Novel pH-sensitive charge-reversal cell penetrating peptide conjugated PEG-PLA micelles for docetaxel delivery: In vitro study

International Journal of Pharmaceutics

Volumn 466, Issue 1-2, 2014, Pages 233-245

  Ouahab, Ammar ^a   Cheraga, Nihad ^a   Onoja, Vitus ^a   Shen, Yan ^a   Tu, Jiasheng ^a  

^a CHINA PHARMACEUTICAL UNIVERSITY   (China)

Author keywords

Cell penetrating peptides; Charge reversal; Docetaxel; pH sensitive delivery; Polymeric micelles

Indexed keywords

CELL PENETRATING PEPTIDE; CELL PENETRATING PEPTIDE ARGININE GLYCINE 5; COPOLYMER; DOCETAXEL; DRUG CARRIER; MACROGOL; PH SENSITIVE MASKING DECAPEPTIDE HISTIDINE GLUTAMIC ACID 5; POLYLACTIDE; UNCLASSIFIED DRUG; AMINO ACID; ANTINEOPLASTIC AGENT; MACROGOL DERIVATIVE; MICELLE; MONOMETHOXYPOLYETHYLENEGLYCOL-POLYLACTIDE BLOCK COPOLYMER; OLIGOPEPTIDE; TAXOID;

ARTICLE; CANCER CELL; CANCER CELL CULTURE; CELL ACTIVITY; CELL KILLING; CELL STRAIN MCF 7; CONTROLLED STUDY; CRITICAL MICELLE CONCENTRATION; DRUG CONJUGATION; DRUG CYTOTOXICITY; DRUG DELIVERY SYSTEM; DRUG EFFECT; DRUG PENETRATION; DRUG SOLUBILITY; DRUG STABILITY; DRUG STRUCTURE; DRUG SYNTHESIS; DRUG TARGETING; DRUG UPTAKE; HUMAN; HUMAN CELL; IN VITRO STUDY; INTERNALIZATION; MICELLE; MOLECULAR INTERACTION; PARTICLE SIZE; PH; PH SENSITIVE WITH PEPTIDES OUTSIDE MICELLE; PRIORITY JOURNAL; PROTEIN PROTEIN INTERACTION; PROTON NUCLEAR MAGNETIC RESONANCE; SGC 7901 CELL; STATIC ELECTRICITY; SURFACE CHARGE; SUSTAINED DRUG RELEASE; ZETA POTENTIAL; CELL SURVIVAL; CHEMISTRY; DRUG EFFECTS; MCF 7 CELL LINE; PHOTOMETRY;

AMINO ACIDS; ANTINEOPLASTIC AGENTS; CELL SURVIVAL; CELL-PENETRATING PEPTIDES; DRUG STABILITY; HUMANS; HYDROGEN-ION CONCENTRATION; MCF-7 CELLS; MICELLES; NEPHELOMETRY AND TURBIDIMETRY; OLIGOPEPTIDES; PARTICLE SIZE; POLYETHYLENE GLYCOLS; TAXOIDS;

EID: 84897547884     PISSN: 03785173     EISSN: 18733476     Source Type: Journal    
DOI: 10.1016/j.ijpharm.2014.03.009     Document Type: Article

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