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Volumn 464, Issue 1-2, 2014, Pages 104-110

Investigating permeability related hurdles in oral delivery of 11-keto-β-boswellic acid

Author keywords

Boswellic acids; Caco 2 cells; Gastrointestinal metabolism; Intestinal absorption; Oral bioavailability; Permeability hurdles

Indexed keywords

11 OXO BETA BOSWELLIC ACID; COLECALCIFEROL; CYTOCHROME P450 3A4;

EID: 84896733622     PISSN: 03785173     EISSN: 18733476     Source Type: Journal    
DOI: 10.1016/j.ijpharm.2014.01.019     Document Type: Article
Times cited : (16)

References (30)
  • 1
    • 0007816143 scopus 로고    scopus 로고
    • Salai Guggal - Boswellia serrata: From a herbal medicine to a specific inhibitor of leukotriene biosynthesis
    • H. Ammon Salai Guggal - Boswellia serrata: from a herbal medicine to a specific inhibitor of leukotriene biosynthesis Phytomedicine 3 1996 67 70
    • (1996) Phytomedicine , vol.3 , pp. 67-70
    • Ammon, H.1
  • 2
    • 0025922660 scopus 로고
    • Inhibition of leukotriene B4 formation in rat peritoneal neutrophils by an ethanolic extract of the gum resin exudate of Boswellia serrata
    • H. Ammon, T. Mack, G. Singh, and H. Safayhi Inhibition of leukotriene B4 formation in rat peritoneal neutrophils by an ethanolic extract of the gum resin exudate of Boswellia serrata Planta Med. 57 1991 203 207
    • (1991) Planta Med. , vol.57 , pp. 203-207
    • Ammon, H.1    Mack, T.2    Singh, G.3    Safayhi, H.4
  • 3
    • 0025804183 scopus 로고
    • Correlation between oral drug absorption in humans and apparent drug permeability coefficients in human intestinal epithelial (Caco-2) cells
    • P. Artursson, and J. Karlsson Correlation between oral drug absorption in humans and apparent drug permeability coefficients in human intestinal epithelial (Caco-2) cells Biochem. Biophys. Res. Commun. 175 1991 880 885
    • (1991) Biochem. Biophys. Res. Commun. , vol.175 , pp. 880-885
    • Artursson, P.1    Karlsson, J.2
  • 4
    • 0031659639 scopus 로고    scopus 로고
    • An improved everted gut sac as a simple and accurate technique to measure paracellular transport across the small intestine
    • L. Barthe, J. Woodley, S. Kenworthy, and G. Houin An improved everted gut sac as a simple and accurate technique to measure paracellular transport across the small intestine Eur. J. Drug Metab. Pharmacokinet. 23 1998 313 323 (Pubitemid 28401125)
    • (1998) European Journal of Drug Metabolism and Pharmacokinetics , vol.23 , Issue.2 , pp. 313-323
    • Barthe, L.1    Woodley, J.F.2    Kenworthy, S.3    Houin, G.4
  • 8
    • 84873350225 scopus 로고    scopus 로고
    • In vitro metabolism, permeation, and brain availability of six major boswellic acids from Boswellia serrata gum resins
    • K. Gerbeth, J. Hüsch, G. Fricker, O. Werz, M. Schubert-Zsilavecz, and M. Abdel-Tawab In vitro metabolism, permeation, and brain availability of six major boswellic acids from Boswellia serrata gum resins Fitoterapia 84 2013 99 106
    • (2013) Fitoterapia , vol.84 , pp. 99-106
    • Gerbeth, K.1    Hüsch, J.2    Fricker, G.3    Werz, O.4    Schubert-Zsilavecz, M.5    Abdel-Tawab, M.6
  • 9
    • 0032541951 scopus 로고    scopus 로고
    • Effects of Boswellia serrata gum resin in patients with bronchial asthma: Results of a double-blind, placebo-controlled, 6-week clinical study
    • I. Gupta, V. Gupta, A. Parihar, S. Gupta, R. Lüdtke, H. Safayhi, and H. Ammon Effects of Boswellia serrata gum resin in patients with bronchial asthma: results of a double-blind, placebo-controlled, 6-week clinical study Eur. J. Med. Res. 3 1998 511
    • (1998) Eur. J. Med. Res. , vol.3 , pp. 511
    • Gupta, I.1    Gupta, V.2    Parihar, A.3    Gupta, S.4    Lüdtke, R.5    Safayhi, H.6    Ammon, H.7
  • 10
    • 0024593744 scopus 로고
    • Characterization of the human colon carcinoma cell line (Caco-2) as a model system for intestinal epithelial permeability
    • I.J. Hidalgo, T.J. Raub, and R.T. Borchardt Characterization of the human colon carcinoma cell line (Caco-2) as a model system for intestinal epithelial permeability Gastroenterology 96 1989 736 749 (Pubitemid 19057595)
    • (1989) Gastroenterology , vol.96 , Issue.3 , pp. 736-749
    • Hidalgo, I.J.1    Raub, T.J.2    Borchardt, R.T.3
  • 14
    • 0035800246 scopus 로고    scopus 로고
    • Permeability of lipophilic compounds in drug discovery using in-vitro human absorption model, Caco-2
    • DOI 10.1016/S0378-5173(01)00698-6, PII S0378517301006986
    • G. Krishna, K.-J. Chen, C.-C. Lin, and A.A. Nomeir Permeability of lipophilic compounds in drug discovery using in-vitro human absorption model, Caco-2 Int. J. Pharm. 222 2001 77 89 (Pubitemid 32525789)
    • (2001) International Journal of Pharmaceutics , vol.222 , Issue.1 , pp. 77-89
