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Volumn 85, Issue 2, 2014, Pages 381-387

Sidedness of carbamazepine accessibility to voltage-gated sodium channels

Author keywords

[No Author keywords available]

Indexed keywords

CARBAMAZEPINE; LIDOCAINE ETHOBROMIDE; SODIUM CHANNEL NAV1.7;

EID: 84891855693     PISSN: 0026895X     EISSN: 15210111     Source Type: Journal    
DOI: 10.1124/mol.113.090472     Document Type: Article
Times cited : (30)

References (24)
  • 2
    • 0014704033 scopus 로고
    • The site of action and active form of local anesthetics II Experiments with quaternary compounds
    • Frazier DT, Narahashi T, and Yamada M (1970) The site of action and active form of local anesthetics. II. Experiments with quaternary compounds. J Pharmacol Exp Ther 171:45-51.
    • (1970) J Pharmacol Exp Ther , vol.171 , pp. 45-51
    • Frazier, D.T.1    Narahashi, T.2    Yamada, M.3
  • 3
    • 0017350085 scopus 로고
    • The pH-dependent rate of action of local anesthetics on the node of Ranvier
    • Hille B (1977a) The pH-dependent rate of action of local anesthetics on the node of Ranvier. J Gen Physiol 69:475-496.
    • (1977) J Gen Physiol , vol.69 , pp. 475-496
    • Hille, B.1
  • 4
    • 0017332486 scopus 로고
    • Local anesthetics: Hydrophilic and hydrophobic pathways for the drug-receptor reaction
    • Hille B (1977b) Local anesthetics: hydrophilic and hydrophobic pathways for the drug-receptor reaction. J Gen Physiol 69:497-515.
    • (1977) J Gen Physiol , vol.69 , pp. 497-515
    • Hille, B.1
  • 6
    • 0031754721 scopus 로고    scopus 로고
    • A common anticonvulsant binding site for phenytoin, carbamazepine, and lamotrigine in neuronal Na1 channels
    • Kuo CC (1998) A common anticonvulsant binding site for phenytoin, carbamazepine, and lamotrigine in neuronal Na1 channels. Mol Pharmacol 54:712-721.
    • (1998) Mol Pharmacol , vol.54 , pp. 712-721
    • Kuo, C.C.1
  • 7
    • 0030949912 scopus 로고    scopus 로고
    • Carbamazepine inhibition of neuronal Na1 currents: Quantitative distinction from phenytoin and possible therapeutic implications
    • Kuo CC, Chen RS, Lu L, and Chen RC (1997) Carbamazepine inhibition of neuronal Na1 currents: quantitative distinction from phenytoin and possible therapeutic implications. Mol Pharmacol 51:1077-1083.
    • (1997) Mol Pharmacol , vol.51 , pp. 1077-1083
    • Kuo, C.C.1    Chen, R.S.2    Lu, L.3    Chen, R.C.4
  • 8
    • 27844589940 scopus 로고    scopus 로고
    • Molecular modeling of local anesthetic drug binding by voltage-gated sodium channels
    • Lipkind GM and Fozzard HA (2005) Molecular modeling of local anesthetic drug binding by voltage-gated sodium channels. Mol Pharmacol 68:1611-1622.
    • (2005) Mol Pharmacol , vol.68 , pp. 1611-1622
    • Lipkind, G.M.1    Fozzard, H.A.2
  • 9
    • 77957223212 scopus 로고    scopus 로고
    • Molecular model of anticonvulsant drug binding to the voltage-gated sodium channel inner pore
    • Lipkind GM and Fozzard HA (2010) Molecular model of anticonvulsant drug binding to the voltage-gated sodium channel inner pore. Mol Pharmacol 78:631-638.
    • (2010) Mol Pharmacol , vol.78 , pp. 631-638
    • Lipkind, G.M.1    Fozzard, H.A.2
  • 10
    • 84861881276 scopus 로고    scopus 로고
    • Modulation of neuronal sodium channels by the sea anemone peptide BDS-I
    • Liu P, Jo S, and Bean BP (2012) Modulation of neuronal sodium channels by the sea anemone peptide BDS-I. J Neurophysiol 107:3155-3167.
