPERCRITICAL ANTISOLVENTS; TADALAFIL;

PARTICLE SIZE;

EID: 84899649687     PISSN: 08968446     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.supflu.2014.04.001     Document Type: Article

References (25)

1. S. Singh, B. Prasad, A.A. Savaliya, R.P. Shah, V.M. Gohil, and A. Kaur Strategies for characterizing sildenafil, vardenafil, tadalafil and their analogues in herbal dietary supplements, and detecting counterfeit products containing these drugs Trends in Analytical Chemistry 28 2009 13 28
2. S. Stegemann, F. Leveiller, D. Franchi, H. de Jong, and H. Lindén When poor solubility becomes an issue: from early stage to proof of concept European Journal of Pharmaceutical Sciences 31 2007 249 261 (Pubitemid 47079001)
3. A.T.M. Serajuddin Solid dispersion of poorly water-soluble drugs: early promises, subsequent problems, and recent breakthroughs Journal of Pharmaceutical Sciences 88 1999 1058 1066
4. C. Leuner, and J. Dressman Improving drug solubility for oral delivery using solid dispersions European Journal of Pharmaceutics and Biopharmaceutics 50 2000 47 60 (Pubitemid 30326688)
5. S. Keiji, and O. Noboru Studies on absorption of eutectic mixture. I: A comparison of the behavior of eutectic mixture of sulfathiazole and that of ordinary sulfathiazole in man Chemical and Pharmaceutical Bulletin 9 1961 866 872
6. T. Tachibana, and A. Nakamura A methode for preparing an aqueous colloidal dispersion of organic materials by using water-soluble polymers: dispersion of β-carotene by polyvinylpyrrolidone Kolloid-Zeitschrift & Zeitschrift für Polymere 203 1965 130 133
7. M.M. Mehanna, A.M. Motawaa, and M.W. Samaha In sight into tadalafil - block copolymer binary solid dispersion: mechanistic investigation of dissolution enhancement International Journal of Pharmaceutics 402 2010 78 88
8. N. Midoux, P. Hošek, L. Pailleres, and J.R. Authelin Micronization of pharmaceutical substances in a spiral jet mill Powder Technology 104 1999 113 120 (Pubitemid 29397414)
9. M. Stievano, and N. Elvassore High-pressure density and vapor-liquid equilibrium for the binary systems carbon dioxide-ethanol, carbon dioxide-acetone and carbon dioxide-dichloromethane Journal of Supercritical Fluids 33 2005 7 14
10. C.J. Chang, C.-Y. Day, C.-M. Ko, and K.-L. Chiu Densities and P-x-y diagrams for carbon dioxide dissolution in methanol, ethanol, and acetone mixtures Fluid Phase Equilibria 131 1997 243 258 (Pubitemid 127421447)
11. R. Tuunila, and L. Nyström Effects of grinding parameters on product fineness in jet mill grinding Minerals Engineering 11 1998 1089 1094 (Pubitemid 128398269)
12. D.H. Won, M.S. Kim, S. Lee, J.S. Park, and S.J. Hwang Improved physicochemical characteristics of felodipine solid dispersion particles by supercritical anti-solvent precipitation process International Journal of Pharmaceutics 301 2005 199 208 (Pubitemid 41206604)
13. J. Park, W. Cho, K.H. Cha, J. Ahn, K. Han, and S.J. Hwang Solubilization of the poorly-water soluble drug, telmisartan, using supercritical anti-solvent (SAS) process International Journal of Pharmaceutics 441 2012 50 55
14. E. Reverchon Supercritical antisolvent precipitation of micro- and nano-particles Journal of Supercritical Fluids 15 1999 1 21 (Pubitemid 129671809)
15. E. Reverchon, and G. Della Porta Production of antibiotic micro- and nano-particles by supercritical antisolvent precipitation Powder Technology 106 1999 23 29 (Pubitemid 30011996)
16. E. Reverchon, I. De Marco, and E. Torino Nanoparticles production by supercritical antisolvent precipitation: a general interpretation Journal of Supercritical Fluids 43 2007 126 138 (Pubitemid 47385121)
17. J.-S. Kim, M.-S. Kim, H.J. Park, S.-J. Jin, S. Lee, and S.-J. Hwang Physicochemical properties and oral bioavailability of amorphous atorvastatin hemi-calcium using spray-drying and SAS process International Journal of Pharmaceutics 359 2008 211 219
18. J. Park, H.J. Park, W. Cho, K.H. Cha, Y.S. Kang, and S.J. Hwang Preparation and pharmaceutical characterization of amorphous cefdinir using spray-drying and SAS-process International Journal of Pharmaceutics 396 2010 239 245
19. M.S. Kim, S.J. Jin, J.S. Kim, H.J. Park, H.S. Song, R.H.H. Neubert, and S.J. Hwang Preparation, characterization and in vivo evaluation of amorphous atorvastatin calcium nanoparticles using supercritical antisolvent (SAS) process European Journal of Pharmacokinetics and Biopharmaceutics 69 2008 454 465
20. E. Reverchon, I. De Marco, and G. Della Porta Tailoring of nano- and micro-particles of some superconductor precursors by supercritical antisolvent precipitation Journal of Supercritical Fluids 23 2002 81 87
21. E. Reverchon, I. De Marco, and G. Della Porta Rifampicin microparticles production by supercritical antisolvent precipitation International Journal of Pharmaceutics 243 2002 83 91
22. M.-S. Kim, S. Lee, J.-S. Park, J.-S. Woo, and S.-J. Hwang Micronization of cilostazol using supercritical antisolvent (SAS) process: effect of process parameters Powder Technology 177 2007 64 70 (Pubitemid 47224964)
23. B. Ma, X. Shang, Q. Zhang, J. Li, Y. Liu, X. Cao, and Q. Xu Rapid analysis of tadalafil in human blood plasma and seminal plasma by liquid chromatography/tandem mass spectrometry Journal of Pharmaceutical and Biomedical Analysis 77 2013 149 157
24. A.K. Jasuja Airblast atomization of alternative liquid petroleum fuels under high pressure conditions Journal of Engineering Power 103 1981 514 518 (Pubitemid 12439658)
25. M. Rantakylä, M. Jäntti, O. Aaltonen, and M. Hurme The effect of initial drop size on particle size in the supercritical antisolvent precipitation (SAS) technique Journal of Supercritical Fluids 24 2002 251 263