Discovery of protein-protein interaction inhibitors of replication protein A

ACS Medicinal Chemistry Letters

Volumn 4, Issue 7, 2013, Pages 601-605

  Patrone, James D ^a   Kennedy, J Phillip ^a   Frank, Andreas O ^a,c   Feldkamp, Michael D ^a   Vangamudi, Bhavatarini ^a   Pelz, Nicholas F ^a   Rossanese, Olivia W ^a   Waterson, Alex G ^a,b   Chazin, Walter J ^a,b   Fesik, Stephen W ^a,b  

^a VANDERBILT UNIVERSITY SCHOOL OF MEDICINE   (United States)

^b VANDERBILT UNIVERSITY   (United States)

^c NOVARTIS INSTITUTES FOR BIOMEDICAL RESEARCH   (United States)

Author keywords

DNA damage; fragment based discovery; Replication protein A

Indexed keywords

BENZOTHIOPHENE DERIVATIVE; REPLICATION FACTOR A; TRIAZOLE DERIVATIVE;

ARTICLE; BINDING AFFINITY; DNA DAMAGE; PRIORITY JOURNAL; PROTEIN BINDING; PROTEIN DOMAIN; PROTEIN PROTEIN INTERACTION; SENSITIVITY ANALYSIS; STRUCTURE ACTIVITY RELATION;

EID: 84880156207     PISSN: None     EISSN: 19485875     Source Type: Journal    
DOI: 10.1021/ml400032y     Document Type: Article

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