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Bioorganic and Medicinal Chemistry Letters

Volumn 23, Issue 20, 2013, Pages 5614-5618

3-Ylidenephthalides as a new class of transient receptor potential channel TRPA1 and TRPM8 modulators

(6) Ortar, Giorgio a Schiano Moriello, Aniello b,c Morera, Enrico a Nalli, Marianna a Di Marzo, Vincenzo c De Petrocellis, Luciano b

a SAPIENZA UNIVERSITY OF ROME (Italy)

b CNR (Italy)

c CNR (Italy)

Author keywords

3 Ylidenephthalides; Transient receptor potential channels; TRPA1; TRPM8

Indexed keywords

3 YLIDENEPHTHALIDE DERIVATIVE; LIGUSTILIDE; PHTHALIDE DERIVATIVE; TRANSIENT RECEPTOR POTENTIAL CHANNEL A1; TRANSIENT RECEPTOR POTENTIAL CHANNEL M8; UNCLASSIFIED DRUG;

ARTICLE; CONTROLLED STUDY; DRUG STRUCTURE; HUMAN; HUMAN CELL; IC 50; MOUSE; NONHUMAN; RECEPTOR POTENTIAL; SYNTHESIS;

3-YLIDENEPHTHALIDES; TRANSIENT RECEPTOR POTENTIAL CHANNELS; TRPA1; TRPM8;

4-BUTYROLACTONE; ANIMALS; BENZOFURANS; HEK293 CELLS; HUMANS; OXIDATION-REDUCTION; PROTEIN BINDING; RATS; TRPC CATION CHANNELS; TRPM CATION CHANNELS;

EID: 84884285185 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2013.08.039 Document Type: Article

Times cited : (37)

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