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Volumn 43, Issue 3, 2014, Pages 884-897

Potential antimicrobial agents for the treatment of multidrug-resistant tuberculosis

Author keywords

[No Author keywords available]

Indexed keywords

ANTIINFECTIVE AGENT; COLECALCIFEROL; COTRIMOXAZOLE; CYTOCHROME P450 1A2; CYTOCHROME P450 2D6; CYTOCHROME P450 3A4; DISULFIRAM; DOXYCYCLINE; ETHAMBUTOL; ISONIAZID; METRONIDAZOLE; PHENOTHIAZINE; PYRAZINAMIDE; RIFAMPICIN; THIORIDAZINE; TIGECYCLINE;

EID: 84895560404     PISSN: 09031936     EISSN: 13993003     Source Type: Journal    
DOI: 10.1183/09031936.00113713     Document Type: Review
Times cited : (56)

References (93)
  • 1
    • 84865677110 scopus 로고    scopus 로고
    • Tuberculosis, drug resistance, and the history of modern medicine
    • Keshavjee S, Farmer PE. Tuberculosis, drug resistance, and the history of modern medicine. N Engl J Med 2012; 367: 931-936.
    • (2012) N Engl J Med , vol.367 , pp. 931-936
    • Keshavjee, S.1    Farmer, P.E.2
  • 2
    • 84860345846 scopus 로고    scopus 로고
    • TB and MDR/XDR-TB in European Union and European Economic Area countries: Managed or mismanaged?
    • Migliori GB, Sotgiu G, D'Ambrosio L, et al. TB and MDR/XDR-TB in European Union and European Economic Area countries: managed or mismanaged? Eur Respir J 2012; 39: 619-625.
    • (2012) Eur Respir J , vol.39 , pp. 619-625
    • Migliori, G.B.1    Sotgiu, G.2    D'ambrosio, L.3
  • 3
    • 84878776777 scopus 로고    scopus 로고
    • Delamanid improves outcomes and reduces mortality in multidrugresistant tuberculosis
    • Skripconoka V, Danilovits M, Pehme L, et al. Delamanid improves outcomes and reduces mortality in multidrugresistant tuberculosis. Eur Respir J 2013; 41: 1393-1400.
    • (2013) Eur Respir J , vol.41 , pp. 1393-1400
    • Skripconoka, V.1    Danilovits, M.2    Pehme, L.3
  • 4
    • 84875844457 scopus 로고    scopus 로고
    • Transmission of multidrug-resistant and extensively drug-resistant tuberculosis in a metropolitan city
    • Leung EC, Leung CC, Kam KM, et al. Transmission of multidrug-resistant and extensively drug-resistant tuberculosis in a metropolitan city. Eur Respir J 2013; 41: 901-908.
    • (2013) Eur Respir J , vol.41 , pp. 901-908
    • Leung, E.C.1    Leung, C.C.2    Kam, K.M.3
  • 5
    • 60749083864 scopus 로고    scopus 로고
    • Treatment outcomes among patients with multidrug-resistant tuberculosis: Systematic review and meta-analysis
    • Orenstein EW, Basu S, Shah NS, et al. Treatment outcomes among patients with multidrug-resistant tuberculosis: systematic review and meta-analysis. Lancet Infect Dis 2009; 9: 153-161.
    • (2009) Lancet Infect Dis , vol.9 , pp. 153-161
    • Orenstein, E.W.1    Basu, S.2    Shah, N.S.3
  • 6
    • 84879670662 scopus 로고    scopus 로고
    • Targeting multidrug-resistant tuberculosis (MDR-TB) by therapeutic vaccines
    • Prabowo SA, Gröschel MI, Schmidt EDL, et al. Targeting multidrug-resistant tuberculosis (MDR-TB) by therapeutic vaccines. Med Microbiol Immunol 2013; 202: 95-104.
    • (2013) Med Microbiol Immunol , vol.202 , pp. 95-104
    • Prabowo, S.A.1    Gröschel, M.I.2    Schmidt, E.D.L.3
  • 7
  • 8
    • 84862650730 scopus 로고    scopus 로고
    • World Health Organization. (WHO/HTM/TB/2010.7). Geneva, WHO Press
    • World Health Organization. Global Tuberculosis Control Report 2010. (WHO/HTM/TB/2010.7). Geneva, WHO Press, 2010.
    • (2010) Global Tuberculosis Control Report 2010
  • 9
    • 84870747517 scopus 로고    scopus 로고
    • Efficacy and safety of meropenem-clavulanate added to linezolid containing regimens in the treatment of MDR-/XDR-TB
    • De Lorenzo S, Alffenaar JW, Sotgiu G, et al. Efficacy and safety of meropenem-clavulanate added to linezolid containing regimens in the treatment of MDR-/XDR-TB. Eur Respir J 2013; 41: 1386-1392.
    • (2013) Eur Respir J , vol.41 , pp. 1386-1392
    • De Lorenzo, S.1    Alffenaar, J.W.2    Sotgiu, G.3
  • 10
    • 84894198937 scopus 로고    scopus 로고
    • World Health Organization. (WHO/HTM/TB/2012.6). Geneva, WHO Press
    • World Health Organization. Global Tuberculosis Report 2012. (WHO/HTM/TB/2012.6). Geneva, WHO Press, 2010.
    • (2010) Global Tuberculosis Report 2012
  • 11
    • 84861880367 scopus 로고    scopus 로고
    • Alarming levels of drug-resistant tuberculosis in Belarus: Results of a survey in Minsk
    • Skrahina A, Hurevich H, Zalutskaya A, et al. Alarming levels of drug-resistant tuberculosis in Belarus: results of a survey in Minsk. Eur Respir J 2012; 39: 1425-1431.
