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Bioorganic and Medicinal Chemistry Letters

Volumn 23, Issue 15, 2013, Pages 4408-4412

Phosphinic acid-based inhibitors of tubulin polyglutamylases

(4) Liu, Yanjie a Garnham, Christopher P b Roll Mecak, Antonina b Tanner, Martin E a

a UNIVERSITY OF BRITISH COLUMBIA (Canada)

b NATIONAL INSTITUTE OF NEUROLOGICAL DISORDERS AND STROKE (United States)

Author keywords

Inhibitor; Ligase; Phosphinic acid; Post translational modification; Tubulin

Indexed keywords

ENZYME INHIBITOR; GLUTAMIC ACID; MICROTUBULE ASSOCIATED PROTEIN; PEPTIDE DERIVATIVE; PHOSPHONIC ACID DERIVATIVE; TUBULIN; TUBULIN POLYGLUTAMYLASE INHIBITOR; UNCLASSIFIED DRUG;

ARTICLE; CARBOXY TERMINAL SEQUENCE; CHEMICAL REACTION; CONFORMATIONAL TRANSITION; DEGLUTAMYLATION; DRUG POTENCY; DRUG SYNTHESIS; ENZYME INHIBITION; ENZYME MECHANISM; ENZYME SUBSTRATE; IC 50; METASTASIS; MOUSE; NERVE CELL DIFFERENTIATION; NONHUMAN; POLYGLUTAMYLATION; PROTEIN FUNCTION; PROTEIN PROCESSING; STRUCTURE ACTIVITY RELATION;

ANIMALS; ENZYME INHIBITORS; MICE; PEPTIDE SYNTHASES; PHOSPHINIC ACIDS; PROTEIN BINDING;

EID: 84879694858 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2013.05.069 Document Type: Article

Times cited : (11)

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