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Volumn 7, Issue 6, 2002, Pages 526-530

High-Throughput Fluorescence Polarization Method for Identification of FKBP12 Ligands

Author keywords

[No Author keywords available]

Indexed keywords

FK 506 BINDING PROTEIN; HISTIDINE; LIGAND; RECOMBINANT PROTEIN;

EID: 0642286481     PISSN: 10870571     EISSN: None     Source Type: Journal    
DOI: 10.1177/1087057102238626     Document Type: Article
Times cited : (45)

References (29)
  • 2
    • 0028358901 scopus 로고
    • Stabilization of calcium release channel (ryanodine receptor) function by FK506-binding protein
    • Brillantes AB, Ondrias K, Scott A, Kobrinsky E, Ondriasova E, Moschella MC, et al: Stabilization of calcium release channel (ryanodine receptor) function by FK506-binding protein. Cell 1994;77:513-523.
    • (1994) Cell , vol.77 , pp. 513-523
    • Brillantes, A.B.1    Ondrias, K.2    Scott, A.3    Kobrinsky, E.4    Ondriasova, E.5    Moschella, M.C.6
  • 4
    • 0028108801 scopus 로고
    • Specific interaction of type I receptors of the TGF-beta family with the immunophilin FKBP-12
    • Wang T, Donahoe PK, Zervos AS: Specific interaction of type I receptors of the TGF-beta family with the immunophilin FKBP-12. Science 1994;265:674-676.
    • (1994) Science , vol.265 , pp. 674-676
    • Wang, T.1    Donahoe, P.K.2    Zervos, A.S.3
  • 5
    • 0028202076 scopus 로고
    • Immunosuppressant FK506 promotes neurite outgrowth in cultures of PC 12 cells and sensory ganglia
    • Lyons WE, George EB, Dawson TM, Steiner JP: Immunosuppressant FK506 promotes neurite outgrowth in cultures of PC 12 cells and sensory ganglia. Proc Nail Acad Sci USA 1994;91:3191-3195.
    • (1994) Proc Nail Acad Sci USA , vol.91 , pp. 3191-3195
    • Lyons, W.E.1    George, E.B.2    Dawson, T.M.3    Steiner, J.P.4
  • 7
    • 0028956418 scopus 로고
    • Neuronal regeneration enhances the expression of the immunophilin FKBP-12
    • Lyons WE, Steiner JP, Snyder SH, Dawson TM: Neuronal regeneration enhances the expression of the immunophilin FKBP-12. J Neiuvsci 1995;15:2985-2994.
    • (1995) J Neiuvsci , vol.15 , pp. 2985-2994
    • Lyons, W.E.1    Steiner, J.P.2    Snyder, S.H.3    Dawson, T.M.4
  • 9
    • 0027192328 scopus 로고
    • Specific interaction of the cyclophilincyclosporin complex with the B subunit of calcineurin
    • Li W, Handschumacher RE: Specific interaction of the cyclophilincyclosporin complex with the B subunit of calcineurin. J Biol Cliem 1993:268:14040-14044.
    • (1993) J Biol Cliem , vol.268 , pp. 14040-14044
    • Li, W.1    Handschumacher, R.E.2
  • 11
    • 0344265121 scopus 로고    scopus 로고
    • Novel neuroimmunophilin ligands for FKBP-12 possess potent neurotrophic activity in the mouse MPTP model of Parkinson's disease
    • Ross DT, Valentine HL, Guo H, Hamilton GS, Huang W, Suzdak PD, et al: Novel neuroimmunophilin ligands for FKBP-12 possess potent neurotrophic activity in the mouse MPTP model of Parkinson's disease. Society for Neuroscie nee 1996:297.14.
    • (1996) Society for Neuroscie Nee , pp. 29714
    • Ross, D.T.1    Valentine, H.L.2    Guo, H.3    Hamilton, G.S.4    Huang, W.5    Suzdak, P.D.6
  • 12
    • 0030975605 scopus 로고    scopus 로고
    • Neurotrophic actions of nonimmunosuppressive analogues of immunosuppressive drugs FK506, rapamycin and cyclosporin a
    • Steiner JP, Connolly MA, Valentine HI, Hamilton GS, Dawson TM, Hester L, et al: Neurotrophic actions of nonimmunosuppressive analogues of immunosuppressive drugs FK506, rapamycin and cyclosporin A. Nature Med 1997;3:421-428.
    • (1997) Nature Med , vol.3 , pp. 421-428
    • Steiner, J.P.1    Connolly, M.A.2    Valentine, H.I.3    Hamilton, G.S.4    Dawson, T.M.5    Hester, L.6
  • 13
    • 33749220854 scopus 로고
    • FK506, an immunosuppressent, increases functional recovery and axonal regeneration in the rat following axotomy of the sciatic nerve
    • Gold BG, Storm-Dickerson T, Austin DR, Katoh K: FK506, an immunosuppressent, increases functional recovery and axonal regeneration in the rat following axotomy of the sciatic nerve. Society for Nenroscience 1993:543.18.