    • (2012) Eur Respir J , vol.39 , pp. 1425-1431
    • Skrahina, A.1    Hurevich, H.2    Zalutskaya, A.3
  • 13
    • 84862214485 scopus 로고    scopus 로고
    • Geno Type MTBDRsl performance on clinical samples with diverse genetic background
    • Miotto P, Cabibbe AM, Mantegani P, et al. Geno Type MTBDRsl performance on clinical samples with diverse genetic background. Eur Respir J 2012; 40: 690-698.
    • (2012) Eur Respir J , vol.40 , pp. 690-698
    • Miotto, P.1    Cabibbe, A.M.2    Mantegani, P.3
  • 14
    • 0042140672 scopus 로고    scopus 로고
    • Inhibition of respiration by nitric oxide induces a Mycobacterium tuberculosis dormancy program
    • Voskuil MI, Schnappinger D, Visconti KC, et al. Inhibition of respiration by nitric oxide induces a Mycobacterium tuberculosis dormancy program. J Exp Med 2003; 198: 705-713.
    • (2003) J Exp Med , vol.198 , pp. 705-713
    • Voskuil, M.I.1    Schnappinger, D.2    Visconti, K.C.3
  • 15
    • 33747852367 scopus 로고    scopus 로고
    • Current status of some antituberculosis drugs and the development of new antituberculous agents with special reference to their in vitro and in vivo antimicrobial activities
    • Tomioka H. Current status of some antituberculosis drugs and the development of new antituberculous agents with special reference to their in vitro and in vivo antimicrobial activities. Curr Pharm Des 2006; 12: 4047-4070.
    • (2006) Curr Pharm des , vol.12 , pp. 4047-4070
    • Tomioka, H.1
  • 16
    • 0030462751 scopus 로고    scopus 로고
    • Inhibition of the respiration of multi-drug resistant clinical isolates of Mycobacterium tuberculosis by thioridazine: Potential use for initial therapy of freshly diagnosed tuberculosis
    • Amaral L, Kristiansen JE, Abebe LS, et al. Inhibition of the respiration of multi-drug resistant clinical isolates of Mycobacterium tuberculosis by thioridazine: potential use for initial therapy of freshly diagnosed tuberculosis. J Antimicrob Chemother 1996; 38: 1049-1053.
    • (1996) J Antimicrob Chemother , vol.38 , pp. 1049-1053
    • Amaral, L.1    Kristiansen, J.E.2    Abebe, L.S.3
  • 17
    • 33846969173 scopus 로고    scopus 로고
    • In vitro and ex vivo activity of thioridazine derivatives against Mycobacterium tuberculosis
    • Martins M, Schelz Z, Martins A, et al. In vitro and ex vivo activity of thioridazine derivatives against Mycobacterium tuberculosis. Int J Antimicrob Agents 2007; 29: 338-340.
    • (2007) Int J Antimicrob Agents , vol.29 , pp. 338-340
    • Martins, M.1    Schelz, Z.2    Martins, A.3
  • 18
    • 35648948351 scopus 로고    scopus 로고
    • The curative activity of thioridazine on mice infected with Mycobacterium tuberculosis
    • Martins M, Viveiros M, Kristiansen JE, et al. The curative activity of thioridazine on mice infected with Mycobacterium tuberculosis. In Vivo 2007; 21: 771-775.
    • (2007) Vivo , vol.21 , pp. 771-775
    • Martins, M.1    Viveiros, M.2    Kristiansen, J.E.3
  • 19
    • 0018135926 scopus 로고
    • Distribution of thioridazine and its metabolites in human tissues and fluids obtained postmortem
    • Dinovo EC, Bost RO, Sunshine I, et al. Distribution of thioridazine and its metabolites in human tissues and fluids obtained postmortem. Clin Chem 1978; 24: 1828-1830.
    • (1978) Clin Chem , vol.24 , pp. 1828-1830
    • Dinovo, E.C.1    Bost, R.O.2    Sunshine, I.3
  • 20
    • 35248895271 scopus 로고    scopus 로고
    • Thioridazine: Resurrection as an antimicrobial agent?
    • Thanacoody HK. Thioridazine: resurrection as an antimicrobial agent? Br J Clin Pharmacol 2007; 64: 566-574.
    • (2007) Br J Clin Pharmacol , vol.64 , pp. 566-574
    • Thanacoody, H.K.1
  • 21
    • 0028024035 scopus 로고
    • Metronidazole is bactericidal to dormant cells of Mycobacterium tuberculosis
    • Wayne LG, Sramek HA. Metronidazole is bactericidal to dormant cells of Mycobacterium tuberculosis. Antimicrob Agents Chemother 1994; 38: 2054-2058.
    • (1994) Antimicrob Agents Chemother , vol.38 , pp. 2054-2058
    • Wayne, L.G.1    Sramek, H.A.2
  • 23
    • 77952638904 scopus 로고    scopus 로고
    • Activity of drug combinations against dormant Mycobacterium tuberculosis
    • Filippini P, Iona E, Piccaro G, et al. Activity of drug combinations against dormant Mycobacterium tuberculosis. Antimicrob Agents Chemother 2010; 54: 2712-2715.
