-
1
-
-
0028149954
-
Tiagabine, SK&F 89976-A, CI-966, and NNC-711 are selective for the cloned GABA transporter GAT-1
-
Borden L.A., Murali Dhar T.G., Smith K.E., Weinshank R.L., Branchek T.A., Gluchowski C. Tiagabine, SK&F 89976-A, CI-966, and NNC-711 are selective for the cloned GABA transporter GAT-1. Eur. J. Pharmacol. 1994, 269:219-224.
-
(1994)
Eur. J. Pharmacol.
, vol.269
, pp. 219-224
-
-
Borden, L.A.1
Murali Dhar, T.G.2
Smith, K.E.3
Weinshank, R.L.4
Branchek, T.A.5
Gluchowski, C.6
-
2
-
-
0029942452
-
Tiagabine pharmacology in profile
-
Brodie M.J. Tiagabine pharmacology in profile. Epilepsia 1995, 36(Suppl. 6):S7-S9.
-
(1995)
Epilepsia
, vol.36
, Issue.SUPPL. 6
-
-
Brodie, M.J.1
-
3
-
-
80054024231
-
Magnolol, a major bioactive constituent of the bark of Magnolia officinalis, exerts antiepileptic effects via the GABA/benzodiazepine receptor complex in mice
-
Chen C.R., Tan R., Qu W.M., Wu Z., Wang Y., Urade Y., Huang Z.L. Magnolol, a major bioactive constituent of the bark of Magnolia officinalis, exerts antiepileptic effects via the GABA/benzodiazepine receptor complex in mice. Br. J. Pharmacol. 2011, 164:1534-1546.
-
(2011)
Br. J. Pharmacol.
, vol.164
, pp. 1534-1546
-
-
Chen, C.R.1
Tan, R.2
Qu, W.M.3
Wu, Z.4
Wang, Y.5
Urade, Y.6
Huang, Z.L.7
-
4
-
-
0036897386
-
Number, density, and surface/cytoplasmic distribution of GABA transporters at presynaptic structures of knock-in mice carrying GABA transporter subtype 1-green fluorescent protein fusions
-
Chiu C.S., Jensen K., Sokolova I., Wang D., Li M., Deshpande P., Davidson N., Mody I., Quick M.W., Quake S.R., Lester H.A. Number, density, and surface/cytoplasmic distribution of GABA transporters at presynaptic structures of knock-in mice carrying GABA transporter subtype 1-green fluorescent protein fusions. J. Neurosci. 2002, 22:10251-10266.
-
(2002)
J. Neurosci.
, vol.22
, pp. 10251-10266
-
-
Chiu, C.S.1
Jensen, K.2
Sokolova, I.3
Wang, D.4
Li, M.5
Deshpande, P.6
Davidson, N.7
Mody, I.8
Quick, M.W.9
Quake, S.R.10
Lester, H.A.11
-
5
-
-
3042649213
-
GABA transporters in the mammalian cerebral cortex: localization, development and pathological implications
-
Conti F., Minelli A., Melone M. GABA transporters in the mammalian cerebral cortex: localization, development and pathological implications. Brain Res. Brain Res. Rev. 2004, 45:196-212.
-
(2004)
Brain Res. Brain Res. Rev.
, vol.45
, pp. 196-212
-
-
Conti, F.1
Minelli, A.2
Melone, M.3
-
6
-
-
33749989285
-
Treating insomnia: current and investigational pharmacological approaches
-
Ebert B., Wafford K.A., Deacon S. Treating insomnia: current and investigational pharmacological approaches. Pharmacol. Ther. 2006, 112:612-629.
-
(2006)
Pharmacol. Ther.
, vol.112
, pp. 612-629
-
-
Ebert, B.1
Wafford, K.A.2
Deacon, S.3
-
8
-
-
0025048435
-
Cloning and expression of a rat brain GABA transporter
-
Guastella J., Nelson N., Nelson H., Czyzyk L., Keynan S., Miedel M.C., Davidson N., Lester H.A., Kanner B.I. Cloning and expression of a rat brain GABA transporter. Science 1990, 249:1303-1306.
-
(1990)
Science
, vol.249
, pp. 1303-1306
-
-
Guastella, J.1
Nelson, N.2
Nelson, H.3
Czyzyk, L.4
Keynan, S.5
Miedel, M.C.6
Davidson, N.7
Lester, H.A.8
Kanner, B.I.9
-
9
-
-
77954354338
-
Benzodiazepine receptor agonists cause drug-specific and state-specific alterations in EEG power and acetylcholine release in rat pontine reticular formation
-
Hambrecht-Wiedbusch V.S., Gauthier E.A., Baghdoyan H.A., Lydic R. Benzodiazepine receptor agonists cause drug-specific and state-specific alterations in EEG power and acetylcholine release in rat pontine reticular formation. Sleep 2010, 33:909-918.
