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Volumn 330, Issue 5, 1997, Pages 141-145

Synthesis and in vitro evaluation of 3-(1-Azolylmethyl)-1H-indoles and 3-(1-azoly1-1-phenylmethyl)-1H-indoles as inhibitors of P450 arom

(8) Le Borgne, Marc a Marchand, Pascal a Duflos, Muriel a Delevoye Seiller, Bénédicte a Piessard Robert, Sylvie a Le Baut, Guillaume a Hartmann, Rolf W b Palzer, M b

a UNIVERSITÉ DE NANTES (France)

b SAARLAND UNIVERSITY (Germany)

Author keywords

Azolyl substituted indoles; Estrogen dependent disease; Nonsteroidal P450 arom inhibitors

Indexed keywords

1 (4 FLUOROBENZYL) 3 (1H 1 IMIDAZOLYLMETHYL) 1H INDOLE; 3 (1 AZOLYLMETHYL) 1H INDOLE DERIVATIVE; AMINOGLUTETHIMIDE; AROMATASE INHIBITOR; CYTOCHROME P450 INHIBITOR; ESTROGEN; INDOLE DERIVATIVE; LIAROZOLE; TRIAZOLE DERIVATIVE; UNCLASSIFIED DRUG;

ADVANCED CANCER; ARTICLE; BREAST CARCINOMA; DRUG POTENCY; DRUG SYNTHESIS; ENZYME INACTIVATION; ESTROGEN SYNTHESIS; PRIORITY JOURNAL;

AROMATASE INHIBITORS; ENZYME INHIBITORS; INDOLES; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 0030746262 PISSN: 03656233 EISSN: None Source Type: Journal
DOI: 10.1002/ardp.19973300506 Document Type: Article

Times cited : (59)

References (15)

1
- 0025728051
- P. Labrie, Mol. Cell. Endocrinol. 1991, 78, C113 -C118.
- (1991) Mol. Cell. Endocrinol. , vol.78
- Labrie, P.¹

2
- 0027985313
- B. Svenstrup, J. Herrstedt, N. Brünner, P. Bennett, H. Wachmann, P. Dombernowsky, Eur. J. Cancer 1994, 30A, 1254-1258.
- (1994) Eur. J. Cancer , vol.30 A , pp. 1254-1258
- Svenstrup, B.¹ Herrstedt, J.² Brünner, N.³ Bennett, P.⁴ Wachmann, H.⁵ Dombernowsky, P.⁶

3
- 0343885445
- Abst 74
- K. Fox, J. Glick, J. Schulz, L. Demers, G. Conner, R. Reynolds, E. Mitchell, R. Capizzi, P. Schein, Proc. Amer. Soc. Clin. Oncol. 1995, 14, Abst 74.
- (1995) Proc. Amer. Soc. Clin. Oncol. , vol.14
- Fox, K.¹ Glick, J.² Schulz, J.³ Demers, L.⁴ Conner, G.⁵ Reynolds, R.⁶ Mitchell, E.⁷ Capizzi, R.⁸ Schein, P.⁹

4
- 0028946611
- P.E. Goss, R.M. Clark, U. Ambus, H.A.E. Weizel, N.A. Wadden, M. Crump, D. Walde, L.M. Tye, R. De Coster, J. Bruynseels, Clin. Cancer Res. 1995, 1, 287-294.
- (1995) Clin. Cancer Res. , vol.1 , pp. 287-294
- Goss, P.E.¹ Clark, R.M.² Ambus, U.³ Weizel, H.A.E.⁴ Wadden, N.A.⁵ Crump, M.⁶ Walde, D.⁷ Tye, L.M.⁸ De Coster, R.⁹ Bruynseels, J.¹⁰

5
- 0028943384
- A. Lipton, L.M. Demers, H.A. Harvey, K.B. Kambic, H. Grossberg, C. Brady, H. Adlercruetz, P.F. Trunet, R.J. Santen, Cancer 1995, 75, 2132-2138.
- (1995) Cancer , vol.75 , pp. 2132-2138
- Lipton, A.¹ Demers, L.M.² Harvey, H.A.³ Kambic, K.B.⁴ Grossberg, H.⁵ Brady, C.⁶ Adlercruetz, H.⁷ Trunet, P.F.⁸ Santen, R.J.⁹