    • (2010) Antimicrob Agents Chemother , vol.54 , pp. 2712-2715
    • Filippini, P.1    Iona, E.2    Piccaro, G.3
  • 24
    • 47649096186 scopus 로고    scopus 로고
    • Metronidazole lacks activity against Mycobacterium tuberculosis in an in vivo hypoxic granuloma model of latency
    • Klinkenberg LG, Sutherland LA, Bishai WR, et al. Metronidazole lacks activity against Mycobacterium tuberculosis in an in vivo hypoxic granuloma model of latency. J Infect Dis 2008; 198: 275-283.
    • (2008) J Infect Dis , vol.198 , pp. 275-283
    • Klinkenberg, L.G.1    Sutherland, L.A.2    Bishai, W.R.3
  • 25
    • 55849117720 scopus 로고    scopus 로고
    • Metronidazole lacks antibacterial activity in guinea pigs infected with Mycobacterium tuberculosis
    • Hoff DR, Caraway ML, Brooks EJ, et al. Metronidazole lacks antibacterial activity in guinea pigs infected with Mycobacterium tuberculosis. Antimicrob Agents Chemother 2008; 52: 4137-4140.
    • (2008) Antimicrob Agents Chemother , vol.52 , pp. 4137-4140
    • Hoff, D.R.1    Caraway, M.L.2    Brooks, E.J.3
  • 26
    • 84861163743 scopus 로고    scopus 로고
    • Evaluation of a mouse model of necrotic granuloma formation using C3HeB/FeJ mice for testing of drugs against Mycobacterium tuberculosis
    • Driver ER, Ryan GJ, Hoff DR, et al. Evaluation of a mouse model of necrotic granuloma formation using C3HeB/FeJ mice for testing of drugs against Mycobacterium tuberculosis. Antimicrob Agents Chemother 2012; 56: 3181-3195.
    • (2012) Antimicrob Agents Chemother , vol.56 , pp. 3181-3195
    • Driver, E.R.1    Ryan, G.J.2    Hoff, D.R.3
  • 27
    • 0032977537 scopus 로고    scopus 로고
    • Pharmacokinetics and pharmacodynamics of the nitroimidazole antimicrobials
    • Lamp KC, Freeman CD, Klutman NE, et al. Pharmacokinetics and pharmacodynamics of the nitroimidazole antimicrobials. Clin Pharmacokinet 1999; 36: 353-373.
    • (1999) Clin Pharmacokinet , vol.36 , pp. 353-373
    • Lamp, K.C.1    Freeman, C.D.2    Klutman, N.E.3
  • 28
    • 85036409910 scopus 로고    scopus 로고
    • In vitro effect of tigecycline against Mycobacterium tuberculosis and a review of the available drugs for tuberculosis
    • Coban AY, Deveci A, Cayci YT, et al. In vitro effect of tigecycline against Mycobacterium tuberculosis and a review of the available drugs for tuberculosis. African J Microbiol Res 2011; 5: 311-315.
    • (2011) African J Microbiol Res , vol.5 , pp. 311-315
    • Coban, A.Y.1    Deveci, A.2    Cayci, Y.T.3
  • 29
    • 1642492861 scopus 로고    scopus 로고
    • The glycylcyclines: A comparative review with the tetracyclines
    • Zhanel GG, Homenuik K, Nichol K, et al. The glycylcyclines: a comparative review with the tetracyclines. Drugs 2004; 64: 63-88.
    • (2004) Drugs , vol.64 , pp. 63-88
    • Zhanel, G.G.1    Homenuik, K.2    Nichol, K.3
  • 30
    • 19544371022 scopus 로고    scopus 로고
    • Steady-state serum and intrapulmonary pharmacokinetics and pharmacodynamics of tigecycline
    • Conte JE Jr, Golden JA, Kelly MG, et al. Steady-state serum and intrapulmonary pharmacokinetics and pharmacodynamics of tigecycline. Int J Antimicrob Agents 2005; 25: 523-529.
    • (2005) Int J Antimicrob Agents , vol.25 , pp. 523-529
    • Conte Jr., J.E.1    Golden, J.A.2    Kelly, M.G.3
  • 31
    • 84860621068 scopus 로고    scopus 로고
    • Doxycycline and HIV infection suppress tuberculosis-induced matrix metalloproteinases
    • Walker NF, Clark SO, Oni T, et al. Doxycycline and HIV infection suppress tuberculosis-induced matrix metalloproteinases. Am J Respir Crit Care Med 2012; 185: 989-997.
    • (2012) Am J Respir Crit Care Med , vol.185 , pp. 989-997
    • Walker, N.F.1    Clark, S.O.2    Oni, T.3
  • 32
    • 16844378627 scopus 로고    scopus 로고
    • Multidrug-resistant tuberculosis in Russia: Clinical characteristics, analysis of second-line drug resistance and development of standardized therapy
    • Balabanova Y, Ruddy M, Hubb J, et al. Multidrug-resistant tuberculosis in Russia: clinical characteristics, analysis of second-line drug resistance and development of standardized therapy. Eur J Clin Microbiol Infect Dis 2005; 24: 136-139.
    • (2005) Eur J Clin Microbiol Infect Dis , vol.24 , pp. 136-139
    • Balabanova, Y.1    Ruddy, M.2    Hubb, J.3
  • 33
    • 36749066063 scopus 로고    scopus 로고
    • Pyrrolidine dithiocarbamate and diethyldithiocarbamate are active against growing and nongrowing persister Mycobacterium tuberculosis
    • Byrne ST, Gu P, Zhou J, et al. Pyrrolidine dithiocarbamate and diethyldithiocarbamate are active against growing and nongrowing persister Mycobacterium tuberculosis. Antimicrob Agents Chemother 2007; 51: 4495-4497.