-
(2010)
Sleep
, vol.33
, pp. 909-918
-
-
Hambrecht-Wiedbusch, V.S.1
Gauthier, E.A.2
Baghdoyan, H.A.3
Lydic, R.4
-
10
-
-
15244362192
-
An adenosine A receptor agonist induces sleep by increasing GABA release in the tuberomammillary nucleus to inhibit histaminergic systems in rats
-
Hong Z.Y., Huang Z.L., Qu W.M., Eguchi N., Urade Y., Hayaishi O. An adenosine A receptor agonist induces sleep by increasing GABA release in the tuberomammillary nucleus to inhibit histaminergic systems in rats. J. Neurochem. 2005, 92:1542-1549.
-
(2005)
J. Neurochem.
, vol.92
, pp. 1542-1549
-
-
Hong, Z.Y.1
Huang, Z.L.2
Qu, W.M.3
Eguchi, N.4
Urade, Y.5
Hayaishi, O.6
-
11
-
-
24944458193
-
Adenosine A2A, but not A1, receptors mediate the arousal effect of caffeine
-
Huang Z.L., Qu W.M., Eguchi N., Chen J.F., Schwarzschild M.A., Fredholm B.B., Urade Y., Hayaishi O. Adenosine A2A, but not A1, receptors mediate the arousal effect of caffeine. Nat. Neurosci. 2005, 8:858-859.
-
(2005)
Nat. Neurosci.
, vol.8
, pp. 858-859
-
-
Huang, Z.L.1
Qu, W.M.2
Eguchi, N.3
Chen, J.F.4
Schwarzschild, M.A.5
Fredholm, B.B.6
Urade, Y.7
Hayaishi, O.8
-
12
-
-
0035859825
-
Arousal effect of orexin A depends on activation of the histaminergic system
-
Huang Z.L., Qu W.M., Li W.D., Mochizuki T., Eguchi N., Watanabe T., Urade Y., Hayaishi O. Arousal effect of orexin A depends on activation of the histaminergic system. Proc. Natl. Acad. Sci. USA 2001, 98:9965-9970.
-
(2001)
Proc. Natl. Acad. Sci. USA
, vol.98
, pp. 9965-9970
-
-
Huang, Z.L.1
Qu, W.M.2
Li, W.D.3
Mochizuki, T.4
Eguchi, N.5
Watanabe, T.6
Urade, Y.7
Hayaishi, O.8
-
13
-
-
0142058598
-
GABA transporter-1 (GAT1)-deficient mice: differential tonic activation of GABAA versus GABAB receptors in the hippocampus
-
Jensen K., Chiu C.S., Sokolova I., Lester H.A., Mody I. GABA transporter-1 (GAT1)-deficient mice: differential tonic activation of GABAA versus GABAB receptors in the hippocampus. J. Neurophysiol. 2003, 90:2690-2701.
-
(2003)
J. Neurophysiol.
, vol.90
, pp. 2690-2701
-
-
Jensen, K.1
Chiu, C.S.2
Sokolova, I.3
Lester, H.A.4
Mody, I.5
-
14
-
-
0031914241
-
Effect of the GABA uptake inhibitor tiagabine on sleep and EEG power spectra in the rat
-
Lancel M., Faulhaber J., Deisz R.A. Effect of the GABA uptake inhibitor tiagabine on sleep and EEG power spectra in the rat. Br. J. Pharmacol. 1998, 123:1471-1477.
-
(1998)
Br. J. Pharmacol.
, vol.123
, pp. 1471-1477
-
-
Lancel, M.1
Faulhaber, J.2
Deisz, R.A.3
-
16
-
-
84864765560
-
Safranal enhances non-rapid eye movement sleep in pentobarbital-treated mice
-
Liu Z., Xu X.H., Liu T.Y., Hong Z.Y., Urade Y., Huang Z.L., Qu W.M. Safranal enhances non-rapid eye movement sleep in pentobarbital-treated mice. CNS Neurosci. Ther. 2012, 18:623-630.
-
(2012)
CNS Neurosci. Ther.
, vol.18
, pp. 623-630
-
-
Liu, Z.1
Xu, X.H.2
Liu, T.Y.3
Hong, Z.Y.4
Urade, Y.5
Huang, Z.L.6
Qu, W.M.7
-
17
-
-
76749145072
-
Neuronal and non-neuronal GABA transporters as targets for antiepileptic drugs
-
Madsen K.K., White H.S., Schousboe A. Neuronal and non-neuronal GABA transporters as targets for antiepileptic drugs. Pharmacol. Ther. 2010, 125:394-401.
-
(2010)
Pharmacol. Ther.
