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Volumn 49, Issue 4, 2013, Pages 782-789

Antimicrobial assay optimization and validation for HTS in 384-well format using a bioluminescent E. coli K-12 strain

Author keywords

Bioluminescence; Cell based assay; High throughput screening; Miniaturization; Transcription; Translation

Indexed keywords

ERYTHROMYCIN; RIFAMPICIN;

EID: 84880184614     PISSN: 09280987     EISSN: 18790720     Source Type: Journal    
DOI: 10.1016/j.ejps.2013.05.024     Document Type: Article
Times cited : (9)

References (31)
  • 1
    • 77954954109 scopus 로고    scopus 로고
    • Cell-based assays for high-throughput screening
    • An, W.F., Tolliday, N., 2010. Cell-based assays for high-throughput screening. Mol. Biotechnol. 45, 180-186.
    • (2010) Mol. Biotechnol. , vol.45 , pp. 180-186
    • An, W.F.1    Tolliday, N.2
  • 3
    • 79959740064 scopus 로고    scopus 로고
    • Antibiotics in the clinical pipeline in 2011
    • Butler, M.S., Cooper, M.A., 2011. Antibiotics in the clinical pipeline in 2011. J. Antibiot. (Tokyo) 64, 413-425.
    • (2011) J. Antibiot. (Tokyo) , vol.64 , pp. 413-425
    • Butler, M.S.1    Cooper, M.A.2
  • 4
    • 84869886623 scopus 로고    scopus 로고
    • Antibiotics in phase II and III clinical trials
    • Coates, A.R.M., Halls, G., 2012. Antibiotics in phase II and III clinical trials. Handb. Exp. Pharmacol. 211, 167-183.
    • (2012) Handb. Exp. Pharmacol. , vol.211 , pp. 167-183
    • Coates, A.R.M.1    Halls, G.2
  • 5
    • 84891402719 scopus 로고    scopus 로고
    • Pharmaceutical drug discovery: Designing the blockbuster drug
    • In: Dean, A.M., Lewis, S. (Eds.), Springer Science + Business Media Inc., New York, USA
    • Cummings, D.J., 2006. Pharmaceutical drug discovery: designing the blockbuster drug. In: Dean, A.M., Lewis, S. (Eds.), Screening: Methods for Experimentation in Industry, Drug Discovery, and Genetics. Springer Science + Business Media Inc., New York, USA, pp. 69-75.
    • (2006) Screening: Methods for Experimentation in Industry, Drug Discovery, and Genetics , pp. 69-75
    • Cummings, D.J.1
  • 6
    • 0030933177 scopus 로고    scopus 로고
    • Quinolones share a common interaction domain on topoisomerase II with other DNA cleavage-enhancing antineoplastic drugs
    • DOI 10.1021/bi962488f
    • Elsea, S.H., Westergaard, M., Burden, D.A., Lomenick, J.P., Osheroff, N., 1997. Quinolones share a common interaction domain on topoisomerase II with other DNA cleavage-enhancing antineoplastic drugs. Biochemistry 36, 2919-2924. (Pubitemid 27138575)
    • (1997) Biochemistry , vol.36 , Issue.10 , pp. 2919-2924
    • Elsea, S.H.1    Westergaard, M.2    Burden, D.A.3    Lomenick, J.P.4    Osheroff, N.5
  • 7
    • 78649712445 scopus 로고    scopus 로고
    • The continuing crisis in antibiotic resistance
    • French, G.L., 2010. The continuing crisis in antibiotic resistance. Int. J. Antimicrob. Agents 36 (Suppl. 3), S3-S7.
    • (2010) Int. J. Antimicrob. Agents , vol.36 , Issue.SUPPL. 3
    • French, G.L.1
  • 8
    • 1542648881 scopus 로고    scopus 로고
    • Amplified detection of transcriptional and translational inhibitors in bioluminescent Escherichia coli K-12
    • Galluzzi, L., Karp, M., 2003. Amplified detection of transcriptional and translational inhibitors in bioluminescent Escherichia coli K-12. J. Biomol. Screen. 8, 340-346.