    • (2007) Antimicrob Agents Chemother , vol.51 , pp. 4495-4497
    • Byrne, S.T.1    Gu, P.2    Zhou, J.3
  • 34
    • 0025831020 scopus 로고
    • Enhancement of monocyte antimycobacterial activity by diethyldithiocarbamate (DTC)
    • Hübner L, Ernst M, von Laer D, et al. Enhancement of monocyte antimycobacterial activity by diethyldithiocarbamate (DTC). Int J Immunopharmacol 1991; 13: 1067-1072.
    • (1991) Int J Immunopharmacol , vol.13 , pp. 1067-1072
    • Hübner, L.1    Ernst, M.2    Von Laer, D.3
  • 35
    • 84864386765 scopus 로고    scopus 로고
    • Antitubercular activity of disulfiram, an antialcoholism drug, against multidrug-and extensively drug-resistant Mycobacterium tuberculosis isolates
    • Horita Y, Takii T, Yagi T, et al. Antitubercular activity of disulfiram, an antialcoholism drug, against multidrug-and extensively drug-resistant Mycobacterium tuberculosis isolates. Antimicrob Agents Chemother 2012; 56: 4140-4145.
    • (2012) Antimicrob Agents Chemother , vol.56 , pp. 4140-4145
    • Horita, Y.1    Takii, T.2    Yagi, T.3
  • 36
    • 0019790376 scopus 로고
    • A comparative review of the pharmacological and toxicological properties of disulfiram and calcium carbimide
    • Peachey JE, Brien JF, Roach CA, et al. A comparative review of the pharmacological and toxicological properties of disulfiram and calcium carbimide. J Clin Psychopharmacol 1981; 1: 21-26.
    • (1981) J Clin Psychopharmacol , vol.1 , pp. 21-26
    • Peachey, J.E.1    Brien, J.F.2    Roach, C.A.3
  • 38
    • 84863042675 scopus 로고    scopus 로고
    • Susceptibility of Mycobacterium tuberculosis to sulfamethoxazole, trimethoprim and their combination over a 12 year period in Taiwan
    • Huang TS, Kunin CM, Yan BS, et al. Susceptibility of Mycobacterium tuberculosis to sulfamethoxazole, trimethoprim and their combination over a 12 year period in Taiwan. J Antimicrob Chemother 2012; 67: 633-637.
    • (2012) J Antimicrob Chemother , vol.67 , pp. 633-637
    • Huang, T.S.1    Kunin, C.M.2    Yan, B.S.3
  • 39
    • 0023023318 scopus 로고
    • Susceptibility testing of slowly growing mycobacteria by a microdilution MIC method with 7H9 broth
    • Wallace RJ Jr, Nash DR, Steele LC, et al. Susceptibility testing of slowly growing mycobacteria by a microdilution MIC method with 7H9 broth. J Clin Microbiol 1986; 24: 976-981.
    • (1986) J Clin Microbiol , vol.24 , pp. 976-981
    • Wallace Jr., R.J.1    Nash, D.R.2    Steele, L.C.3
  • 40
    • 84866328705 scopus 로고    scopus 로고
    • The combination of sulfamethoxazole, trimethoprim, and isoniazid or rifampin is bactericidal and prevents the emergence of drug resistance in Mycobacterium tuberculosis
    • Vilchèze C, Jacobs WR Jr. The combination of sulfamethoxazole, trimethoprim, and isoniazid or rifampin is bactericidal and prevents the emergence of drug resistance in Mycobacterium tuberculosis. Antimicrob Agents Chemother 2012; 56: 5142-5148.
    • (2012) Antimicrob Agents Chemother , vol.56 , pp. 5142-5148
    • Vilchèze, C.1    Jacobs Jr., W.R.2
  • 41
    • 84869484254 scopus 로고    scopus 로고
    • Sulfamethoxazole enhances the antimycobacterial activity of rifampicin
    • Macingwana L, Baker B, Ngwane AH, et al. Sulfamethoxazole enhances the antimycobacterial activity of rifampicin. J Antimicrob Chemother 2012; 67: 2908-2911.
    • (2012) J Antimicrob Chemother , vol.67 , pp. 2908-2911
    • Macingwana, L.1    Baker, B.2    Ngwane, A.H.3
  • 42
    • 0018325009 scopus 로고
    • The pharmacokinetics of trimethoprim and trimethoprim/sulphonamide combinations, including penetration into body tissues
    • Reeves DS, Wilkinson PJ. The pharmacokinetics of trimethoprim and trimethoprim/sulphonamide combinations, including penetration into body tissues. Infection 1979; 7: Suppl. 4, S330-S341.
    • (1979) Infection , vol.7 , Issue.SUPPL. 4
    • Reeves, D.S.1    Wilkinson, P.J.2
  • 43
    • 0037416986 scopus 로고    scopus 로고
    • Clinical concentrations of thioridazine kill intracellular multidrugresistant Mycobacterium tuberculosis
    • Ordway D, Viveiros M, Leandro C, et al. Clinical concentrations of thioridazine kill intracellular multidrugresistant Mycobacterium tuberculosis. Antimicrob Agents Chemother 2003; 47: 917-922.
    • (2003) Antimicrob Agents Chemother , vol.47 , pp. 917-922
    • Ordway, D.1    Viveiros, M.2    Leandro, C.3
  • 44
    • 0035098674 scopus 로고    scopus 로고
    • Enhancement of antibiotic activity against poly-drug resistant Mycobacterium tuberculosis by phenothiazines
    • Viveiros M, Amaral L. Enhancement of antibiotic activity against poly-drug resistant Mycobacterium tuberculosis by phenothiazines. Int J Antimicrob Agents 2001; 17: 225-228.
