Plasmodium gametocyte inhibition identified from a natural-product-based fragment library

ACS Chemical Biology

Volumn 8, Issue 12, 2013, Pages 2654-2659

  Vu, Hoan ^a   Roullier, Catherine ^a   Campitelli, Marc ^a   Trenholme, Katharine R ^b,c   Gardiner, Donald L ^b   Andrews, Katherine T ^a   Skinner Adams, Tina ^a   Crowther, Gregory J ^d   Van Voorhis, Wesley C ^d   Quinn, Ronald J ^a  

^a GRIFFITH UNIVERSITY   (Australia)

^b QIMR BERGHOFER MEDICAL RESEARCH INSTITUTE   (Australia)

^c UNIVERSITY OF QUEENSLAND   (Australia)

^d UNIVERSITY OF WASHINGTON   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

DEOXYURIDINE TRIPHOSPHATE PYROPHOSPHATASE; NATURAL PRODUCT; SECURININE;

ARTICLE; CONTROLLED STUDY; ENZYME ACTIVITY; GAMETOCYTE; MASS SPECTROMETRY; NONHUMAN; PLASMODIUM; PLASMODIUM FALCIPARUM; PRIORITY JOURNAL;

ALKALOIDS; ANTIMALARIALS; AZEPINES; BIOLOGICAL PRODUCTS; DEOXYURACIL NUCLEOTIDES; DOSE-RESPONSE RELATIONSHIP, DRUG; HETEROCYCLIC COMPOUNDS, BRIDGED-RING; KINETICS; LACTONES; LIFE CYCLE STAGES; PIPERIDINES; PLASMODIUM FALCIPARUM; PROTOZOAN PROTEINS; RECOMBINANT FUSION PROTEINS; SMALL MOLECULE LIBRARIES; SPECTROMETRY, MASS, ELECTROSPRAY IONIZATION; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 84890854772     PISSN: 15548929     EISSN: 15548937     Source Type: Journal    
DOI: 10.1021/cb400582b     Document Type: Article

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