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Volumn 49, Issue 74, 2013, Pages 8187-8189

Acid-cleavable thiomaleamic acid linker for homogeneous antibody–drug conjugation

(9) Castañeda, Lourdes a Maruani, Antoine a Schumacher, Felix F a Miranda, Enrique b Chudasama, Vijay a Chester, Kerry A b Baker, James R a Smith, Mark E B a Caddick, Stephen a

a UNIVERSITY COLLEGE LONDON (United Kingdom)

b UNIVERSITY COLLEGE LONDON (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

ANTIBODIES, MONOCLONAL, HUMANIZED; DISULFIDES; HYDROGEN-ION CONCENTRATION; MALEATES; MOLECULAR STRUCTURE; PHARMACEUTICAL PREPARATIONS; TEMPERATURE;

ACID; DISULFIDE; DOXORUBICIN; IMMUNOGLOBULIN F(AB) FRAGMENT; THIOMALEAMIC ACID; TRASTUZUMAB EMTANSINE; UNCLASSIFIED DRUG;

ACIDIFICATION; ANTIBODY DRUG CONJUGATION; ARTICLE; DISULFIDE BOND; DRUG CONJUGATION; HYDROLYSIS; LYSOSOME; PH; QUANTITATIVE ANALYSIS; SYNTHESIS; TEMPERATURE;

EID: 84882673481 PISSN: 13597345 EISSN: 1364548X Source Type: Journal
DOI: 10.1039/c3cc45220d Document Type: Article

Times cited : (68)

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