, vol.125
, pp. 394-401
-
-
Madsen, K.K.1
White, H.S.2
Schousboe, A.3
-
18
-
-
0035115746
-
The GABA uptake inhibitor tiagabine promotes slow wave sleep in normal elderly subjects
-
Mathias S., Wetter T.C., Steiger A., Lancel M. The GABA uptake inhibitor tiagabine promotes slow wave sleep in normal elderly subjects. Neurobiol. Aging 2001, 22:247-253.
-
(2001)
Neurobiol. Aging
, vol.22
, pp. 247-253
-
-
Mathias, S.1
Wetter, T.C.2
Steiger, A.3
Lancel, M.4
-
19
-
-
0034839786
-
Brain structures and mechanisms involved in the generation of NREM sleep: focus on the preoptic hypothalamus
-
McGinty D., Szymusiak R. Brain structures and mechanisms involved in the generation of NREM sleep: focus on the preoptic hypothalamus. Sleep Med. Rev. 2001, 5:323-342.
-
(2001)
Sleep Med. Rev.
, vol.5
, pp. 323-342
-
-
McGinty, D.1
Szymusiak, R.2
-
20
-
-
0030458402
-
GABA release in posterior hypothalamus across sleep-wake cycle
-
Nitz D., Siegel J.M. GABA release in posterior hypothalamus across sleep-wake cycle. Am. J. Physiol. 1996, 271:R1707-1712.
-
(1996)
Am. J. Physiol.
, vol.271
-
-
Nitz, D.1
Siegel, J.M.2
-
21
-
-
0026643143
-
GABA and behavior: the role of receptor subtypes
-
Paredes R.G., Agmo A. GABA and behavior: the role of receptor subtypes. Neurosci. Biobehav. Rev. 1992, 16:145-170.
-
(1992)
Neurosci. Biobehav. Rev.
, vol.16
, pp. 145-170
-
-
Paredes, R.G.1
Agmo, A.2
-
22
-
-
70349214740
-
D(1)/D(2) receptor-targeting l-stepholidine, an active ingredient of the Chinese herb Stephonia, induces non-rapid eye movement sleep in mice
-
Qiu M.H., Qu W.M., Xu X.H., Yan M.M., Urade Y., Huang Z.L. D(1)/D(2) receptor-targeting l-stepholidine, an active ingredient of the Chinese herb Stephonia, induces non-rapid eye movement sleep in mice. Pharmacol. Biochem. Behav. 2009, 94:16-23.
-
(2009)
Pharmacol. Biochem. Behav.
, vol.94
, pp. 16-23
-
-
Qiu, M.H.1
Qu, W.M.2
Xu, X.H.3
Yan, M.M.4
Urade, Y.5
Huang, Z.L.6
-
23
-
-
33845195769
-
Lipocalin-type prostaglandin D synthase produces prostaglandin D2 involved in regulation of physiological sleep
-
Qu W.M., Huang Z.L., Xu X.H., Aritake K., Eguchi N., Nambu F., Narumiya S., Urade Y., Hayaishi O. Lipocalin-type prostaglandin D synthase produces prostaglandin D2 involved in regulation of physiological sleep. Proc. Natl. Acad. Sci. USA 2006, 103:17949-17954.
-
(2006)
Proc. Natl. Acad. Sci. USA
, vol.103
, pp. 17949-17954
-
-
Qu, W.M.1
Huang, Z.L.2
Xu, X.H.3
Aritake, K.4
Eguchi, N.5
Nambu, F.6
Narumiya, S.7
Urade, Y.8
Hayaishi, O.9
-
24
-
-
77949870971
-
Essential role of dopamine D2 receptor in the maintenance of wakefulness, but not in homeostatic regulation of sleep, in mice
-
Qu W.M., Xu X.H., Yan M.M., Wang Y.Q., Urade Y., Huang Z.L. Essential role of dopamine D2 receptor in the maintenance of wakefulness, but not in homeostatic regulation of sleep, in mice. J. Neurosci. 2010, 30:4382-4389.
-
(2010)
J. Neurosci.
, vol.30
, pp. 4382-4389
-
-
Qu, W.M.1
Xu, X.H.2
Yan, M.M.3
Wang, Y.Q.4
Urade, Y.5
Huang, Z.L.6
-
25
-
-
0023891990
-
Expression of c-Fos protein in brain: metabolic mapping at the cellular level
-
Sagar S.M., Sharp F.R., Curran T. Expression of c-Fos protein in brain: metabolic mapping at the cellular level. Science 1988, 240:1328-1331.