    • (2003) J. Biomol. Screen. , vol.8 , pp. 340-346
    • Galluzzi, L.1    Karp, M.2
  • 9
    • 33746629426 scopus 로고    scopus 로고
    • Whole cell strategies based on lux genes for high throughput applications toward new antimicrobials
    • DOI 10.2174/138620706777935351
    • Galluzzi, L., Karp, M., 2006. Whole cell strategies based on lux genes for high throughput applications toward new antimicrobials. Comb. Chem. High Throughput Screen. 9, 501-514. (Pubitemid 44156708)
    • (2006) Combinatorial Chemistry and High Throughput Screening , vol.9 , Issue.7 , pp. 501-514
    • Galluzzi, L.1    Karp, M.2
  • 11
    • 77958151574 scopus 로고    scopus 로고
    • The global need for effective antibiotics: Challenges and recent advances
    • Hogberg, L.D., Heddini, A., Cars, O., 2010. The global need for effective antibiotics: challenges and recent advances. Trends Pharmacol. Sci. 31, 509-515.
    • (2010) Trends Pharmacol. Sci. , vol.31 , pp. 509-515
    • Hogberg, L.D.1    Heddini, A.2    Cars, O.3
  • 12
    • 84872861438 scopus 로고    scopus 로고
    • HTS assay validation
    • In: Sittampalam, G.S., Gal-Edd, N., Arkin, M., Auld, D., Austin, C., Bejcek, B., Glicksman, M., Inglese, J., Lemmon, V., Li, Z., McGee, J., McManus, O., Minor, L., Napper, A., Riss, T., Trask, O.J., Weidner, J. (Eds.),. Eli Lilly & Company and the National Center for Advancing Translational Sciences, Bethesda (MD)
    • Iversen, P.W., Beck, B., Chen, Y.F., Dere, W., Devanarayan, V., Eastwood, B.J., Farmen, M.W., Iturria, S.J., Montrose, C., Moore, R.A., Weidner, J.R., Sittampalam, G.S., 2004. HTS assay validation. In: Sittampalam, G.S., Gal-Edd, N., Arkin, M., Auld, D., Austin, C., Bejcek, B., Glicksman, M., Inglese, J., Lemmon, V., Li, Z., McGee, J., McManus, O., Minor, L., Napper, A., Riss, T., Trask, O.J., Weidner, J. (Eds.), Assay Guidance Manual. Eli Lilly & Company and the National Center for Advancing Translational Sciences, Bethesda (MD).
    • (2004) Assay Guidance Manual
    • Iversen, P.W.1    Beck, B.2    Chen, Y.F.3    Dere, W.4    Devanarayan, V.5    Eastwood, B.J.6    Farmen, M.W.7    Iturria, S.J.8    Montrose, C.9    Moore, R.A.10    Weidner, J.R.11    Sittampalam, G.S.12
  • 13
    • 0032213906 scopus 로고    scopus 로고
    • A recombinant Escherichia coli sensor strain for the detection of tetracyclines
    • Korpela, M.T., Kurittu, J.S., Karvinen, J.T., Karp, M.T., 1998. A recombinant Escherichia coli sensor strain for the detection of tetracyclines. Anal. Chem. 70, 4457-4462.
    • (1998) Anal. Chem. , vol.70 , pp. 4457-4462
    • Korpela, M.T.1    Kurittu, J.S.2    Karvinen, J.T.3    Karp, M.T.4
  • 14
    • 34250675757 scopus 로고    scopus 로고
    • Estimation of antimicrobial activity of selected non-antibiotic products
    • Kruszewska, H., Zareba, T., Tyski, S., 2006. Estimation of antimicrobial activity of selected non-antibiotic products. Acta Pol. Pharm. 63, 457-460.
    • (2006) Acta Pol. Pharm. , vol.63 , pp. 457-460
    • Kruszewska, H.1    Zareba, T.2    Tyski, S.3
  • 15
    • 79955666400 scopus 로고    scopus 로고
    • The WHO policy package to combat antimicrobial resistance
    • World Health Organization World Health Day Antimicrobial Resistance Technical Working Group
