Nonsteroidal anti-inflammatory drugs and other anthranilic acids inhibit the Na+/dicarboxylate symporter from Staphylococcus aureus

Biochemistry

Volumn 52, Issue 17, 2013, Pages 2924-2932

  Pajor, Ana M ^a   Sun, Nina N ^a  

^a UNIVERSITY OF CALIFORNIA SAN DIEGO   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ALLOSTERIC INHIBITOR; ANTHRANILIC ACID; CO-TRANSPORTERS; DIVALENT ANIONS; HILL COEFFICIENT; NON-STEROIDAL ANTI-INFLAMMATORY DRUGS; STAPHYLOCOCCUS AUREUS;

AMINO ACIDS; BACTERIA; MAMMALS; SODIUM;

CARBOXYLATION;

ANTHRANILIC ACID DERIVATIVE; CYSTEINE; DICARBOXYLATE TRANSPORTER; DICARBOXYLIC ACID; FLUFENAMIC ACID; MEFENAMIC ACID; NIFLUMIC ACID; NONSTEROID ANTIINFLAMMATORY AGENT; SODIUM ION; SUCCINIC ACID;

ARTICLE; BACTERIAL STRAIN; BINDING SITE; CHEMICAL REACTION KINETICS; CONTROLLED STUDY; DRUG INHIBITION; ESCHERICHIA COLI; HUMAN; HUMAN CELL; IC 50; MEMBRANE VESICLE; MUTANT; NONHUMAN; PRIORITY JOURNAL; STAPHYLOCOCCUS AUREUS;

ANTI-INFLAMMATORY AGENTS, NON-STEROIDAL; CELL LINE; DICARBOXYLIC ACID TRANSPORTERS; HUMANS; KINETICS; ORTHO-AMINOBENZOATES; STAPHYLOCOCCUS AUREUS; SYMPORTERS;

MAMMALIA; STAPHYLOCOCCUS AUREUS;

EID: 84877040978     PISSN: 00062960     EISSN: 15204995     Source Type: Journal    
DOI: 10.1021/bi301611u     Document Type: Article

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