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Bioorganic and Medicinal Chemistry Letters

Volumn 23, Issue 23, 2013, Pages 6455-6458

Design, synthesis, and biological evaluation of bone-targeted proteasome inhibitors for multiple myeloma

(3) Agyin, Joseph K a Santhamma, Bindu b Roy, Sudipa S a

a UNIVERSITY OF TEXAS HEALTH SCIENCE CENTER AT SAN ANTONIO (United States)

b EVESTRA INC (United States)

Author keywords

Bisphosphonate conjugate; Bone targeted; Boronic acid; Multiple myeloma; Proteasome inhibitor

Indexed keywords

BISPHOSPHONIC ACID DERIVATIVE; BORTEZOMIB; MG 262BP; PROTEASOME INHIBITOR; PS 341BP 1; PS 341BP 2; UNCLASSIFIED DRUG;

ANIMAL CELL; ANTINEOPLASTIC ACTIVITY; ANTIPROLIFERATIVE ACTIVITY; ARTICLE; BONE DESTRUCTION; BONE TISSUE; CANCER CELL CULTURE; CANCER INHIBITION; CELL PROLIFERATION; CELL VIABILITY; CONTROLLED STUDY; DRUG CONJUGATION; DRUG DESIGN; DRUG SCREENING; DRUG STRUCTURE; DRUG SYNTHESIS; DRUG TARGETING; HUMAN; HUMAN CELL; IN VITRO STUDY; MOUSE; MULTIPLE MYELOMA; MYELOMA CELL; NONHUMAN; TUMOR MICROENVIRONMENT;

BISPHOSPHONATE CONJUGATE; BONE-TARGETED; BORONIC ACID; MULTIPLE MYELOMA; PROTEASOME INHIBITOR;

ANIMALS; ANTINEOPLASTIC AGENTS; BONE AND BONES; BONE DENSITY CONSERVATION AGENTS; BORONIC ACIDS; CELL LINE, TUMOR; CELL PROLIFERATION; DIPHOSPHONATES; HUMANS; MICE; MULTIPLE MYELOMA; PROTEASOME INHIBITORS;

EID: 84886951236 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2013.09.043 Document Type: Article

Times cited : (20)

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