메뉴 건너뛰기




Volumn 6, Issue , 2013, Pages 75-79

Atypical mechanism of glucose modulation by colesevelam in patients with type 2 diabetes

Author keywords

Colesevelam; Pharmacology; Type 2 diabetes mellitus

Indexed keywords

2,4 THIAZOLIDINEDIONE DERIVATIVE; ADIPONECTIN; ALPHA GLUCOSIDASE INHIBITOR; BILE ACID; COLESEVELAM; DIPEPTIDYL PEPTIDASE IV INHIBITOR; FARNESOID X RECEPTOR; FATTY ACID; G PROTEIN COUPLED RECEPTOR; GLUCAGON LIKE PEPTIDE 1 DERIVATIVE; INCRETIN; INSULIN DERIVATIVE; MEGLITINIDE; METFORMIN; PLACEBO; ROSIGLITAZONE; SITAGLIPTIN; SULFONYLUREA; TGR5 PROTEIN; UNCLASSIFIED DRUG;

EID: 84890085853     PISSN: 11795514     EISSN: 11795514     Source Type: Journal    
DOI: 10.4137/CMed.s12590     Document Type: Article
Times cited : (25)

References (38)
  • 1
    • 84855539606 scopus 로고    scopus 로고
    • AACE Task Force for Developing Diabetes Comprehensive Care Plan. American Association of Clinical Endocrinologists Medical Guidelines for Clinical Practice for developing a diabetes mellitus comprehensive care plan
    • Handelsman Y, Mechanick JI, Blonde L, et al. AACE Task Force for Developing Diabetes Comprehensive Care Plan. American Association of Clinical Endocrinologists Medical Guidelines for Clinical Practice for developing a diabetes mellitus comprehensive care plan. Endocr Pract. 2011;17 Suppl 2:1-53.
    • (2011) Endocr Pract , vol.17 , Issue.SUPPL. 2 , pp. 1-53
    • Handelsman, Y.1    Mechanick, J.I.2    Blonde, L.3
  • 2
    • 84866268783 scopus 로고    scopus 로고
    • Management of hyperglycemia in type 2 diabetes: A patient-centered approach. Position statement of the American Diabetes Association (ADA) and the European Association for the Study of Diabetes (EASD)
    • Inzucchi SE, Bergenstal RM, Buse JB, et al. Management of hyperglycemia in type 2 diabetes: a patient-centered approach. Position statement of the American Diabetes Association (ADA) and the European Association for the Study of Diabetes (EASD). Diabetes Care. 2012;35(6):1364-1379.
    • (2012) Diabetes Care , vol.35 , Issue.6 , pp. 1364-1379
    • Inzucchi, S.E.1    Bergenstal, R.M.2    Buse, J.B.3
  • 3
    • 23044439087 scopus 로고    scopus 로고
    • Efects of colesevelam HCl on sterol and bile acid excretion in patients with type IIa hypercholesterolemia
    • Donovan JM, Von Bergmann K, Setchell KDR, et al. Efects of colesevelam HCl on sterol and bile acid excretion in patients with type IIa hypercholesterolemia. Dig Dis Sci. 2005;50(7):1232-1238.
    • (2005) Dig Dis Sci , vol.50 , Issue.7 , pp. 1232-1238
    • Donovan, J.M.1    von Bergmann, K.2    Setchell, K.D.R.3
  • 5
    • 84874031840 scopus 로고    scopus 로고
    • Colesevelam suppresses hepatic glycogenolysis by TGR5-mediated induction of GLP-1 action in DIO mice
    • Potthof MJ, Potts A, He T, et al. Colesevelam suppresses hepatic glycogenolysis by TGR5-mediated induction of GLP-1 action in DIO mice. Am J Physiol Gas-trointest Liver Physiol. 2013;304(4):G371-G380.
    • (2013) Am J Physiol Gas-trointest Liver Physiol , vol.304 , Issue.4
    • Potthof, M.J.1    Potts, A.2    He, T.3
  • 6
    • 77249142314 scopus 로고    scopus 로고
    • Colesevelam improves insulin resistance in a diet-induced obesity (F-DIO) rat model by increasing the release of GLP-1
    • Shang Q, Saumoy M, Holst JJ, Salen G, Xu G. Colesevelam improves insulin resistance in a diet-induced obesity (F-DIO) rat model by increasing the release of GLP-1. Am J Physiol Gastrointest Liver Physiol. 2010;298(3):G419-G424.