    • Leung, E., Weil, D.E., Raviglione, M., Nakatani, H., World Health Organization World Health Day Antimicrobial Resistance Technical Working Group, 2011. The WHO policy package to combat antimicrobial resistance. Bull. World Health Organ. 89, 390-392.
    • (2011) Bull. World Health Organ. , vol.89 , pp. 390-392
    • Leung, E.1    Weil, D.E.2    Raviglione, M.3    Nakatani, H.4
  • 16
    • 79955845844 scopus 로고    scopus 로고
    • Design and implementation of high throughput screening assays
    • Macarron, R., Hertzberg, R.P., 2011. Design and implementation of high throughput screening assays. Mol. Biotechnol. 47, 270-285.
    • (2011) Mol. Biotechnol. , vol.47 , pp. 270-285
    • MacArron, R.1    Hertzberg, R.P.2
  • 17
    • 0026071817 scopus 로고
    • Molecular biology of bacterial bioluminescence
    • Meighen, E.A., 1991. Molecular biology of bacterial bioluminescence. Microbiol. Rev. 55, 123-142. (Pubitemid 21895148)
    • (1991) Microbiological Reviews , vol.55 , Issue.1 , pp. 123-142
    • Meighen, E.A.1
  • 19
    • 33644504461 scopus 로고    scopus 로고
    • Antibacterial drug discovery-then, now and the genomics future
    • Monaghan, R.L., Barrett, J.F., 2006. Antibacterial drug discovery-then, now and the genomics future. Biochem. Pharmacol. 71, 901-909.
    • (2006) Biochem. Pharmacol. , vol.71 , pp. 901-909
    • Monaghan, R.L.1    Barrett, J.F.2
  • 20
    • 12944302098 scopus 로고    scopus 로고
    • Lack of development of new antimicrobial drugs: A potential serious threat to public health
    • DOI 10.1016/S1473-3099(05)01283-1, PII S1473309905012831
    • Norrby, S.R., Nord, C.E., Finch, R., European Society of Clinical Microbiology and Infectious Diseases, 2005. Lack of development of new antimicrobial drugs: a potential serious threat to public health. Lancet Infect. Dis. 5, 115-119. (Pubitemid 40174782)
    • (2005) Lancet Infectious Diseases , vol.5 , Issue.2 , pp. 115-119
    • Norrby, S.R.1    Nord, C.E.2    Finch, R.3
  • 21
    • 40949099893 scopus 로고    scopus 로고
    • New antibacterial agents for treating infections caused by multi-drug resistant gram-negative bacteria
    • DOI 10.1517/13543784.17.3.297
    • O'Neill, A.J., 2008. New antibacterial agents for treating infections caused by multidrug resistant Gram-negative bacteria. Expert Opin. Investig. Drugs 17, 297-302. (Pubitemid 351578182)
    • (2008) Expert Opinion on Investigational Drugs , vol.17 , Issue.3 , pp. 297-302
    • O'Neill, A.J.1
  • 23
    • 0025779537 scopus 로고
    • Mechanisms of bacterial resistance to non-antibiotics: Food additives and food and pharmaceutical preservatives
    • Russell, A.D., 1991. Mechanisms of bacterial resistance to non-antibiotics: food additives and food and pharmaceutical preservatives. J. Appl. Bacteriol. 71, 191-201.
    • (1991) J. Appl. Bacteriol. , vol.71 , pp. 191-201
    • Russell, A.D.1
  • 24
    • 34249800918 scopus 로고    scopus 로고
    • Microtitre plate-based antibacterial assay incorporating resazurin as an indicator of cell growth, and its application in the in vitro antibacterial screening of phytochemicals
    • DOI 10.1016/j.ymeth.2007.01.006, PII S1046202307000096, Natural Product Research: The Challenges Facing the Modern Researcher
    • Sarker, S.D., Nahar, L., Kumarasamy, Y., 2007. Microtitre plate-based antibacterial assay incorporating resazurin as an indicator of cell growth, and its application in the in vitro antibacterial screening of phytochemicals. Methods 42, 321-324. (Pubitemid 46856865)