    • (2012) J Neurophysiol , vol.107 , pp. 3155-3167
    • Liu, P.1    Jo, S.2    Bean, B.P.3
  • 11
    • 79960621367 scopus 로고    scopus 로고
    • The crystal structure of a voltage-gated sodium channel
    • Payandeh J, Scheuer T, Zheng N, and Catterall WA (2011) The crystal structure of a voltage-gated sodium channel. Nature 475:353-358.
    • (2011) Nature , vol.475 , pp. 353-358
    • Payandeh, J.1    Scheuer, T.2    Zheng, N.3    Catterall, W.A.4
  • 12
    • 0025827588 scopus 로고
    • Frequency and voltage-dependent inhibition of type IIA Na1 channels, expressed in a mammalian cell line, by local anesthetic, antiarrhythmic, and anticonvulsant drugs
    • Ragsdale DS, Scheuer T, and Catterall WA (1991) Frequency and voltage-dependent inhibition of type IIA Na1 channels, expressed in a mammalian cell line, by local anesthetic, antiarrhythmic, and anticonvulsant drugs. Mol Pharmacol 40:756-765.
    • (1991) Mol Pharmacol , vol.40 , pp. 756-765
    • Ragsdale, D.S.1    Scheuer, T.2    Catterall, W.A.3
  • 13
    • 0027944683 scopus 로고
    • Molecular determinants of state-dependent block of Na1 channels by local anesthetics
    • Ragsdale DS, McPhee JC, Scheuer T, and Catterall WA (1994) Molecular determinants of state-dependent block of Na1 channels by local anesthetics. Science 265: 1724-1728.
    • (1994) Science , vol.265 , pp. 1724-1728
    • Ragsdale, D.S.1    McPhee, J.C.2    Scheuer, T.3    Catterall, W.A.4
  • 14
    • 0029787945 scopus 로고    scopus 로고
    • Common molecular determinants of local anesthetic, antiarrhythmic, and anticonvulsant block of voltage-gated Na1 channels
    • Ragsdale DS, McPhee JC, Scheuer T, and Catterall WA (1996) Common molecular determinants of local anesthetic, antiarrhythmic, and anticonvulsant block of voltage-gated Na1 channels. Proc Natl Acad Sci USA 93:9270-9275.
    • (1996) Proc Natl Acad Sci USA , vol.93 , pp. 9270-9275
    • Ragsdale, D.S.1    McPhee, J.C.2    Scheuer, T.3    Catterall, W.A.4
  • 15
    • 3042798891 scopus 로고    scopus 로고
    • The neurobiology of antiepileptic drugs
    • Rogawski MA and Löscher W (2004) The neurobiology of antiepileptic drugs. Nat Rev Neurosci 5:553-564.
    • (2004) Nat Rev Neurosci , vol.5 , pp. 553-564
    • Rogawski, M.A.1    Löscher, W.2
  • 16
    • 0017746139 scopus 로고
    • Local anesthetics effect of ph on usedependent block of sodium channels in frog muscle
    • Schwarz W, Palade PT, and Hille B (1977) Local anesthetics. Effect of pH on usedependent block of sodium channels in frog muscle. Biophys J 20:343-368.
    • (1977) Biophys J , vol.20 , pp. 343-368
    • Schwarz, W.1    Palade, P.T.2    Hille, B.3
  • 17
    • 45749155596 scopus 로고    scopus 로고
    • Differential block of sensory neuronal voltage-gated sodium channels by lacosamide [(2R)-2-(acetylamino)-Nbenzyl- 3-methoxypropanamide], lidocaine, and carbamazepine
    • Sheets PL, Heers C, Stoehr T, and Cummins TR (2008) Differential block of sensory neuronal voltage-gated sodium channels by lacosamide [(2R)-2-(acetylamino)-Nbenzyl- 3-methoxypropanamide], lidocaine, and carbamazepine. J Pharmacol Exp Ther 326:89-99.
    • (2008) J Pharmacol Exp Ther , vol.326 , pp. 89-99
    • Sheets, P.L.1    Heers, C.2    Stoehr, T.3    Cummins, T.R.4
  • 18
    • 0015784454 scopus 로고
    • The inhibition of sodium currents in myelinated nerve by quaternary derivatives of lidocaine