    • (2010) Am J Physiol Gastrointest Liver Physiol , vol.298 , Issue.3
    • Shang, Q.1    Saumoy, M.2    Holst, J.J.3    Salen, G.4    Xu, G.5
  • 7
    • 80455126992 scopus 로고    scopus 로고
    • Bile acid sequestration reduces plasma glucose levels in db/db mice by increasing its metabolic clearance rate
    • Meissner M, Herrema H, van Dijk TH, et al. Bile acid sequestration reduces plasma glucose levels in db/db mice by increasing its metabolic clearance rate. PLoS One. 2011;6(11):e24564.
    • (2011) PLoS One , vol.6 , Issue.11
    • Meissner, M.1    Herrema, H.2    van Dijk, T.H.3
  • 8
    • 79960838523 scopus 로고    scopus 로고
    • Farnesoid X receptor defciency improves glucose homeostasis in mouse models of obesity
    • Prawitt J, Abdelkarim M, Stroeve JHM, et al. Farnesoid X receptor defciency improves glucose homeostasis in mouse models of obesity. Diabetes. 2011;60(7): 1861-1871.
    • (2011) Diabetes , vol.60 , Issue.7 , pp. 1861-1871
    • Prawitt, J.1    Abdelkarim, M.2    Stroeve, J.H.M.3
  • 10
    • 0037283601 scopus 로고    scopus 로고
    • Te relative contributions of insulin resistance and beta-cell dysfunction to the pathophysiology of Type 2 diabetes
    • Kahn SE. Te relative contributions of insulin resistance and beta-cell dysfunction to the pathophysiology of Type 2 diabetes. Diabetologia. 2003;46(1):3-19.
    • (2003) Diabetologia , vol.46 , Issue.1 , pp. 3-19
    • Kahn, S.E.1
  • 11
    • 7844240131 scopus 로고    scopus 로고
    • Role of skeletal muscle in thiazolidin-edione insulin sensitizer (PPARγ agonist) action
    • Zierath JR, Ryder J W, Doebber T, et al. Role of skeletal muscle in thiazolidin-edione insulin sensitizer (PPARγ agonist) action. Endocrinology. 1998;139(12): 5034-5041.
    • (1998) Endocrinology , vol.139 , Issue.12 , pp. 5034-5041
    • Zierath, J.R.1    Ryder, J.W.2    Doebber, T.3
  • 12
    • 77649176059 scopus 로고    scopus 로고
    • Efects of colesevelam, rosiglitazone, or sitagliptin on glycemic control and lipid profle in patients with type 2 diabetes mellitus inadequately controlled by metformin monotherapy
    • Rigby SP, Handelsman Y, Lai Y-L, Abby SL, Tao B, Jones MR. Efects of colesevelam, rosiglitazone, or sitagliptin on glycemic control and lipid profle in patients with type 2 diabetes mellitus inadequately controlled by metformin monotherapy. Endocr Pract. 2010;16(1):53-63.
    • (2010) Endocr Pract , vol.16 , Issue.1 , pp. 53-63
    • Rigby, S.P.1    Handelsman, Y.2    Lai, Y.-L.3    Abby, S.L.4    Tao, B.5    Jones, M.R.6
  • 13
    • 54049103635 scopus 로고    scopus 로고
    • Colesevelam hydrochloride therapy in patients with type 2 diabetes mellitus treated with metformin: Glucose and lipid efects
    • Bays HE, Goldberg RB, Truitt KE, Jones MR. Colesevelam hydrochloride therapy in patients with type 2 diabetes mellitus treated with metformin: glucose and lipid efects. Arch Intern Med. 2008;168(18):1975-1983.
    • (2008) Arch Intern Med , vol.168 , Issue.18 , pp. 1975-1983
    • Bays, H.E.1    Goldberg, R.B.2    Truitt, K.E.3    Jones, M.R.4
  • 14
    • 84856701167 scopus 로고    scopus 로고
    • Effect of bile acid sequestrants on glucose metabolism, hepatic de novo lipogenesis, and cholesterol and bile acid kinetics in type 2 diabetes: A randomised controlled study
    • Beysen C, Murphy EJ, Deines K, et al. Effect of bile acid sequestrants on glucose metabolism, hepatic de novo lipogenesis, and cholesterol and bile acid kinetics in type 2 diabetes: a randomised controlled study. Diabetologia. 2012;55(2):432-442.