-
(1988)
Science
, vol.240
, pp. 1328-1331
-
-
Sagar, S.M.1
Sharp, F.R.2
Curran, T.3
-
26
-
-
78650230533
-
Sleep state switching
-
Saper, C.B., Fuller, P.M., Pedersen, N.P., Lu, J., Scammell, T.E., 2010. Sleep state switching. Neuron 68, 1023-1042.
-
(2010)
Neuron
, vol.68
, pp. 1023-1042
-
-
Saper, C.B.1
Fuller, P.M.2
Pedersen, N.P.3
Lu, J.4
Scammell, T.E.5
-
27
-
-
0032703335
-
A review of the antiepileptic drug tiagabine
-
Schachter S.C. A review of the antiepileptic drug tiagabine. Clin. Neuropharmacol. 1999, 22:312-317.
-
(1999)
Clin. Neuropharmacol.
, vol.22
, pp. 312-317
-
-
Schachter, S.C.1
-
28
-
-
0029671044
-
Activation of ventrolateral preoptic neurons during sleep
-
Sherin J.E., Shiromani P.J., McCarley R.W., Saper C.B. Activation of ventrolateral preoptic neurons during sleep. Science 1996, 271:216-219.
-
(1996)
Science
, vol.271
, pp. 216-219
-
-
Sherin, J.E.1
Shiromani, P.J.2
McCarley, R.W.3
Saper, C.B.4
-
29
-
-
0026539825
-
NNC-711, a novel potent and selective gamma-aminobutyric acid uptake inhibitor: pharmacological characterization
-
Suzdak P.D., Frederiksen K., Andersen K.E., Sorensen P.O., Knutsen L.J., Nielsen E.B. NNC-711, a novel potent and selective gamma-aminobutyric acid uptake inhibitor: pharmacological characterization. Eur. J. Pharmacol. 1992, 224:189-198.
-
(1992)
Eur. J. Pharmacol.
, vol.224
, pp. 189-198
-
-
Suzdak, P.D.1
Frederiksen, K.2
Andersen, K.E.3
Sorensen, P.O.4
Knutsen, L.J.5
Nielsen, E.B.6
-
30
-
-
0035933064
-
Diazepam-induced changes in sleep: role of the alpha 1 GABA(A) receptor subtype
-
Tobler I., Kopp C., Deboer T., Rudolph U. Diazepam-induced changes in sleep: role of the alpha 1 GABA(A) receptor subtype. Proc. Natl. Acad. Sci. USA 2001, 98:6464-6469.
-
(2001)
Proc. Natl. Acad. Sci. USA
, vol.98
, pp. 6464-6469
-
-
Tobler, I.1
Kopp, C.2
Deboer, T.3
Rudolph, U.4
-
31
-
-
77958586336
-
Differential effects of GABAB receptor subtypes, {gamma}-hydroxybutyric acid, and Baclofen on EEG activity and sleep regulation
-
Vienne J., Bettler B., Franken P., Tafti M. Differential effects of GABAB receptor subtypes, {gamma}-hydroxybutyric acid, and Baclofen on EEG activity and sleep regulation. J. Neurosci. 2010, 30:14194-14204.
-
(2010)
J. Neurosci.
, vol.30
, pp. 14194-14204
-
-
Vienne, J.1
Bettler, B.2
Franken, P.3
Tafti, M.4
-
32
-
-
44449104126
-
Emerging anti-insomnia drugs: tackling sleeplessness and the quality of wake time
-
Wafford K.A., Ebert B. Emerging anti-insomnia drugs: tackling sleeplessness and the quality of wake time. Nat. Rev. Drug. Discov. 2008, 7:530-540.
-
(2008)
Nat. Rev. Drug. Discov.
, vol.7
, pp. 530-540
-
-
Wafford, K.A.1
Ebert, B.2
-
33
-
-
84895888864
-
Essential roles of GABA transporter-1 in controlling rapid eye movement sleep and in increased slow wave activity after sleep deprivation
-
PLoS One, (in press)
-
Xu, Qu, Bian, Huang, Fei, Urade and Huang, Essential roles of GABA transporter-1 in controlling rapid eye movement sleep and in increased slow wave activity after sleep deprivation, PLoS One, (in press).
-
-
-
Xu1
Qu2
Bian3
Huang4
Fei5
Urade6
Huang7
-
34
-
-
78751476671
-
Selection of optimal epoch duration in assessment of rodent sleep-wake profiles
-
Yan M.M., Xu X.H., Huang Z.L., Yao M.H., Urade Y., QU W.M. Selection of optimal epoch duration in assessment of rodent sleep-wake profiles. Sleep Biol. Rhythms 2011, 9:46-55.
-
(2011)
Sleep Biol. Rhythms
, vol.9
, pp. 46-55
-
-
Yan, M.M.1
Xu, X.H.2
Huang, Z.L.3
Yao, M.H.4
Urade, Y.5
QU, W.M.6
|