    • (2007) Methods , vol.42 , Issue.4 , pp. 321-324
    • Sarker, S.D.1    Nahar, L.2    Kumarasamy, Y.3
  • 26
    • 39449103059 scopus 로고    scopus 로고
    • The epidemic of antibiotic-resistant infections: A call to action for the medical community from the infectious diseases society of America
    • DOI 10.1086/524891
    • Spellberg, B., Guidos, R., Gilbert, D., Bradley, J., Boucher, H.W., Scheld, W.M., Bartlett, J.G., Edwards Jr., J., Infectious Diseases Society of America, 2008. The epidemic of antibiotic-resistant infections: a call to action for the medical community from the Infectious Diseases Society of America. Clin. Infect. Dis. 46, 155-164. (Pubitemid 351269151)
    • (2008) Clinical Infectious Diseases , vol.46 , Issue.2 , pp. 155-164
    • Spellberg, B.1    Guidos, R.2    Gilbert, D.3    Bradley, J.4    Boucher, H.W.5    Scheld, W.M.6    Bartlett, J.G.7    Edwards Jr., J.8
  • 27
    • 0035189959 scopus 로고    scopus 로고
    • Measurement of effects of antibiotics in bioluminescent Staphylococcus aureus RN4220
    • DOI 10.1128/AAC.45.12.3456-3461.2001
    • Tenhami, M., Hakkila, K., Karp, M., 2001. Measurement of the effects of antibiotics in bioluminescent Staphylococcus aureus RN4220. Antimicrob. Agents Chemother. 45, 3456-3461. (Pubitemid 33107862)
    • (2001) Antimicrobial Agents and Chemotherapy , vol.45 , Issue.12 , pp. 3456-3461
    • Tenhami, M.1    Hakkila, K.2    Karp, M.3
  • 28
    • 84858282874 scopus 로고    scopus 로고
    • Accelerating resistance, inadequate antibacterial drug pipelines and international responses
    • Theuretzbacher, U., 2012. Accelerating resistance, inadequate antibacterial drug pipelines and international responses. Int. J. Antimicrob. Agents 39, 295-299.
    • (2012) Int. J. Antimicrob. Agents , vol.39 , pp. 295-299
    • Theuretzbacher, U.1
  • 29
    • 4944225004 scopus 로고    scopus 로고
    • The antibacterial principle of Caesalpina sappan
    • DOI 10.1002/ptr.1524
    • Xu, H.X., Lee, S.F., 2004. The antibacterial principle of Caesalpina sappan. Phytother. Res. 18, 647-651. (Pubitemid 39329715)
    • (2004) Phytotherapy Research , vol.18 , Issue.8 , pp. 647-651
    • Xu, H.-X.1    Lee, S.F.2
  • 30
    • 0033003760 scopus 로고    scopus 로고
    • A simple statistical parameter for use in evaluation and validation of high throughput screening assays
    • DOI 10.1177/108705719900400206
    • Zhang, J.H., Chung, T.D., Oldenburg, K.R., 1999. A simple statistical parameter for use in evaluation and validation of high throughput screening assays. J. Biomol. Screen. 4, 67-73. (Pubitemid 29278954)
    • (1999) Journal of Biomolecular Screening , vol.4 , Issue.2 , pp. 67-73
    • Zhang, J.-H.1    Chung, T.D.Y.2    Oldenburg, K.R.3
  • 31
    • 69849091689 scopus 로고    scopus 로고
    • Brazilein inhibits survivin protein and mRNA expression and induces apoptosis in hepatocellular carcinoma HepG2 cells
    • Zhong, X., Wu, B., Pan, Y.J., Zheng, S., 2009. Brazilein inhibits survivin protein and mRNA expression and induces apoptosis in hepatocellular carcinoma HepG2 cells. Neoplasma 56, 387-392.
    • (2009) Neoplasma , vol.56 , pp. 387-392
    • Zhong, X.1    Wu, B.2    Pan, Y.J.3    Zheng, S.4


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