    • (2012) Diabetologia , vol.55 , Issue.2 , pp. 432-442
    • Beysen, C.1    Murphy, E.J.2    Deines, K.3
  • 15
    • 83655161342 scopus 로고    scopus 로고
    • Effects of colesevelam on glucose absorption and hepatic/peripheral insulin sensitivity in patients with type 2 diabetes mellitus
    • Henry RR, Aroda VR, Mudaliar S, Garvey WT, Chou HS, Jones MR. Effects of colesevelam on glucose absorption and hepatic/peripheral insulin sensitivity in patients with type 2 diabetes mellitus. Diabetes Obes Metab. 2012;14(1): 40-46.
    • (2012) Diabetes Obes Metab , vol.14 , Issue.1 , pp. 40-46
    • Henry, R.R.1    Aroda, V.R.2    Mudaliar, S.3    Garvey, W.T.4    Chou, H.S.5    Jones, M.R.6
  • 16
    • 77950620903 scopus 로고    scopus 로고
    • Te efect of colesevelam hydrochloride on insulin sensitivity and secretion in patients with type 2 diabetes: A pilot study
    • Schwartz SL, Lai Y-L, Xu J, et al. Te efect of colesevelam hydrochloride on insulin sensitivity and secretion in patients with type 2 diabetes: a pilot study. Metab Syndr Relat Disord. 2010;8(2):179-188.
    • (2010) Metab Syndr Relat Disord , vol.8 , Issue.2 , pp. 179-188
    • Schwartz, S.L.1    Lai, Y.-L.2    Xu, J.3
  • 17
    • 80053954040 scopus 로고    scopus 로고
    • Efect of colesevelam hydrochloride on gly-cemia and insulin sensitivity in men with the metabolic syndrome
    • Vega GL, Dunn FL, Grundy SM. Efect of colesevelam hydrochloride on gly-cemia and insulin sensitivity in men with the metabolic syndrome. Am J Cardiol. 2011;108(8):1129-1135.
    • (2011) Am J Cardiol , vol.108 , Issue.8 , pp. 1129-1135
    • Vega, G.L.1    Dunn, F.L.2    Grundy, S.M.3
  • 18
    • 78650205817 scopus 로고    scopus 로고
    • Initial combination therapy with metformin and colesevelam for achievement of glycemic and lipid goals in early type 2 diabetes
    • Rosenstock J, Fonseca VA, Garvey W T, et al. Initial combination therapy with metformin and colesevelam for achievement of glycemic and lipid goals in early type 2 diabetes. Endocr Pract. 2010;16(4):629-640.
    • (2010) Endocr Pract , vol.16 , Issue.4 , pp. 629-640
    • Rosenstock, J.1    Fonseca, V.A.2    Garvey, W.T.3
  • 19
    • 0027180608 scopus 로고
    • How good a marker is insulin level for insulin resistance?
    • Laakso M. How good a marker is insulin level for insulin resistance? Am J Epidemiol. 1993;137(9):959-965.
    • (1993) Am J Epidemiol , vol.137 , Issue.9 , pp. 959-965
    • Laakso, M.1
  • 20
    • 17944365228 scopus 로고    scopus 로고
    • Te fat-derived hormone adiponectin reverses insulin resistance associated with both lipoatrophy and obesity
    • Yamauchi T, Kamon J, Waki H, et al. Te fat-derived hormone adiponectin reverses insulin resistance associated with both lipoatrophy and obesity. Nat Med. 2001;7(8):941-946.
    • (2001) Nat Med , vol.7 , Issue.8 , pp. 941-946
    • Yamauchi, T.1    Kamon, J.2    Waki, H.3
  • 21
    • 0037303077 scopus 로고    scopus 로고
    • Free fatty acids increase basal hepatic glucose production and induce hepatic insulin resistance at different sites
    • Lam TKT, van de Werve G, Giacca A. Free fatty acids increase basal hepatic glucose production and induce hepatic insulin resistance at different sites. Am J Physiol Endocrinol Metab. 2003;284(2):E281-E290.
    • (2003) Am J Physiol Endocrinol Metab , vol.284 , Issue.2
    • Lam, T.K.T.1    van de Werve, G.2    Giacca, A.3
  • 22
    • 33947134267 scopus 로고    scopus 로고
    • Tiazolidinediones and the risk of edema: A meta-analysis
    • Berlie HD, Kalus JS, Jaber LA. Tiazolidinediones and the risk of edema: a meta-analysis. Diabetes Res Clin Pract. 2007;76(2):279-289.
    • (2007) Diabetes Res Clin Pract , vol.76 , Issue.2 , pp. 279-289
    • Berlie, H.D.1    Kalus, J.S.2    Jaber, L.A.3
  • 23
    • 7044253431 scopus 로고    scopus 로고
    • A meta-analysis comparing the efect of thiazolidinediones on cardiovascular risk factors
    • Chiquette E, Ramirez G, DeFronzo R. A meta-analysis comparing the efect of thiazolidinediones on cardiovascular risk factors. Arch Intern Med. 2004; 164(19):2097-2104.
