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Bioorganic and Medicinal Chemistry Letters

Volumn 23, Issue 6, 2013, Pages 1891-1895

Synthesis and evaluation of methylsulfonylnitrobenzamides (MSNBAs) as inhibitors of the thyroid hormone receptor-coactivator interaction

(5) Hwang, Jong Yeon a Attia, Ramy R a Carrillo, Angela K a Connelly, Michele C a Guy, R Kiplin a

a ST JUDE CHILDREN S RESEARCH HOSPITAL (United States)

Author keywords

Coactivator; Inhibitor; Protein interaction; Thyroid

Indexed keywords

HORMONE ANTAGONIST; METHYLSULFONYLNITROBENZOATE DERIVATIVE; NITROBENZOIC ACID DERIVATIVE; THIAZOLE; THYROID HORMONE RECEPTOR; UNCLASSIFIED DRUG;

ARTICLE; CONFORMATIONAL TRANSITION; DRUG CYTOTOXICITY; DRUG SCREENING; DRUG SYNTHESIS; FLUORESCENCE POLARIZATION; HYDROPHOBICITY; IC 50; LIGAND BINDING; OXIDATION; PROCESS OPTIMIZATION; PROTEIN PROTEIN INTERACTION; SIGNAL TRANSDUCTION; STATIC ELECTRICITY;

BENZAMIDES; CELL SURVIVAL; HEP G2 CELLS; HUMANS; NUCLEAR RECEPTOR COACTIVATOR 1; PROTEIN INTERACTION MAPS; RECEPTORS, THYROID HORMONE; STRUCTURE-ACTIVITY RELATIONSHIP; THIAZOLES; TRANSFECTION;

EID: 84874656022 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2012.12.055 Document Type: Article

Times cited : (6)

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