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Volumn 718, Issue 1-3, 2013, Pages 167-172

Effects of the sazetidine-a family of compounds on the body temperature in wildtype, nicotinic receptor β2-/- and α7-/- mice

Author keywords

Desensitization; Knockout; Nicotinic; Sazetidine A; Temperature regulation

Indexed keywords

BUNGAROTOXIN RECEPTOR; DESENSITIZING AGENT; NICOTINE; NICOTINIC RECEPTOR BETA2; RECEPTOR SUBTYPE; SAZETIDINE A; TRIAZETIDINE O; UNCLASSIFIED DRUG; VMY 2 95; YL 1 127;

EID: 84887069104     PISSN: 00142999     EISSN: 18790712     Source Type: Journal    
DOI: 10.1016/j.ejphar.2013.08.037     Document Type: Article
Times cited : (2)

References (30)
  • 3
    • 0036889388 scopus 로고    scopus 로고
    • Effects of repeated nicotine exposure on core temperature and motor activity in male and female rats
    • C.J. Gordon, P.J. Rowse, and Y.L. Yang Effects of repeated nicotine exposure on core temperature and motor activity in male and female rats Journal of Thermal Biology 27 2002 485 492
    • (2002) Journal of Thermal Biology , vol.27 , pp. 485-492
    • Gordon, C.J.1    Rowse, P.J.2    Yang, Y.L.3
  • 4
    • 0015522557 scopus 로고
    • Temperature changes produced by nicotine injected into the hypothalamus of the conscious monkey
    • G.H. Hall, and R.D. Myers Temperature changes produced by nicotine injected into the hypothalamus of the conscious monkey Brain Res 37 1972 241 251
    • (1972) Brain Res , vol.37 , pp. 241-251
    • Hall, G.H.1    Myers, R.D.2
  • 5
    • 0025138223 scopus 로고
    • Acute effects of nicotine on prolactin release in the rat: Agonist and antagonist effects of a single injection of nicotine
    • B.A. Hulihan-Giblin, M.L. Lumpkin, and K.J. Kellar Acute effects of nicotine on prolactin release in the rat: Agonist and antagonist effects of a single injection of nicotine The Journal of Pharmacology and Experimental Therapeutics 252 1990 15 20
    • (1990) The Journal of Pharmacology and Experimental Therapeutics , vol.252 , pp. 15-20
    • Hulihan-Giblin, B.A.1    Lumpkin, M.L.2    Kellar, K.J.3
  • 6
    • 84965075853 scopus 로고
    • A study of the desensitization produced by acetylcholine at the motor end-plate
    • B. Katz, and S. Thesleff A study of the desensitization produced by acetylcholine at the motor end-plate Journal of Physiology 138 1957 63 80
    • (1957) Journal of Physiology , vol.138 , pp. 63-80
    • Katz, B.1    Thesleff, S.2
  • 7
    • 67649380330 scopus 로고    scopus 로고
    • Cholinergic mechanisms of the medial preoptic areas of the hypothalamus in the control of thermoregulation and the states of sleep and waking in pigeons
    • T.G. Komarova Cholinergic mechanisms of the medial preoptic areas of the hypothalamus in the control of thermoregulation and the states of sleep and waking in pigeons Neuroscience and Behavioral Physiology 39 2009 553 558
    • (2009) Neuroscience and Behavioral Physiology , vol.39 , pp. 553-558
    • Komarova, T.G.1
  • 9
    • 77957898423 scopus 로고    scopus 로고
    • Chemistry and pharmacological characterization of novel nitrogen analogues of AMOP-H-OH (Sazetidine-A, 6-[5-(azetidin-2-ylmethoxy)pyridin-3-yl] hex-5-yn-1-ol) as alpha4beta2-nicotinic acetylcholine receptor-selective partial agonists
    • J. Liu, J.B. Eaton, B. Caldarone, R.J. Lukas, and A.P. Kozikowski Chemistry and pharmacological characterization of novel nitrogen analogues of AMOP-H-OH (Sazetidine-A, 6-[5-(azetidin-2-ylmethoxy)pyridin-3-yl]hex-5-yn-1-ol) as alpha4beta2-nicotinic acetylcholine receptor-selective partial agonists Journal of Medicinal Chemistry 53 2010 6973 6985
    • (2010) Journal of Medicinal Chemistry , vol.53 , pp. 6973-6985
    • Liu, J.1    Eaton, J.B.2    Caldarone, B.3    Lukas, R.J.4    Kozikowski, A.P.5
  • 13
    • 0020539924 scopus 로고
    • Pharmacodynamic effects of nicotine and acetylcholine biosynthesis in mouse brain
    • A. Nordberg, and A. Sundwall Pharmacodynamic effects of nicotine and acetylcholine biosynthesis in mouse brain Acta Pharmacologica et Toxicologica 52 1983 341 347
    • (1983) Acta Pharmacologica et Toxicologica , vol.52 , pp. 341-347
    • Nordberg, A.1    Sundwall, A.2
  • 15
    • 41149145063 scopus 로고    scopus 로고
    • It is not "either/or": Activation and desensitization of nicotinic acetylcholine receptors both contribute to behaviors related to nicotine addiction and mood
    • M.R. Picciotto, N.A. Addy, Y.S. Mineur, and D.H. Brunzell It is not "either/or": activation and desensitization of nicotinic acetylcholine receptors both contribute to behaviors related to nicotine addiction and mood Progress in Neurobiology 84 2008 329 342
    • (2008) Progress in Neurobiology , vol.84 , pp. 329-342
    • Picciotto, M.R.1    Addy, N.A.2    Mineur, Y.S.3    Brunzell, D.H.4
