Route design and development of a MET kinase inhibitor: A copper-catalyzed preparation of an N 1 - Methylindazole

Organic Process Research and Development

Volumn 18, Issue 4, 2014, Pages 501-510

  Kallman, Neil J ^a   Liu, Chin ^a   Yates, Matthew H ^a   Linder, Ryan J ^a   Ruble, J Craig ^a   Kogut, Eugene F ^a   Patterson, Lawrence E ^a   Laird, Dana L T ^a   Hansen, Marvin M ^a  

^a ELI LILLY AND COMPANY   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

CATALYSIS; ENZYME INHIBITION;

ARYL BROMIDES; DEPROTECTION; DESIGN AND DEVELOPMENT; DRUG CANDIDATES; KINASE INHIBITORS; PROCESS CHEMISTRY; ROUTE DESIGN; SUZUKI CROSS COUPLING;

CYCLIZATION;

EID: 84898994044     PISSN: 10836160     EISSN: 1520586X     Source Type: Journal    
DOI: 10.1021/op400317z     Document Type: Article

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