Kappa-opioid receptor-selective dicarboxylic ester-derived salvinorin A ligands

Bioorganic and Medicinal Chemistry Letters

Volumn 23, Issue 10, 2013, Pages 2860-2862

  Polepally, Prabhakar R ^a   White, Kate ^b   Vardy, Eyal ^b   Roth, Bryan L ^b   Ferreira, Daneel ^a   Zjawiony, Jordan K ^a  

^a UNIVERSITY OF MISSISSIPPI   (United States)

^b UNIVERSITY OF NORTH CAROLINA SCHOOL OF MEDICINE   (United States)

Author keywords

Salvia divinorum Salvinorin A and B Dicarboxylic ester type ligands Kappa opioid receptor agonists

Indexed keywords

DELTA OPIATE RECEPTOR; DICARBOXYLIC ACID; KAPPA OPIATE RECEPTOR; MU OPIATE RECEPTOR; SALVINORIN A;

ARTICLE; BINDING AFFINITY; DRUG SYNTHESIS; NONHUMAN;

DITERPENES, CLERODANE; DOSE-RESPONSE RELATIONSHIP, DRUG; DRUGS, CHINESE HERBAL; HEK293 CELLS; HUMANS; MOLECULAR CONFORMATION; RECEPTORS, OPIOID, KAPPA; SALVIA; STRUCTURE-ACTIVITY RELATIONSHIP;

SALVIA DIVINORUM;

EID: 84876686778     PISSN: 0960894X     EISSN: 14643405     Source Type: Journal    
DOI: 10.1016/j.bmcl.2013.03.111     Document Type: Article

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