Active site-directed inhibitors of Rhodococcus 20 S proteasome. Kinetics and mechanism

Journal of Biological Chemistry

Volumn 272, Issue 42, 1997, Pages 26103-26109

  Mc Cormack, Teresa ^a   Baumeister, Wolfgang ^c   Grenier, Louis ^a   Moomaw, Carolyn ^b   Plamondon, Louis ^a   Pramanik, Bikash ^b   Slaughter, Clive ^b   Soucy, François ^a   Stein, Ross ^a   Zühl, Frank ^c   Dick, Lawrence ^a  

^a ProScript Inc   (United States)

^b UNIVERSITY OF TEXAS SOUTHWESTERN MEDICAL CENTER   (United States)

^c MAX PLANCK INSTITUTE OF BIOCHEMISTRY   (Germany)

Author keywords

[No Author keywords available]

Indexed keywords

BORONIC ACID DERIVATIVE; ENZYME INHIBITOR; LACTACYSTIN BETA LACTONE; LACTONE DERIVATIVE; PEPTIDYL VINYL SULFONE; PROTEASOME; THREONINE; UNCLASSIFIED DRUG; VINYL DERIVATIVE;

ARTICLE; BETA CHAIN; CONTROLLED STUDY; ENZYME ACTIVE SITE; ENZYME INHIBITION; ENZYME KINETICS; ENZYME MECHANISM; NONHUMAN; PRIORITY JOURNAL; RHODOCOCCUS;

BINDING SITES; CYSTEINE ENDOPEPTIDASES; CYSTEINE PROTEINASE INHIBITORS; KINETICS; LACTONES; MULTIENZYME COMPLEXES; PROTEASOME ENDOPEPTIDASE COMPLEX; RECOMBINANT PROTEINS; RHODOCOCCUS;

RHODOCOCCUS;

EID: 0030671540     PISSN: 00219258     EISSN: None     Source Type: Journal    
DOI: 10.1074/jbc.272.42.26103     Document Type: Article

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