    • (2004) Arch Intern Med , vol.164 , Issue.19 , pp. 2097-2104
    • Chiquette, E.1    Ramirez, G.2    Defronzo, R.3
  • 24
    • 84875463321 scopus 로고    scopus 로고
    • Te effect of a bile acid sequestrant on glucose metabolism in subjects with type 2 diabetes
    • Smushkin G, Sathananthan M, Piccinini F, et al. Te effect of a bile acid sequestrant on glucose metabolism in subjects with type 2 diabetes. Diabetes. 2013;62(4):1094-1101.
    • (2013) Diabetes , vol.62 , Issue.4 , pp. 1094-1101
    • Smushkin, G.1    Sathananthan, M.2    Piccinini, F.3
  • 25
    • 84862172072 scopus 로고    scopus 로고
    • Oral diabetes medications for adults with type 2 diabetes: An update
    • Accessed March 18, 2013
    • Bennett WL, Wilson LM, Bolen S, et al. Oral diabetes medications for adults with type 2 diabetes: an update. Rockville, MD: Agency for Healthcare Policy and Research; 2011. http://efectivehealthcare.ahrq.gov/ehc/products/155/644/CER27_OralDiabetesMeds_20110623.pdf. Accessed March 18, 2013.
    • (2011) Rockville, MD: Agency For Healthcare Policy and Research
    • Bennett, W.L.1    Wilson, L.M.2    Bolen, S.3
  • 26
    • 36749059401 scopus 로고    scopus 로고
    • Who should benefit from the use of alpha-glucosidase inhibitors?
    • Godbout A, Chiasson JL. Who should benefit from the use of alpha-glucosidase inhibitors? Curr Diab Rep. 2007;7(5):333-339.
    • (2007) Curr Diab Rep , vol.7 , Issue.5 , pp. 333-339
    • Godbout, A.1    Chiasson, J.L.2
  • 27
    • 84862087518 scopus 로고    scopus 로고
    • Colesevelam improves oral but not intravenous glucose tolerance by a mechanism independent of insulin sensitivity and β-cell function
    • Marina AL, Utzschneider KM, Wright LA, et al. Colesevelam improves oral but not intravenous glucose tolerance by a mechanism independent of insulin sensitivity and β-cell function. Diabetes Care. 2012;35(5):1119-1125.
    • (2012) Diabetes Care , vol.35 , Issue.5 , pp. 1119-1125
    • Marina, A.L.1    Utzschneider, K.M.2    Wright, L.A.3
  • 28
    • 75349109261 scopus 로고    scopus 로고
    • Efects of chenodeoxy-cholate and a bile acid sequestrant, colesevelam, on intestinal transit and bowel function
    • Odunsi-Shiyanbade ST, Camilleri M, McKinzie S, et al. Efects of chenodeoxy-cholate and a bile acid sequestrant, colesevelam, on intestinal transit and bowel function. Clin Gastroenterol Hepatol. 2010;8(2):159-165.
    • (2010) Clin Gastroenterol Hepatol , vol.8 , Issue.2 , pp. 159-165
    • Odunsi-Shiyanbade, S.T.1    Camilleri, M.2    McKinzie, S.3
  • 30
    • 0028240330 scopus 로고
    • Loss of the first phase insulin response to intravenous glucose in subjects with persistent impaired glucose tolerance
    • Davies MJ, Rayman G, Grenfell A, et al. Loss of the first phase insulin response to intravenous glucose in subjects with persistent impaired glucose tolerance. Diabet Med. 1994;11(5):432-436.
    • (1994) Diabet Med , vol.11 , Issue.5 , pp. 432-436
    • Davies, M.J.1    Rayman, G.2    Grenfell, A.3
  • 31
    • 33749347851 scopus 로고    scopus 로고
    • Paradoxical stimulation of glucagon secretion by high glucose concentrations
    • Salehi A, Vieira E, Gylfe E. Paradoxical stimulation of glucagon secretion by high glucose concentrations. Diabetes. 2006;55(8):2318-2323.