    • Strichartz GR (1973) The inhibition of sodium currents in myelinated nerve by quaternary derivatives of lidocaine. J Gen Physiol 62:37-57.
    • (1973) J Gen Physiol , vol.62 , pp. 37-57
    • Strichartz, G.R.1
  • 19
    • 80053185917 scopus 로고    scopus 로고
    • Inhibition of Navb4 peptide-mediated resurgent sodium currents in Nav1.7 channels by carbamazepine, riluzole, and anandamide
    • Theile JW and Cummins TR (2011) Inhibition of Navb4 peptide-mediated resurgent sodium currents in Nav1.7 channels by carbamazepine, riluzole, and anandamide. Mol Pharm 80:724-734.
    • (2011) Mol Pharm , vol.80 , pp. 724-734
    • Theile, J.W.1    Cummins, T.R.2
  • 20
    • 13444269678 scopus 로고    scopus 로고
    • A multifunctional aromatic residue in the external pore vestibule of Na1 channels contributes to the local anesthetic receptor
    • Tsang SY, Tsushima RG, Tomaselli GF, Li RA, and Backx PH (2005) A multifunctional aromatic residue in the external pore vestibule of Na1 channels contributes to the local anesthetic receptor. Mol Pharmacol 67:424-434.
    • (2005) Mol Pharmacol , vol.67 , pp. 424-434
    • Tsang, S.Y.1    Tsushima, R.G.2    Tomaselli, G.F.3    Li, R.A.4    Backx, P.H.5
  • 21
    • 0021913947 scopus 로고
    • Voltage clamp analysis of the inhibitory actions of diphenylhydantoin and carbamazepine on voltage-sensitive sodium channels in neuroblastoma cells
    • Willow M, Gonoi T, and Catterall WA (1985) Voltage clamp analysis of the inhibitory actions of diphenylhydantoin and carbamazepine on voltage-sensitive sodium channels in neuroblastoma cells. Mol Pharmacol 27:549-558.
    • (1985) Mol Pharmacol , vol.27 , pp. 549-558
    • Willow, M.1    Gonoi, T.2    Catterall, W.A.3
  • 22
    • 77954175713 scopus 로고    scopus 로고
    • Lidocaine, carbamazepine, and imipramine have partially overlapping binding sites and additive inhibitory effect on neuronal Na1 channels
    • Yang YC, Huang CS, and Kuo CC (2010) Lidocaine, carbamazepine, and imipramine have partially overlapping binding sites and additive inhibitory effect on neuronal Na1 channels. Anesthesiology 113:160-174.
    • (2010) Anesthesiology , vol.113 , pp. 160-174
    • Yang, Y.C.1    Huang, C.S.2    Kuo, C.C.3
  • 23
    • 0035808309 scopus 로고    scopus 로고
    • Molecular determinants of voltage-dependent gating and binding of pore-blocking drugs in transmembrane segment IIIS6 of the Na(1) channel alpha subunit
    • Yarov-Yarovoy V, Brown J, Sharp EM, Clare JJ, Scheuer T, and Catterall WA (2001) Molecular determinants of voltage-dependent gating and binding of pore-blocking drugs in transmembrane segment IIIS6 of the Na(1) channel alpha subunit. J Biol Chem 276:20-27.
    • (2001) J Biol Chem , vol.276 , pp. 20-27
    • Yarov-Yarovoy, V.1    Brown, J.2    Sharp, E.M.3    Clare, J.J.4    Scheuer, T.5    Catterall, W.A.6
  • 24
    • 0037144493 scopus 로고    scopus 로고
    • Role of amino acid residues in transmembrane segments IS6 and IIS6 of the Na1 channel alpha subunit in voltage-dependent gating and drug block
    • Yarov-Yarovoy V, McPhee JC, Idsvoog D, Pate C, Scheuer T, and Catterall WA (2002) Role of amino acid residues in transmembrane segments IS6 and IIS6 of the Na1 channel alpha subunit in voltage-dependent gating and drug block. J Biol Chem 277:35393-35401.
    • (2002) J Biol Chem , vol.277 , pp. 35393-35401
    • Yarov-Yarovoy, V.1    McPhee, J.C.2    Idsvoog, D.3    Pate, C.4    Scheuer, T.5    Catterall, W.A.6


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.