    • (2001) Int J Antimicrob Agents , vol.17 , pp. 225-228
    • Viveiros, M.1    Amaral, L.2
  • 45
    • 0026441418 scopus 로고
    • Drug distribution between blood and brain as a determinant of antipsychotic drug effects
    • Tsuneizumi T, Babb SM, Cohen BM. Drug distribution between blood and brain as a determinant of antipsychotic drug effects. Biol Psychiatry 1992; 32: 817-824.
    • (1992) Biol Psychiatry , vol.32 , pp. 817-824
    • Tsuneizumi, T.1    Babb, S.M.2    Cohen, B.M.3
  • 46
    • 0018135058 scopus 로고
    • Binding of thioridazine and thioridazine metabolites to serum proteins in psychiatric patients
    • Nyberg G, Axelsson R, Martensson E. Binding of thioridazine and thioridazine metabolites to serum proteins in psychiatric patients. Eur J Clin Pharmacol 1978; 14: 341-350.
    • (1978) Eur J Clin Pharmacol , vol.14 , pp. 341-350
    • Nyberg, G.1    Axelsson, R.2    Martensson, E.3
  • 47
    • 78449274705 scopus 로고    scopus 로고
    • Drugs in development for tuberculosis
    • Ginsberg AM. Drugs in development for tuberculosis. Drugs 2010; 70: 2201-2214.
    • (2010) Drugs , vol.70 , pp. 2201-2214
    • Ginsberg, A.M.1
  • 48
    • 0029976980 scopus 로고    scopus 로고
    • An in vitro model for sequential study of shiftdown of Mycobacterium tuberculosis through two stages of nonreplicating persistence
    • Wayne LG, Hayes LG. An in vitro model for sequential study of shiftdown of Mycobacterium tuberculosis through two stages of nonreplicating persistence. Infect Immun 1996; 64: 2062-2069.
    • (1996) Infect Immun , vol.64 , pp. 2062-2069
    • Wayne, L.G.1    Hayes, L.G.2
  • 49
    • 0020521954 scopus 로고
    • Single-and multiple-dose metronidazole kinetics
    • Jensen JC, Gugler R. Single-and multiple-dose metronidazole kinetics. Clin Pharmacol Ther 1983; 34: 481-487.
    • (1983) Clin Pharmacol Ther , vol.34 , pp. 481-487
    • Jensen, J.C.1    Gugler, R.2
  • 50
    • 0024759118 scopus 로고
    • Role of metronidazole in improving response and specific drug sensitivity in advanced pulmonary tuberculosis
    • Desai CR, Heera S, Patel A, et al. Role of metronidazole in improving response and specific drug sensitivity in advanced pulmonary tuberculosis. J Assoc Physicians India 1989; 37: 694-697.
    • (1989) J Assoc Physicians India , vol.37 , pp. 694-697
    • Desai, C.R.1    Heera, S.2    Patel, A.3
  • 52
    • 22944432859 scopus 로고    scopus 로고
    • Tigecycline: A novel glycylcycline
    • Rubinstein E, Vaughan D. Tigecycline: a novel glycylcycline. Drugs 2005; 65: 1317-1336.
    • (2005) Drugs , vol.65 , pp. 1317-1336
    • Rubinstein, E.1    Vaughan, D.2
  • 53
    • 0036783671 scopus 로고    scopus 로고
    • Comparison of the in vitro activity of the glycylcycline tigecycline (formerly GAR-936) with those of tetracycline, minocycline, and doxycycline against isolates of nontuberculous mycobacteria
    • Wallace RJ Jr, Brown-Elliott BA, Crist CJ, et al. Comparison of the in vitro activity of the glycylcycline tigecycline (formerly GAR-936) with those of tetracycline, minocycline, and doxycycline against isolates of nontuberculous mycobacteria. Antimicrob Agents Chemother 2002; 46: 3164-3167.
    • (2002) Antimicrob Agents Chemother , vol.46 , pp. 3164-3167
    • Wallace Jr., R.J.1    Brown-Elliott, B.A.2    Crist, C.J.3
  • 54
    • 11244353707 scopus 로고    scopus 로고
    • Pharmacokinetics of tigecycline after single and multiple doses in healthy subjects
    • Muralidharan G, Micalizzi M, Speth J, et al. Pharmacokinetics of tigecycline after single and multiple doses in healthy subjects. Antimicrob Agents Chemother 2005; 49: 220-229.
    • (2005) Antimicrob Agents Chemother , vol.49 , pp. 220-229
    • Muralidharan, G.1    Micalizzi, M.2    Speth, J.3
  • 55
    • 84882601099 scopus 로고    scopus 로고
    • Evaluation of co-trimoxazole in the treatment of multidrug-resistant tuberculosis
    • Alsaad N, van Altena R, Pranger AD, et al. Evaluation of co-trimoxazole in the treatment of multidrug-resistant tuberculosis. Eur Respir J 2013; 42: 504-512.
    • (2013) Eur Respir J , vol.42 , pp. 504-512
    • Alsaad, N.1    Van Altena, R.2    Pranger, A.D.3
  • 58
    • 84855829764 scopus 로고    scopus 로고
    • Successful alternative treatment of extensively drug-resistant tuberculosis in Argentina with a combination of linezolid, moxifloxacin and thioridazine
    • Abbate E, Vescovo M, Natiello M, et al. Successful alternative treatment of extensively drug-resistant tuberculosis in Argentina with a combination of linezolid, moxifloxacin and thioridazine. J Antimicrob Chemother 2012; 67: 473-477.
