Inclusion of fenofibrate in a series of mesoporous silicas using microwave irradiation

European Journal of Pharmaceutics and Biopharmaceutics

Volumn 85, Issue 3 PART B, 2013, Pages 936-941

  Waters, Laura J ^a   Hussain, Talib ^a   Parkes, Gareth ^a   Hanrahan, John P ^b   Tobin, Joseph M ^b  

^a UNIVERSITY OF HUDDERSFIELD   (United Kingdom)

^b Glantreo Ltd   (Ireland)

Author keywords

Core shell silica; Drug release; Enhanced release; Fenofibrate; Microwave irradiation; Porous silica

Indexed keywords

EXCIPIENT; FENOFIBRATE; SILICA GEL; SILICON DIOXIDE; WATER;

ARTICLE; CONTROLLED STUDY; DIFFERENTIAL SCANNING CALORIMETRY; DRUG ADSORPTION; DRUG FORMULATION; DRUG RELEASE; DRUG SOLUBILITY; FLUIDIZATION; HEATING; IN VITRO STUDY; INFRARED SPECTROSCOPY; INTERMETHOD COMPARISON; MICROWAVE COOKING; MICROWAVE IRRADIATION; PARTICLE SIZE; PHYSICAL CHEMISTRY; POROSITY; SCANNING ELECTRON MICROSCOPY; SURFACE PROPERTY; X RAY DIFFRACTION;

CORE SHELL SILICA; DRUG RELEASE; ENHANCED RELEASE; FENOFIBRATE; MICROWAVE IRRADIATION; POROUS SILICA;

ADSORPTION; BIOLOGICAL AVAILABILITY; CALORIMETRY, DIFFERENTIAL SCANNING; DRUG CARRIERS; EXCIPIENTS; FENOFIBRATE; MICROSCOPY, ELECTRON, SCANNING; MICROWAVES; POWDERS; SILICON DIOXIDE; SOLUBILITY; SPECTROSCOPY, FOURIER TRANSFORM INFRARED; TECHNOLOGY, PHARMACEUTICAL; TEMPERATURE; X-RAY DIFFRACTION;

EID: 84889084784     PISSN: 09396411     EISSN: 18733441     Source Type: Journal    
DOI: 10.1016/j.ejpb.2013.08.002     Document Type: Article

References (31)