  • 16
    • 0036891571 scopus 로고    scopus 로고
    • Desensitization of neuronal nicotinic receptors
    • M. Quick, and R. Lester Desensitization of neuronal nicotinic receptors Journal of Neurobiology 53 2002 457 478
    • (2002) Journal of Neurobiology , vol.53 , pp. 457-478
    • Quick, M.1    Lester, R.2
  • 17
    • 84859108539 scopus 로고    scopus 로고
    • Effects of sazetidine-A, a selective α4β2 nicotinic receptor desensitizing agent and partial agonist, on core body temperature in mice and rats
    • A.H. Rezvani, O. Timofeeva, D. DeCuir, H.G. Sexton, X. Xiao, C.J. Gordon, K.J. Kellar, and E.D. Levin Effects of sazetidine-A, a selective α4β2 nicotinic receptor desensitizing agent and partial agonist, on core body temperature in mice and rats European Journal of Pharmacology 682 2012 110 117
    • (2012) European Journal of Pharmacology , vol.682 , pp. 110-117
    • Rezvani, A.H.1    Timofeeva, O.2    Decuir, D.3    Sexton, H.G.4    Xiao, X.5    Gordon, C.J.6    Kellar, K.J.7    Levin, E.D.8
  • 18
    • 57049163448 scopus 로고    scopus 로고
    • Chronic menthol attenuates the effect of nicotine on body temperature in adolescent rats
    • D.N. Ruskin, R. Anand, and G.J. LaHoste Chronic menthol attenuates the effect of nicotine on body temperature in adolescent rats Nicotine and Tobacco Research 10 2008 1753 1759
    • (2008) Nicotine and Tobacco Research , vol.10 , pp. 1753-1759
    • Ruskin, D.N.1    Anand, R.2    Lahoste, G.J.3
  • 19
    • 19544383094 scopus 로고    scopus 로고
    • Lower core body temperature and attenuated nicotine-induced hypothermic response in mice lacking the beta4 neuronal nicotinic acetylcholine receptor subunit
    • R. Sack, A. Gochberg-Sarver, U. Rozovsky, M. Kedmi, S. Rosner, and A. Orr-Urtreger Lower core body temperature and attenuated nicotine-induced hypothermic response in mice lacking the beta4 neuronal nicotinic acetylcholine receptor subunit Brain Research Bulletin 66 2005 30 36
    • (2005) Brain Research Bulletin , vol.66 , pp. 30-36
    • Sack, R.1    Gochberg-Sarver, A.2    Rozovsky, U.3    Kedmi, M.4    Rosner, S.5    Orr-Urtreger, A.6
  • 20
    • 0034697353 scopus 로고    scopus 로고
    • The effects of acute nicotine on the body temperature and striatal dopamine metabolism of mice during chronic nicotine infusion
    • O. Salminen, and L. Ahtee The effects of acute nicotine on the body temperature and striatal dopamine metabolism of mice during chronic nicotine infusion Neuroscience Letters 284 2000 37 40
    • (2000) Neuroscience Letters , vol.284 , pp. 37-40
    • Salminen, O.1    Ahtee, L.2
  • 21
    • 0022521721 scopus 로고
    • Rapid desensitization of the acute stimulatory effects of nicotine on rat plasma adrenocorticotropin and prolactin
    • B.M. Sharp, and H.S. Beyer Rapid desensitization of the acute stimulatory effects of nicotine on rat plasma adrenocorticotropin and prolactin The Journal of Pharmacology and Experimental Therapeutics 238 1986 486 491
    • (1986) The Journal of Pharmacology and Experimental Therapeutics , vol.238 , pp. 486-491
    • Sharp, B.M.1    Beyer, H.S.2
  • 23
    • 36248947308 scopus 로고    scopus 로고
    • Nicotine responses in hypersensitive and knockout alpha 4 mice account for tolerance to both hypothermia and locomotor suppression in wild-type mice
    • A.R. Tapper, S.L. McKinney, M.J. Marks, and H.A. Lester Nicotine responses in hypersensitive and knockout alpha 4 mice account for tolerance to both hypothermia and locomotor suppression in wild-type mice Physiological Genomics 31 2007 422 428
    • (2007) Physiological Genomics , vol.31 , pp. 422-428
    • Tapper, A.R.1    McKinney, S.L.2    Marks, M.J.3    Lester, H.A.4
  • 24
    • 33748927988 scopus 로고    scopus 로고
    • Sazetidine-A, a novel ligand that desensitizes alpha4beta2 nicotinic acetylcholine receptors without activating them
    • Y. Xiao, H. Fan, J.L. Musachio, Z.L. Wei, S.K. Chellappan, A.P. Kozikowski, and K.J. Kellar Sazetidine-A, a novel ligand that desensitizes alpha4beta2 nicotinic acetylcholine receptors without activating them Molecular Pharmacology 70 2006 1454 1460
    • (2006) Molecular Pharmacology , vol.70 , pp. 1454-1460
    • Xiao, Y.1    Fan, H.2    Musachio, J.L.3    Wei, Z.L.4    Chellappan, S.K.5    Kozikowski, A.P.6    Kellar, K.J.7
  • 29
    • 0028901467 scopus 로고
    • Nicotine-induced hypothermia through an indirect dopaminergic mechanism
    • M.R. Zarrindast, A. Zarghi, and A. Amiri Nicotine-induced hypothermia through an indirect dopaminergic mechanism Journal of Psychopharmacology 9 1995 20 24
    • (1995) Journal of Psychopharmacology , vol.9 , pp. 20-24
    • Zarrindast, M.R.1    Zarghi, A.2    Amiri, A.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.