    • (2012) J Antimicrob Chemother , vol.67 , pp. 473-477
    • Abbate, E.1    Vescovo, M.2    Natiello, M.3
  • 59
    • 81555214621 scopus 로고    scopus 로고
    • Phenothiazines as anti-tubercular agents: Mechanistic insights and clinical implications
    • Sharma S, Singh A. Phenothiazines as anti-tubercular agents: mechanistic insights and clinical implications. Expert Opin Investig Drugs 2011; 20: 1665-1676.
    • (2011) Expert Opin Investig Drugs , vol.20 , pp. 1665-1676
    • Sharma, S.1    Singh, A.2
  • 60
    • 11844292801 scopus 로고    scopus 로고
    • Antimicrobial activity of phenothiazines
    • Amaral L, Viveiros M, Molnar J. Antimicrobial activity of phenothiazines. In Vivo 2004; 18: 725-731.
    • (2004) Vivo , vol.18 , pp. 725-731
    • Amaral, L.1    Viveiros, M.2    Molnar, J.3
  • 61
    • 84859428822 scopus 로고    scopus 로고
    • Why thioridazine in combination with antibiotics cures extensively drug-resistant Mycobacterium tuberculosis infections
    • Amaral L, Viveiros M. Why thioridazine in combination with antibiotics cures extensively drug-resistant Mycobacterium tuberculosis infections. Int J Antimicrob Agents 2012; 39: 376-380.
    • (2012) Int J Antimicrob Agents , vol.39 , pp. 376-380
    • Amaral, L.1    Viveiros, M.2
  • 62
    • 33344460427 scopus 로고    scopus 로고
    • Characterization of human cytochrome p450 enzymes involved in the metabolism of the piperidine-type phenothiazine neuroleptic thioridazine
    • Wójcikowski J, Maurel P, Daniel WA. Characterization of human cytochrome p450 enzymes involved in the metabolism of the piperidine-type phenothiazine neuroleptic thioridazine. Drug Metab Dispos 2006; 34: 471-476.
    • (2006) Drug Metab Dispos , vol.34 , pp. 471-476
    • Wójcikowski, J.1    Maurel, P.2    Daniel, W.A.3
  • 63
    • 77950849122 scopus 로고    scopus 로고
    • Thioridazine cures extensively drug-resistant tuberculosis (XDR-TB) and the need for global trials is now!
    • Amaral L, Boeree MJ, Gillespie SH, et al. Thioridazine cures extensively drug-resistant tuberculosis (XDR-TB) and the need for global trials is now!. Int J Antimicrob Agents 2010; 35: 524-526.
    • (2010) Int J Antimicrob Agents , vol.35 , pp. 524-526
    • Amaral, L.1    Boeree, M.J.2    Gillespie, S.H.3
  • 64
    • 38649084124 scopus 로고    scopus 로고
    • Cardiac side effects of psychiatric drugs
    • Mackin P. Cardiac side effects of psychiatric drugs. Hum Psychopharmacol 2008; 23: Suppl. 1, 3-14.
    • (2008) Hum Psychopharmacol , vol.23 , Issue.SUPPL. 1 , pp. 3-14
    • Mackin, P.1
  • 65
    • 21344462866 scopus 로고    scopus 로고
    • The in vitro activity of phenothiazines against Mycobacterium avium: Potential of thioridazine for therapy of the co-infected AIDS patient
    • Viveiros M, Martins M, Couto I, et al. The in vitro activity of phenothiazines against Mycobacterium avium: potential of thioridazine for therapy of the co-infected AIDS patient. In Vivo 2005; 19: 733-736.
    • (2005) Vivo , vol.19 , pp. 733-736
    • Viveiros, M.1    Martins, M.2    Couto, I.3
  • 66
    • 0018707163 scopus 로고
    • Mechanism of antimicrobial action of metronidazole
    • Edwards DI. Mechanism of antimicrobial action of metronidazole. J Antimicrob Chemother 1979; 5: 499-502.
    • (1979) J Antimicrob Chemother , vol.5 , pp. 499-502
    • Edwards, D.I.1
  • 67
    • 0031442875 scopus 로고    scopus 로고
    • Progression of chronic pulmonary tuberculosis in mice aerogenically infected with virulent Mycobacterium tuberculosis
    • Rhoades ER, Frank AA, Orme IM. Progression of chronic pulmonary tuberculosis in mice aerogenically infected with virulent Mycobacterium tuberculosis. Tuber Lung Dis 1997; 78: 57-66.
    • (1997) Tuber Lung Dis , vol.78 , pp. 57-66
    • Rhoades, E.R.1    Frank, A.A.2    Orme, I.M.3
  • 68
    • 0018140266 scopus 로고
    • Pharmacokinetics and therapeutic efficacy of metronidazole at different dosages
    • Amon I, Amon K, Hüller H. Pharmacokinetics and therapeutic efficacy of metronidazole at different dosages. Int J Clin Pharmacol Biopharm 1978; 16: 384-386.
    • (1978) Int J Clin Pharmacol Biopharm , vol.16 , pp. 384-386
    • Amon, I.1    Amon, K.2    Hüller, H.3
  • 69
    • 0020401715 scopus 로고
    • Activity of metronidazole and its hydroxy and acid metabolites against clinical isolates of anaerobic bacteria
    • O'Keefe JP, Troc KA, Thompson KD. Activity of metronidazole and its hydroxy and acid metabolites against clinical isolates of anaerobic bacteria. Antimicrob Agents Chemother 1982; 22: 426-430.
