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Bioorganic and Medicinal Chemistry Letters

Volumn 23, Issue 23, 2013, Pages 6481-6485

Design, synthesis and binding affinity of acetylcholine carbamoyl analogues

(10) Bolchi, Cristiano a Valoti, Ermanno a Binda, Matteo a Fasoli, Francesca a Ferrara, Rossana a Fumagalli, Laura a Gotti, Cecilia a Matucci, Rosanna b Vistoli, Giulio a Pallavicini, Marco a

a UNIVERSITY OF MILAN (Italy)

b UNIVERSITY OF FLORENCE (Italy)

Author keywords

Affinity; Carbachol; Carbamoyl; Ligand; nAChR; Oxazolidinone

Indexed keywords

5 DIMETHYLAMINOMETHYL 2 OXAZOLIDINONE; 5 TRIMETHYLAMMONIOMETHYL 2 OXAZOLIDINONE; ACETYLCHOLINE CARBAMOYL ANALOGUE; ACETYLCHOLINE DERIVATIVE; CARBACHOL; CARBAMIC ACID DERIVATIVE; MUSCARINIC RECEPTOR; N METHYLPROLINOL CARBAMATE; NICOTINIC RECEPTOR ALPHA4BETA2; NITROGEN DERIVATIVE; OXAZOLIDINONE DERIVATIVE; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; BINDING AFFINITY; BRAIN CORTEX; CONTROLLED STUDY; CYCLIZATION; DIASTEREOISOMER; DRUG DESIGN; DRUG RECEPTOR BINDING; DRUG STRUCTURE; DRUG SYNTHESIS; ENANTIOMER; FEMALE; HIPPOCAMPUS; HYBRIDIZATION; METHYLATION; MOLECULAR DOCKING; NONHUMAN; RAT; STEREOISOMERISM; STRUCTURE ACTIVITY RELATION;

AFFINITY; CARBACHOL; CARBAMOYL; LIGAND; NACHR; OXAZOLIDINONE;

ACETYLCHOLINE; ANIMALS; BINDING SITES; CARBACHOL; CARBAMATES; CHO CELLS; CRICETULUS; DRUG DESIGN; HUMANS; LIGANDS; MODELS, MOLECULAR; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 84886947582 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2013.09.023 Document Type: Article

Times cited : (4)

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