6
- 0028838392
- M. Kudoh, Y. Susaki, Y. Ideyama, T. Nanya, M. Okada, H. Shikama, T. Fujikura, J. Steroid Biochem. Mol. Biol. 1995, 54, 265-271.
- (1995) J. Steroid Biochem. Mol. Biol. , vol.54 , pp. 265-271
- Kudoh, M.¹ Susaki, Y.² Ideyama, Y.³ Nanya, T.⁴ Okada, M.⁵ Shikama, H.⁶ Fujikura, T.⁷

7
- 0343885443
- Abst 175
- J. Wolter, N. Robert, H. Harvey, I. Berkowitz, P. V. Plourde, Proc. Amer. Soc. Clin. Oncol. 1995, 14, Abst 175.
- (1995) Proc. Amer. Soc. Clin. Oncol. , vol.14
- Wolter, J.¹ Robert, N.² Harvey, H.³ Berkowitz, I.⁴ Plourde, P.V.⁵

8
- 0026742178
- W. Wouters, J. Van Dun, A. Dillen, M-C. Coene, W. Cools, R. De Coster, Cancer Res. 1992, 52, 2841-2846.
- (1992) Cancer Res. , vol.52 , pp. 2841-2846
- Wouters, W.¹ Van Dun, J.² Dillen, A.³ Coene, M.-C.⁴ Cools, W.⁵ De Coster, R.⁶

9
- 0021232351
- V. Cavrini, R. Gatti, P. Roveri, M.R. Cesaroni, Arch. Pharm. 1984, 317, 662-668.
- (1984) Arch. Pharm. , vol.317 , pp. 662-668
- Cavrini, V.¹ Gatti, R.² Roveri, P.³ Cesaroni, M.R.⁴

10
- 0025157171
- C.D. Jones, M.A. Winter, K.S. Hirsch, N. Stamm, H.M. Taylor, H.E. Holden, J.D. Davenport, E.V. Krumkalns, R.G. Suhr, J. Med. Chem. 1990, 33, 416-429.
- (1990) J. Med. Chem. , vol.33 , pp. 416-429
- Jones, C.D.¹ Winter, M.A.² Hirsch, K.S.³ Stamm, N.⁴ Taylor, H.M.⁵ Holden, H.E.⁶ Davenport, J.D.⁷ Krumkalns, E.V.⁸ Suhr, R.G.⁹

11
- 0026787091
- S. Massa, R. Di Santo, A. Retico, M. Artico, N. Simonetti, G. Fabrizi, D. Lamba, Eur. J. Med. Chem. 1992, 27, 495-502,
- (1992) Eur. J. Med. Chem. , vol.27 , pp. 495-502
- Massa, S.¹ Di Santo, R.² Retico, A.³ Artico, M.⁴ Simonetti, N.⁵ Fabrizi, G.⁶ Lamba, D.⁷

12
- 0025755870
- M.R. Bell, T.E. D'Ambra, V. Kumar, M.A. Eissenstat, J.L. Herrmann Jr., J.R. Wetzel, D. Rosi, R.E. Philion, S.J. Daum, D.J. Hlasta, R.K. Kullnig, J.H. Ackerman, D.R. Haubrich, D.A. Luttinger, E.R. Baizman, M.S. Miller, S.J. Ward, J. Med. Chem. 1991, 34, 1099-1110.
- (1991) J. Med. Chem. , vol.34 , pp. 1099-1110
- Bell, M.R.¹ D'Ambra, T.E.² Kumar, V.³ Eissenstat, M.A.⁴ Herrmann Jr., J.L.⁵ Wetzel, J.R.⁶ Rosi, D.⁷ Philion, R.E.⁸ Daum, S.J.⁹ Hlasta, D.J.¹⁰ Kullnig, R.K.¹¹ Ackerman, J.H.¹² Haubrich, D.R.¹³ Luttinger, D.A.¹⁴ Baizman, E.R.¹⁵ Miller, M.S.¹⁶ Ward, S.J.¹⁷

13
- 0016293443
- E.A. Thompson Jr., P.K. Siiteri, J. Biol. Chem. 1974, 249, 5364-5372.
- (1974) J. Biol. Chem. , vol.249 , pp. 5364-5372
- Thompson Jr., E.A.¹ Siiteri, P.K.²

14
- 0343013962
- K. Takushi, T. Fujimoto, Synth. Comm. 1987, 17, 396-397.
- (1987) Synth. Comm. , vol.17 , pp. 396-397
- Takushi, K.¹ Fujimoto, T.²

15
- 0022470925
- R.W. Hartmann, C. Batzl, J. Med. Chem. 1986, 29, 1362-1369.
- (1986) J. Med. Chem. , vol.29 , pp. 1362-1369
- Hartmann, R.W.¹ Batzl, C.²

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