    • (1982) Antimicrob Agents Chemother , vol.22 , pp. 426-430
    • O'keefe, J.P.1    Troc, K.A.2    Thompson, K.D.3
  • 70
    • 0016798872 scopus 로고
    • Bioassay of metronidazole with either anaerobic or aerobic incubation
    • Ralph ED, Kirby WM. Bioassay of metronidazole with either anaerobic or aerobic incubation. J Infect Dis 1975; 132: 587-591.
    • (1975) J Infect Dis , vol.132 , pp. 587-591
    • Ralph, E.D.1    Kirby, W.M.2
  • 71
    • 0016914401 scopus 로고
    • Comparative pharmacokinetic studies of ornidazole and metronidazole in man
    • Schwartz DE, Jeunet F. Comparative pharmacokinetic studies of ornidazole and metronidazole in man. Chemotherapy 1976; 22: 19-29.
    • (1976) Chemotherapy , vol.22 , pp. 19-29
    • Schwartz, D.E.1    Jeunet, F.2
  • 72
    • 84895540772 scopus 로고    scopus 로고
    • ClinicalTrials.gov identifier: NCT00425113, Date last updated: October 21, 2013
    • Clinicaltrials.gov.Metronidazole for pulmonary tuberculosis (South Korea). ClinicalTrials.gov identifier: NCT00425113. http://clinicaltrials.gov/ show/NCT00425113 Date last updated: October 21, 2013.
    • Metronidazole for Pulmonary Tuberculosis (South Korea)
  • 73
  • 74
    • 33646136687 scopus 로고    scopus 로고
    • Matrix metalloproteinase inhibitors as prospective agents for the prevention and treatment of cardiovascular and neoplastic diseases
    • Sang QX, Jin Y, Newcomer RG, et al. Matrix metalloproteinase inhibitors as prospective agents for the prevention and treatment of cardiovascular and neoplastic diseases. Curr Top Med Chem 2006; 6: 289-316.
    • (2006) Curr Top Med Chem , vol.6 , pp. 289-316
    • Sang, Q.X.1    Jin, Y.2    Newcomer, R.G.3
  • 75
    • 65549151744 scopus 로고    scopus 로고
    • Farmakokinetika tetracyklinu a glycylcyklinu [Pharmacokinetics of tetracyclines and glycylcyclines]
    • Vojtova V, Urbanek K. Farmakokinetika tetracyklinu a glycylcyklinu [Pharmacokinetics of tetracyclines and glycylcyclines]. Klin Mikrobiol Infekc Lek 2009; 15: 17-21.
    • (2009) Klin Mikrobiol Infekc Lek , vol.15 , pp. 17-21
    • Vojtova, V.1    Urbanek, K.2
  • 76
    • 23844496128 scopus 로고    scopus 로고
    • Tigecycline: A new glycylcycline for treatment of serious infections
    • Noskin GA. Tigecycline: a new glycylcycline for treatment of serious infections. Clin Infect Dis 2005; 41: Suppl. 5, S303-S314.
    • (2005) Clin Infect Dis , vol.41 , Issue.SUPPL. 5
    • Noskin, G.A.1
  • 77
    • 27744585664 scopus 로고    scopus 로고
    • Safety of doxycycline and minocycline: A systematic review
    • Smith K, Leyden JJ. Safety of doxycycline and minocycline: a systematic review. Clin Ther 2005; 27: 1329-1342.
    • (2005) Clin Ther , vol.27 , pp. 1329-1342
    • Smith, K.1    Leyden, J.J.2
  • 78
    • 84874604544 scopus 로고    scopus 로고
    • Dithiocarbamates strongly inhibit the b-class carbonic anhydrases from Mycobacterium tuberculosis
    • Maresca A, Carta F, Vullo D, et al. Dithiocarbamates strongly inhibit the b-class carbonic anhydrases from Mycobacterium tuberculosis. J Enzyme Inhib Med Chem 2013; 28: 407-411.
    • (2013) J Enzyme Inhib Med Chem , vol.28 , pp. 407-411
    • Maresca, A.1    Carta, F.2    Vullo, D.3
  • 79
    • 69949170494 scopus 로고    scopus 로고
    • Effect of 1, 25 dihydroxyvitamin D3 on matrix metalloproteinases MMP-7, MMP-9 and the inhibitor TIMP-1 in pulmonary tuberculosis
    • Anand SP, Selvaraj P. Effect of 1, 25 dihydroxyvitamin D3 on matrix metalloproteinases MMP-7, MMP-9 and the inhibitor TIMP-1 in pulmonary tuberculosis. Clin Immunol 2009; 133: 126-131.
    • (2009) Clin Immunol , vol.133 , pp. 126-131
    • Anand, S.P.1    Selvaraj, P.2
  • 80
    • 33645224419 scopus 로고    scopus 로고
    • Toll-like receptor triggering of a vitamin D-mediated human antimicrobial response
    • Liu PT, Stenger S, Li H, et al. Toll-like receptor triggering of a vitamin D-mediated human antimicrobial response. Science 2006; 311: 1770-1773.
    • (2006) Science , vol.311 , pp. 1770-1773
    • Liu, P.T.1    Stenger, S.2    Li, H.3
  • 81
    • 0032897832 scopus 로고    scopus 로고
    • Safety issues concerning the use of disulfiram in treating alcohol dependence
    • Chick J. Safety issues concerning the use of disulfiram in treating alcohol dependence. Drug Saf 1999; 20: 427-435.
    • (1999) Drug Saf , vol.20 , pp. 427-435
    • Chick, J.1
  • 82
    • 33644508373 scopus 로고    scopus 로고
    • Dihydrofolate reductase inhibitors as antibacterial agents
    • Hawser S, Lociuro S, Islam K. Dihydrofolate reductase inhibitors as antibacterial agents. Biochem Pharmacol 2006; 71: 941-948.