1. S. Torrado, J.J. Torrado, and R. Cadórniga Preparation, dissolution and characterization of albendazole solid dispersions International Journal of Pharmaceutics 140 1996 247 250
2. M. Vallet-Regí, F. Balas, and D. Arcos Mesoporous materials for drug delivery Angewandte Chemie - International Edition 46 2007 7548 7558
3. C. Barbé, J. Bartlett, L. Kong, K. Finnie, H.Q. Lin, M. Larkin, S. Calleja, A. Bush, and G. Calleja Silica particles: a novel drug-delivery system Advanced Materials 16 2004 1959 1966
4. H.J. Kim, K.J. Shin, M.K. Han, K. An, J.K. Lee, I. Honma, and H. Kim One-pot synthesis of multifunctional mesoporous silica nanoparticle incorporated with zinc(II) phthalocyanine and iron oxide Scripta Materialia 61 2009 1137 1140
5. P. Kinnari, E. Mäkilä, T. Heikkilä, J. Salonen, J. Hirvonen, and H.A. Santos Comparison of mesoporous silicon and non-ordered mesoporous silica materials as drug carriers for itraconazole International Journal of Pharmaceutics 414 2011 148 156
6. R. Mellaerts, J.A.G. Jammaer, M. Van Speybroeck, C. Hong, J. Van Humbeeck, P. Augustijns, G. Van Den Mooter, and J.A. Martens Physical state of poorly water soluble therapeutic molecules loaded into SBA-15 ordered mesoporous silica carriers: a case study with itraconazole and ibuprofen Langmuir 24 2008 8651 8659
7. J. Andersson, J. Rosenholm, S. Areva, and M. Lindén Influences of material characteristics on ibuprofen drug loading and release profiles from ordered micro- and mesoporous silica matrices Chemistry of Materials 16 2004 4160 4167
8. Y.F. Zhu, J.L. Shi, Y.S. Li, H.R. Chen, W.H. Shen, and X.P. Dong Storage and release of ibuprofen drug molecules in hollow mesoporous silica spheres with modified pore surface Microporous and Mesoporous Materials 85 2005 75 81
9. C. Charnay, S. Bégu, C. Tourné-Péteilh, L. Nicole, D.A. Lerner, and J.M. Devoisselle Inclusion of ibuprofen in mesoporous templated silica: drug loading and release property European Journal of Pharmaceutics and Biopharmaceutics 57 2004 533 540
10. M. Van Speybroeck, V. Barillaro, T.D. Thi, R. Mellaerts, J. Martens, J. Van Humbeeck, J. Vermant, P. Annaert, G. Van Den Mooter, and P. Augustijns Ordered mesoporous silica material SBA-15: a broad-spectrum formulation platform for poorly soluble drugs Journal of Pharmaceutical Sciences 98 2009 2648 2658
11. Y. Zhang, Z. Zhi, T. Jiang, J. Zhang, Z. Wang, and S. Wang Spherical mesoporous silica nanoparticles for loading and release of the poorly water-soluble drug telmisartan Journal of Controlled Release 145 2010 257 263
12. Q. Tang, Y. Xu, D. Wu, and Y. Sun A study of carboxylic-modified mesoporous silica in controlled delivery for drug famotidine Journal of Solid State Chemistry 179 2006 1513 1520
13. M.J.K. Thomas, I. Slipper, A. Walunj, A. Jain, M.E. Favretto, P. Kallinteri, and D. Douroumis Inclusion of poorly soluble drugs in highly ordered mesoporous silica nanoparticles International Journal of Pharmaceutics 387 2010 272 277
14. T. Lebold, C. Jung, J. Michaelis, and C. Bräuchle Nanostructured silica materials as drug-delivery systems for doxorubicin: single molecule and cellular studies Nano Letters 9 2009 2877 2883
15. S.W. Song, K. Hidajat, and S. Kawi Functionalized SBA-15 materials as carriers for controlled drug delivery: influence of surface properties on matrix-drug interactions Langmuir 21 2005 9568 9575
16. Q. Yang, S. Wang, P. Fan, L. Wang, Y. Di, K. Lin, and F.S. Xiao PH-responsive carrier system based on carboxylic acid modified mesoporous silica and polyelectrolyte for drug delivery Chemistry of Materials 17 2005 5999 6003
17. M. van Speybroeck, R. Mellaerts, T.D. Thi, J.A. Martens, J. Van Humbeeck, P. Annaert, G. Van den Mooter, and P. Augustijns Preventing release in the acidic environment of the stomach via occlusion in ordered mesoporous silica enhances the absorption of poorly soluble weakly acidic drugs Journal of Pharmaceutical Sciences 100 2011 4864 4876
18. H. Takeuchi, S. Nagira, H. Yamamoto, and Y. Kawashima Solid dispersion particles of tolbutamide prepared with fine silica particles by the spray-drying method Powder Technology 141 2004 187 195
19. H. Takeuchi, S. Nagira, H. Yamamoto, and Y. Kawashima Solid dispersion particles of amorphous indomethacin with fine porous silica particles by using spray-drying method International Journal of Pharmaceutics 293 2005 155 164
20. M. Vialpando, F. Backhuijs, J.A. Martens, and G. Van Den Mooter Risk assessment of premature drug release during wet granulation of ordered mesoporous silica loaded with poorly soluble compounds itraconazole, fenofibrate, naproxen, and ibuprofen European Journal of Pharmaceutics and Biopharmaceutics 81 2012 190 198
21. Y. Tozuka, E. Sugiyama, and H. Takeuchi Release profile of insulin entrapped on mesoporous materials by freeze-thaw method International Journal of Pharmaceutics 386 2010 172 177
22. 2) processing conditions on drug loading and physicochemical properties International Journal of Pharmaceutics 439 2012 92 99
23. T. Limnell, H.A. Santos, E. Mäkilä, T. Heikkilä, J. Salonen, D.Y. Murzin, N. Kumar, T. Laaksonen, L. Peltonen, and J. Hirvonen Drug delivery formulations of ordered and nonordered mesoporous silica: comparison of three drug loading methods Journal of Pharmaceutical Sciences 100 2011 3294 3306
24. Y. Lang, D.P. Finn, A. Pandit, and P.J. Walsh Pharmacological activity of ibuprofen released from mesoporous silica Journal of Materials Science. Materials in Medicine 23 2012 73 80
25. W. Xu, J. Riikonen, and V.P. Lehto Mesoporous systems for poorly soluble drugs International Journal of Pharmaceutics 2012
26. R. Mellaerts, R. Mols, J.A.G. Jammaer, C.A. Aerts, P. Annaert, J. Van Humbeeck, G. Van den Mooter, P. Augustijns, and J.A. Martens Increasing the oral bioavailability of the poorly water soluble drug itraconazole with ordered mesoporous silica European Journal of Pharmaceutics and Biopharmaceutics 69 2008 223 230
27. J.M. Rosenholm, and M. Lindén Towards establishing structure-activity relationships for mesoporous silica in drug delivery applications Journal of Controlled Release 128 2008 157 164
28. Z. Jia, P. Lin, Y. Xiang, X. Wang, J. Wang, X. Zhang, and Q. Zhang A novel nanomatrix system consisted of colloidal silica and pH-sensitive polymethylacrylate improves the oral bioavailability of fenofibrate European Journal of Pharmaceutics and Biopharmaceutics 79 2011 126 134
29. M. Van Speybroeck, R. Mellaerts, R. Mols, T.D. Thi, J.A. Martens, J. Van Humbeeck, P. Annaert, G. Van den Mooter, and P. Augustijns Enhanced absorption of the poorly soluble drug fenofibrate by tuning its release rate from ordered mesoporous silica European Journal of Pharmaceutical Sciences 41 2010 623 630
30. A. Nacsa, R. Ambrus, O. Berkesi, P. Szabó-Révész, and Z. Aigner Water-soluble loratadine inclusion complex: analytical control of the preparation by microwave irradiation Journal of Pharmaceutical and Biomedical Analysis 48 2008 1020 1023
31. L.J. Waters, S. Bedford, and G.M.B. Parkes Controlled microwave processing applied to the pharmaceutical formulation of ibuprofen AAPS PharmSciTech 12 2011 1038 1043