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ChemMedChem

Volumn 8, Issue 8, 2013, Pages 1283-1294

Design of a highly selective and potent class of non-planar estrogen receptorβ agonists

(6) Sundén, Henrik a Ma, Jian Nong b Hansen, Lars K c Gustavsson, Anna Lena d Burstein, Ethan S b Olsson, Roger a,b,e

a UNIVERSITY OF GOTHENBURG (Sweden)

b ACADIA PHARMACEUTICALS INC (United States)

c UNIVERSITY OF TROMSØ (Norway)

d KAROLINSKA INSTITUTE (Sweden)

e LUND UNIVERSITY (Sweden)

Author keywords

Asymmetric synthesis; Estrogen receptors; Modulators; Neurological agents; Parkinson's disease

Indexed keywords

CYCLOHEXANE; DIHYDROBENZOFURAN DERIVATIVE; ESTROGEN RECEPTOR BETA;

ARTICLE; CATALYSIS; CONCENTRATION RESPONSE; DIASTEREOISOMER; DRUG DESIGN; DRUG EFFICACY; DRUG POTENCY; DRUG SYNTHESIS; ENANTIOSELECTIVITY; ESTROGEN BINDING; HECK REACTION; IN VITRO STUDY; MOLECULAR MODEL; PRIORITY JOURNAL; STRUCTURE ACTIVITY RELATION;

EID: 84881026267 PISSN: 18607179 EISSN: 18607187 Source Type: Journal
DOI: 10.1002/cmdc.201300175 Document Type: Article

Times cited : (9)

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