    • (1993) Society for Nenroscience , pp. 54318
    • Gold, B.G.1    Storm-Dickerson, T.2    Austin, D.R.3    Katoh, K.4
  • 15
    • 0025868143 scopus 로고
    • Determination of kinetic constants for peptidyl-prolyl cis-trans isomerases by an improved spectrophotometric assay
    • Kofron JL, Kuzmic P, Kishore V, Colon-Bonilla E, Rich DH: Determination of kinetic constants for peptidyl-prolyl cis-trans isomerases by an improved spectrophotometric assay. Biochemistry 1991;30:6127-6134.
    • (1991) Biochemistry , vol.30 , pp. 6127-6134
    • Kofron, J.L.1    Kuzmic, P.2    Kishore, V.3    Colon-Bonilla, E.4    Rich, D.H.5
  • 18
    • 0032943217 scopus 로고    scopus 로고
    • High throughput scintillation proximity assay for the identification of FKBP-12 ligands
    • Graziani F, Aldegheri L, Terstappen GC: High throughput scintillation proximity assay for the identification of FKBP-12 ligands. J Biomol Screening 1999;4:3-7.
    • (1999) J Biomol Screening , vol.4 , pp. 3-7
    • Graziani, F.1    Aldegheri, L.2    Terstappen, G.C.3
  • 19
    • 77956786849 scopus 로고
    • Rotational Brownian motion and polarization of the fluorescence in solutions
    • Weber G: Rotational Brownian motion and polarization of the fluorescence in solutions. Adv Protein Cliem 1953;8:415. l
    • (1953) Adv Protein Cliem , vol.8
    • Weber, G.1
  • 20
    • 0000547815 scopus 로고
    • Quantification of the antigen-antibody reaction by the polarization of fluorescence
    • Dandliker WB, Feigen GA: Quantification of the antigen-antibody reaction by the polarization of fluorescence. Biochem Biophys Res Commun 1961;5:299-304.
    • (1961) Biochem Biophys Res Commun , vol.5 , pp. 299-304
    • Dandliker, W.B.1    Feigen, G.A.2
  • 23
    • 0001019593 scopus 로고
    • Design, synthesis, and kinetic evaluation of high-affinity FKBP ligands and the X-ray crystal structures of their complexes with FKBP 12
    • Holt DA, Luengo JI, Yamashita DS, Oh HJ, Konialian AL, Yen HK, et al: Design, synthesis, and kinetic evaluation of high-affinity FKBP ligands and the X-ray crystal structures of their complexes with FKBP 12. J Am ChemSoc 1993;115:9925-9938.
    • (1993) J Am ChemSoc , vol.115 , pp. 9925-9938
    • Holt, D.A.1    Luengo, J.I.2    Yamashita, D.S.3    Oh, H.J.4    Konialian, A.L.5    Yen, H.K.6
  • 25
    • 0030799884 scopus 로고    scopus 로고
    • Neuroimmunophilin ligands and novel therapeutics for the treatment of degenerative disorders of the nervous system
    • Hamilton GS, Steiner JP: Neuroimmunophilin ligands and novel therapeutics for the treatment of degenerative disorders of the nervous system. Curr Pharin Des 1997;3:405-428.
    • (1997) Curr Pharin Des , vol.3 , pp. 405-428
    • Hamilton, G.S.1    Steiner, J.P.2
  • 26
    • 0033773937 scopus 로고    scopus 로고
    • Fluorescence polarization and anisotropy in high throughput screening: Perspectives and primer
    • Owicki JC: Fluorescence polarization and anisotropy in high throughput screening: perspectives and primer. J Biomol Screen 2000;5:297-306.
    • (2000) J Biomol Screen , vol.5 , pp. 297-306
    • Owicki, J.C.1
  • 27
    • 0019813536 scopus 로고
    • Corrected equations for the calculation of protein-ligand binding results from fluorescence polarization data
    • Rajkowski KM, Cittanova N: Corrected equations for the calculation of protein-ligand binding results from fluorescence polarization data. J Theor Biol 1981 ;93:691 -696.
    • (1981) J Theor Biol , vol.93 , pp. 691-696
    • Rajkowski, K.M.1    Cittanova, N.2
  • 28
    • 12644257556 scopus 로고    scopus 로고
    • Neurotrophic immunophilin ligands stimulate structural and functional recovery in neurodegenerative animal models
    • Steiner JP, Hamilton GS, Ross DT, Valentine HL, Guo HZ, Connolly MA, et al: Neurotrophic immunophilin ligands stimulate structural and functional recovery in neurodegenerative animal models. Proc Nail Acad Sci USA 1997;94:2019-2024.
    • (1997) Proc Nail Acad Sci USA , vol.94 , pp. 2019-2024
    • Steiner, J.P.1    Hamilton, G.S.2    Ross, D.T.3    Valentine, H.L.4    Guo, H.Z.5    Connolly, M.A.6


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.