    • (2006) Diabetes , vol.55 , Issue.8 , pp. 2318-2323
    • Salehi, A.1    Vieira, E.2    Gylfe, E.3
  • 32
    • 0024507794 scopus 로고
    • Fasting hyperglycemia in non-insulin-dependent diabetes mellitus: Contributions of excessive hepatic glucose production and impaired tissue glucose uptake
    • DeFronzo RA, Ferrannini E, Simonson DC. Fasting hyperglycemia in non-insulin-dependent diabetes mellitus: contributions of excessive hepatic glucose production and impaired tissue glucose uptake. Metabolism. 1989;38(4):387-395.
    • (1989) Metabolism , vol.38 , Issue.4 , pp. 387-395
    • Defronzo, R.A.1    Ferrannini, E.2    Simonson, D.C.3
  • 33
    • 2342599057 scopus 로고    scopus 로고
    • One week's treatment with the long-acting glucagon-like peptide 1 derivative liraglutide (NN2211) markedly improves 24-h glycemia and α- and β-cell function and reduces endogenous glucose release in patients with type 2 diabetes
    • Degn KB, Juhl CB, Sturis J, et al. One week's treatment with the long-acting glucagon-like peptide 1 derivative liraglutide (NN2211) markedly improves 24-h glycemia and α- and β-cell function and reduces endogenous glucose release in patients with type 2 diabetes. Diabetes. 2004;53(5):1187-1194.
    • (2004) Diabetes , vol.53 , Issue.5 , pp. 1187-1194
    • Degn, K.B.1    Juhl, C.B.2    Sturis, J.3
  • 34
    • 63249101127 scopus 로고    scopus 로고
    • Inhibition of dipeptidyl peptidase-4 by vildagliptin during glucagon-like peptide 1 infusion increases liver glucose uptake in the conscious dog
    • Edgerton DS, Johnson KMS, Neal DW, et al. Inhibition of dipeptidyl peptidase-4 by vildagliptin during glucagon-like peptide 1 infusion increases liver glucose uptake in the conscious dog. Diabetes. 2009;58(1):243-249.
    • (2009) Diabetes , vol.58 , Issue.1 , pp. 243-249
    • Edgerton, D.S.1    Johnson, K.M.S.2    Neal, D.W.3
  • 35
    • 0141615898 scopus 로고    scopus 로고
    • Suppression of glucose production by GLP-1 independent of islet hormones: A novel extrapancreatic efect
    • Prigeon RL, Quddusi S, Paty B, D'Alessio DA. Suppression of glucose production by GLP-1 independent of islet hormones: a novel extrapancreatic efect. Am J Physiol Endocrinol Metab. 2003;285(4):E701-E707.
    • (2003) Am J Physiol Endocrinol Metab , vol.285 , Issue.4
    • Prigeon, R.L.1    Quddusi, S.2    Paty, B.3    D'Alessio, D.A.4
  • 36
    • 31044456099 scopus 로고    scopus 로고
    • Brain glucagon-like peptide-1 increases insulin secretion and muscle insulin resistance to favor hepatic glycogen storage
    • Knauf C, Cani PD, Perrin C, et al. Brain glucagon-like peptide-1 increases insulin secretion and muscle insulin resistance to favor hepatic glycogen storage. J Clin Invest. 2005;115(12):3554-3563.
    • (2005) J Clin Invest , vol.115 , Issue.12 , pp. 3554-3563
    • Knauf, C.1    Cani, P.D.2    Perrin, C.3
  • 37
    • 34948828109 scopus 로고    scopus 로고
    • Colestimide lowers plasma glucose levels and increases plasma glucagon-like peptide-1 (7-36) levels in patients with type 2 diabetes mellitus complicated by hypercholesterolemia
    • Suzuki T, Oba K, Igari Y, et al. Colestimide lowers plasma glucose levels and increases plasma glucagon-like peptide-1 (7-36) levels in patients with type 2 diabetes mellitus complicated by hypercholesterolemia. J Nippon Med Sch. 2007;74(5):338-343.
    • (2007) J Nippon Med Sch , vol.74 , Issue.5 , pp. 338-343
    • Suzuki, T.1    Oba, K.2    Igari, Y.3
  • 38
    • 13844299425 scopus 로고    scopus 로고
    • Bile acids promote glucagon-like peptide-1 secretion through TGR5 in a murine enteroendocrine cell line STC-1
    • Katsuma S, Hirasawa A, Tsujimoto G. Bile acids promote glucagon-like peptide-1 secretion through TGR5 in a murine enteroendocrine cell line STC-1. Biochem Biophys Res Commun. 2005;329(1):386-390.
    • (2005) Biochem Biophys Res Commun , vol.329 , Issue.1 , pp. 386-390
    • Katsuma, S.1    Hirasawa, A.2    Tsujimoto, G.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.