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Bioorganic and Medicinal Chemistry Letters

Volumn 23, Issue 10, 2013, Pages 2920-2924

Discovery of novel orally bioavailable GPR40 agonists

(10) Lu, Hejun a Fei, Hongbo a Yang, Fanglong a Zheng, Suxin a Hu, Qiyue a Zhang, Lei a Yuan, Jijun a Feng, Jun a Sun, Piaoyang a Dong, Qing a

a Shanghai Hengrui Pharmaceuticals Co Ltd (China)

Author keywords

Diabetes GPR40 Agonist Orally bioavailable Species specificity

Indexed keywords

G PROTEIN COUPLED RECEPTOR 40; G PROTEIN COUPLED RECEPTOR 40 AGONIST; UNCLASSIFIED DRUG;

ANIMAL EXPERIMENT; ARTICLE; DRUG BIOAVAILABILITY; DRUG EFFICACY; IN VIVO STUDY; NONHUMAN; RHESUS MONKEY;

ADMINISTRATION, ORAL; ANIMALS; BENZOFURANS; DIABETES MELLITUS, TYPE 2; DISEASE MODELS, ANIMAL; DOGS; DOSE-RESPONSE RELATIONSHIP, DRUG; DRUG DISCOVERY; HUMANS; MACACA MULATTA; MICE; MODELS, MOLECULAR; MOLECULAR STRUCTURE; RATS; RECEPTORS, G-PROTEIN-COUPLED; SMALL MOLECULE LIBRARIES; STRUCTURE-ACTIVITY RELATIONSHIP; SULFONES;

MACACA MULATTA;

EID: 84876665196 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2013.03.060 Document Type: Article

Times cited : (15)

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