    • (2006) Biochem Pharmacol , vol.71 , pp. 941-948
    • Hawser, S.1    Lociuro, S.2    Islam, K.3
  • 83
    • 77952880349 scopus 로고    scopus 로고
    • The HIV-associated tuberculosis epidemic-when will we act?
    • Harries AD, Zachariah R, Corbett EL, et al. The HIV-associated tuberculosis epidemic-when will we act? Lancet 2010; 375: 1906-1919.
    • (2010) Lancet , vol.375 , pp. 1906-1919
    • Harries, A.D.1    Zachariah, R.2    Corbett, E.L.3
  • 84
    • 0032444693 scopus 로고    scopus 로고
    • Susceptibilities of Mycobacterium tuberculosis and Mycobacterium avium complex to lipophilic deazapteridine derivatives, inhibitors of dihydrofolate reductase
    • Suling WJ, Reynolds RC, Barrow EW, et al. Susceptibilities of Mycobacterium tuberculosis and Mycobacterium avium complex to lipophilic deazapteridine derivatives, inhibitors of dihydrofolate reductase. J Antimicrob Chemother 1998; 42: 811-815.
    • (1998) J Antimicrob Chemother , vol.42 , pp. 811-815
    • Suling, W.J.1    Reynolds, R.C.2    Barrow, E.W.3
  • 85
    • 0019214479 scopus 로고
    • Clinical pharmacokinetics of co-trimoxazole (trimethoprim- sulphamethoxazole)
    • Patel RB, Welling PG. Clinical pharmacokinetics of co-trimoxazole (trimethoprim-sulphamethoxazole). Clin Pharmacokinet 1980; 5: 405-423.
    • (1980) Clin Pharmacokinet , vol.5 , pp. 405-423
    • Patel, R.B.1    Welling, P.G.2
  • 87
    • 0033033406 scopus 로고    scopus 로고
    • Trimethoprim-sulfamethoxazole
    • Smilack JD. Trimethoprim-sulfamethoxazole. Mayo Clin Proc 1999; 74: 730-734.
    • (1999) Mayo Clin Proc , vol.74 , pp. 730-734
    • Smilack, J.D.1
  • 88
    • 0033135568 scopus 로고    scopus 로고
    • Efficacy of trimethoprim-sulphamethoxazole prophylaxis to decrease morbidity and mortality in HIV-1-infected patients with tuberculosis in Abidjan, Cô te d'Ivoire: A randomised controlled trial
    • Wiktor SZ, Sassan-Morokro M, Grant AD, et al. Efficacy of trimethoprim-sulphamethoxazole prophylaxis to decrease morbidity and mortality in HIV-1-infected patients with tuberculosis in Abidjan, Cô te d'Ivoire: a randomised controlled trial. Lancet 1999; 353: 1469-1475.
    • (1999) Lancet , vol.353 , pp. 1469-1475
    • Wiktor, S.Z.1    Sassan-Morokro, M.2    Grant, A.D.3
  • 89
    • 2642558026 scopus 로고    scopus 로고
    • Cotrimoxazole prophylaxis reduces mortality in human immunodeficiency virus-positive tuberculosis patients in Karonga District, Malawi
    • Mwaungulu FB, Floyd S, Crampin AC, et al. Cotrimoxazole prophylaxis reduces mortality in human immunodeficiency virus-positive tuberculosis patients in Karonga District, Malawi. Bull World Health Organ 2004; 82: 354-363.
    • (2004) Bull World Health Organ , vol.82 , pp. 354-363
    • Mwaungulu, F.B.1    Floyd, S.2    Crampin, A.C.3
  • 90
    • 0037463683 scopus 로고    scopus 로고
    • Trimethoprim-sulfamethoxazole revisited
    • Masters PA, O'Bryan TA, Zurlo J, et al. Trimethoprim-sulfamethoxazole revisited. Arch InternMed 2003; 163: 402-410.
    • (2003) Arch InternMed , vol.163 , pp. 402-410
    • Masters, P.A.1    O'bryan, T.A.2    Zurlo, J.3
  • 91
    • 0042975077 scopus 로고    scopus 로고
    • Hyponatremia and/or hyperkalemia in patients treated with the standard dose of trimethoprim-sulfamethoxazole
    • Mori H, Kuroda Y, Imamura S, et al. Hyponatremia and/or hyperkalemia in patients treated with the standard dose of trimethoprim-sulfamethoxazole. Intern Med 2003; 42: 665-669.
    • (2003) Intern Med , vol.42 , pp. 665-669
    • Mori, H.1    Kuroda, Y.2    Imamura, S.3
  • 92
    • 0023511693 scopus 로고
    • Hematological side effects of co-trimoxazole
    • Heimpel H, Raghavachar A. Hematological side effects of co-trimoxazole. Infection 1987; 15: Suppl. 5, S248-S253.
    • (1987) Infection , vol.15 , Issue.SUPPL. 5
    • Heimpel, H.1    Raghavachar, A.2
  • 93
    • 0033986977 scopus 로고    scopus 로고
    • Use of genomics and combinatorial chemistry in the development of new antimycobacterial drugs
    • Barry CE 3rd, Slayden RA, Sampson AE, et al. Use of genomics and combinatorial chemistry in the development of new antimycobacterial drugs. Biochem Pharmacol 2000; 59: 221-231.
    • (2000) Biochem Pharmacol , vol.59 , pp. 221-231
    • Barry III, C.E.1    Slayden, R.A.2    Sampson, A.E.3


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