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Bioorganic and Medicinal Chemistry Letters

Volumn 23, Issue 9, 2013, Pages 2647-2652

Carbonic anhydrase inhibitors: Inhibition of the β-class enzyme from the pathogenic yeast Candida glabrata with sulfonamides, sulfamates and sulfamides

(6) Vullo, Daniela a Leewattanapasuk, Worraanong b Mühlschlegel, Fritz A b Mastrolorenzo, Antonio a Capasso, Clemente c Supuran, Claudiu T a

a UNIVERSITY OF FLORENCE (Italy)

b UNIVERSITY OF KENT (United Kingdom)

c INSTITUTE OF PROTEIN BIOCHEMISTRY (Italy)

Author keywords

Class enzyme; Antifungal; Carbonic anhydrase; Inhibitor; Sulfamate; Sulfamide; Sulfonamide

Indexed keywords

ACETAZOLAMIDE; ANTIFUNGAL AGENT; BRINZOLAMIDE; CARBONATE DEHYDRATASE; CARBONATE DEHYDRATASE INHIBITOR; CELECOXIB; CGNCE 103; DICLOFENAMIDE; DORZOLAMIDE; ETHOXZOLAMIDE; FUNGAL ENZYME; INDISULAM; METHAZOLAMIDE; SULFAMIDE DERIVATIVE; SULFONAMIDE; SULPIRIDE; TOPIRAMATE; UNCLASSIFIED DRUG; VALDECOXIB; ZONISAMIDE;

ANTIFUNGAL RESISTANCE; ARTICLE; CANDIDA GLABRATA; ENZYME INHIBITION; FUNGUS GROWTH; FUNGUS ISOLATION; NONHUMAN;

ACETAZOLAMIDE; AMINO ACID SEQUENCE; ANTIFUNGAL AGENTS; CANDIDA GLABRATA; CARBONIC ANHYDRASE INHIBITORS; CARBONIC ANHYDRASES; HUMANS; KINETICS; MOLECULAR SEQUENCE DATA; PHYLOGENY; PROTEIN BINDING; SEQUENCE ALIGNMENT; STRUCTURE-ACTIVITY RELATIONSHIP; SULFONAMIDES; SULFONIC ACIDS;

CANDIDA GLABRATA;

EID: 84876100737 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2013.02.092 Document Type: Article

Times cited : (43)

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