    • Krishna, G.1    Chen, K.-J.2    Lin, C.-C.3    Nomeir, A.A.4
  • 15
    • 58149168822 scopus 로고    scopus 로고
    • Permeation of Boswellia extract in the Caco-2 model and possible interactions of its constituents KBA and AKBA with OATP1B3 and MRP2
    • P. Krüger, J. Kanzer, J. Hummel, G. Fricker, M. Schubert-Zsilavecz, and M. Abdel-Tawab Permeation of Boswellia extract in the Caco-2 model and possible interactions of its constituents KBA and AKBA with OATP1B3 and MRP2 Eur. J. Pharm. Sci. 36 2009 275 284
    • (2009) Eur. J. Pharm. Sci. , vol.36 , pp. 275-284
    • Krüger, P.1    Kanzer, J.2    Hummel, J.3    Fricker, G.4    Schubert-Zsilavecz, M.5    Abdel-Tawab, M.6
  • 17
    • 33845321884 scopus 로고    scopus 로고
    • Boswellic acids: Biological actions and molecular targets
    • DOI 10.2174/092986706779010333
    • D. Poeckel, and O. Werz Boswellic acids: biological actions and molecular targets Curr. Med. Chem. 13 2006 3359 3369 (Pubitemid 44873750)
    • (2006) Current Medicinal Chemistry , vol.13 , Issue.28 , pp. 3359-3369
    • Poeckel, D.1    Werz, O.2
  • 21
    • 0024462668 scopus 로고
    • Anti-arthritic activity of boswellic acids in bovine serum albumin (BSA)-induced arthritis
    • M. Sharma, S. Bani, and G. Singh Anti-arthritic activity of boswellic acids in bovine serum albumin (BSA)-induced arthritis Int. J. Immunopharmacol. 11 1989 647 652 (Pubitemid 19239439)
    • (1989) International Journal of Immunopharmacology , vol.11 , Issue.6 , pp. 647-652
    • Sharma, M.L.1    Bani, S.2    Singh, G.B.3
  • 22
    • 0024023609 scopus 로고
    • Effect of salai guggal ex-Boswellia serrata on cellular and humoral immune responses and leucocyte migration
    • M. Sharma, A. Khajuria, A. Kaul, S. Singh, G. Singh, and C. Atal Effect of salai guggal ex-Boswellia serrata on cellular and humoral immune responses and leucocyte migration Agents Actions 24 1988 161 164
    • (1988) Agents Actions , vol.24 , pp. 161-164
    • Sharma, M.1    Khajuria, A.2    Kaul, A.3    Singh, S.4    Singh, G.5    Atal, C.6
  • 24
    • 3042613491 scopus 로고    scopus 로고
    • Characterization of the rates of testosterone metabolism to various products and of glutathione transferase and sulfotransferase activities in rat intestine and comparison to the corresponding hepatic and renal drug-metabolizing enzymes
    • DOI 10.1016/j.cbi.2004.05.001, PII S0009279704000481
    • A.-K. Sohlenius-Sternbeck, and A. Orzechowski Characterization of the rates of testosterone metabolism to various products and of glutathione transferase and sulfotransferase activities in rat intestine and comparison to the corresponding hepatic and renal drug-metabolizing enzymes Chem. Biol. Interact. 148 2004 49 56 (Pubitemid 38824660)
    • (2004) Chemico-Biological Interactions , vol.148 , Issue.1-2 , pp. 49-56
    • Sohlenius-Sternbeck, A.-K.1    Orzechowski, A.2
  • 26
    • 79551514621 scopus 로고    scopus 로고
    • Identification of permeability-related hurdles in oral delivery of curcumin using the Caco-2 cell model
    • B. Wahlang, Y.B. Pawar, and A.K. Bansal Identification of permeability-related hurdles in oral delivery of curcumin using the Caco-2 cell model Eur. J. Pharm. Biopharm. 77 2011 275 282
    • (2011) Eur. J. Pharm. Biopharm. , vol.77 , pp. 275-282
    • Wahlang, B.1    Pawar, Y.B.2    Bansal, A.K.3
  • 27
    • 6544259277 scopus 로고
    • The use of sacs of everted small intestine for the study of the transference of substances from the mucosal to the serosal surface
    • T.H. Wilson, and G. Wiseman The use of sacs of everted small intestine for the study of the transference of substances from the mucosal to the serosal surface J. Physiol. 123 1954 116 125
    • (1954) J. Physiol. , vol.123 , pp. 116-125
    • Wilson, T.H.1    Wiseman, G.2
  • 29
    • 0030990079 scopus 로고    scopus 로고
    • In vitro permeability across Caco-2 cells (colonic) can predict in vivo (small intestinal) absorption in man - Fact or myth
    • DOI 10.1023/A:1012102522787
    • S. Yee In vitro permeability across Caco-2 cells (colonic) can predict in vivo (small intestinal) absorption in man - fact or myth Pharm. Res. 14 1997 763 766 (Pubitemid 27281671)
    • (1997) Pharmaceutical Research , vol.14 , Issue.6 , pp. 763-766
    • Yee, S.1
  • 30
    • 0037457790 scopus 로고    scopus 로고
    • In vitro and in vivo models for assessing drug efflux transporter activity
    • DOI 10.1016/S0169-409X(02)00170-9, PII S0169409X02001709
    • Y. Zhang, C. Bachmeier, and D.W. Miller In vitro and in vivo models for assessing drug efflux transporter activity Adv. Drug Deliv. Rev. 55 2003 31 51 (Pubitemid 36078453)
    • (2003) Advanced Drug Delivery Reviews , vol.55 , Issue.1 , pp. 31-51
    • Zhang, Y.1    Bachmeier, C.2    Miller, D.W.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.