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Bioorganic and Medicinal Chemistry Letters

Volumn 23, Issue 6, 2013, Pages 1760-1762

Design, synthesis and aromatase inhibitory activities of novel indole-imidazole derivatives

(6) Wang, Rui a Shi, Hong Fan a Zhao, Jing Feng a He, Yan Ping a Zhang, Hong Bin a Liu, Jian Ping a

a YUNNAN UNIVERSITY (China)

Author keywords

Aromatase inhibitor (AI); Breast cancer; Indole imidazole derivatives; Structure activity relationship; Synthesis

Indexed keywords

AROMATASE INHIBITOR; IMIDAZOLE DERIVATIVE; INDOLE DERIVATIVE; LETROZOLE;

ALDOL REACTION; ARTICLE; DRUG DESIGN; DRUG POTENCY; DRUG SYNTHESIS; ENZYME ACTIVITY; HUMAN; HUMAN CELL; IC 50; IN VITRO STUDY; STRUCTURE ACTIVITY RELATION;

AROMATASE; AROMATASE INHIBITORS; CRYSTALLOGRAPHY, X-RAY; DRUG DESIGN; IMIDAZOLES; INDOLES; MOLECULAR CONFORMATION; PROTEIN BINDING; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 84874667729 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2013.01.045 Document Type: Article

Times cited : (36)

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