Skin accumulation and penetration of a hydrophilic compound by a novel gemini surfactant, sodium dilauramidoglutamide lysine

International Journal of Pharmaceutics

Volumn 443, Issue 1-2, 2013, Pages 288-292

  Hikima, Tomohiro ^a   Tamura, Yoshinaga ^b   Yamawaki, Yukio ^b   Yamamoto, Masashi ^b   Tojo, Kakuji ^a  

^a KYUSHU INSTITUTE OF TECHNOLOGY   (Japan)

^b Asahi Kasei Chemicals Corporation   (Japan)

Author keywords

Chemical enhancer; Gemini amphiphilic compound; Peptide; Sodium dilauramidoglutamide lysine

Indexed keywords

AMPHOPHILE; SODIUM DILAURAMIDOGLUTAMIDE LYSINE; SODIUM LAURAMIDOGLUTAMIDE; UNCLASSIFIED DRUG;

ARTICLE; CONCENTRATION (PARAMETERS); CONTROLLED STUDY; DRUG DISTRIBUTION; DRUG PENETRATION; HUMAN; HUMAN CELL; IN VITRO STUDY; LIMIT OF DETECTION; LOCAL THERAPY; PRIORITY JOURNAL; SKIN ABSORPTION; SKIN PENETRATION;

ASCORBIC ACID; CHROMATOGRAPHY, HIGH PRESSURE LIQUID; EXCIPIENTS; HUMANS; HYDROPHOBIC AND HYDROPHILIC INTERACTIONS; MODELS, BIOLOGICAL; MOLECULAR STRUCTURE; OLIGOPEPTIDES; SKIN; SKIN ABSORPTION; SURFACE-ACTIVE AGENTS; TIME FACTORS; TISSUE DISTRIBUTION;

EID: 84873999376     PISSN: 03785173     EISSN: 18733476     Source Type: Journal    
DOI: 10.1016/j.ijpharm.2012.12.034     Document Type: Article

References (24)

1. V. Andronis Design and evaluation of transdermal chlorpheniramine maleate drug delivery system Pharm. Acta Helv. 70 1995 301 306
2. C. Bombelli Gemini surfactant based carriers in gene and drug delivery Curr. Med. Chem. 16 2009 71 83
3. Z. Chen Determination of nanograms of proteins based on decreased resonance light scattering of zwitterionic gemini surfactant Anal. Biochem. 384 2009 337 342
4. EC 7th Amendment to the EC cosmetic Directive (L66/26-35) 27th February 2003, Brussels, Belgium 2003
5. I. Effendy, and H.I. Maibach Detergents and skin irritation Clin. Dermatol. 14 1996 15 21
6. J.Y. Fang Development and evaluation on transdermal delivery of enoxacin via chemical enhancers and physical iontophoresis J. Control. Rel. 54 1998 293 304
7. T. Hikima, and K. Tojo Binding of prednisolone and its ester prodrugs in the skin Pharm. Res. 14 1997 197 202
8. T. Hikima, and K. Tojo Skin models for percutaneous absorption Drug Deliv. Syst. 16 2001 179 181
9. M. Kumar Gemini amphiphiles: a novel class of nonviral gene delivery vectors Crit. Rev. Ther. Drug Carrier Syst. 27 2010 237 278
10. ® on the in vitro percutaneous penetration of compounds with different lipophilicities Int. J. Pharm. 202 2000 133 140
11. O. López Structural modifications in the stratum corneum by effect of different solubilizing agents: a study based on high-resolution low-temperature scanning electron microscopy Skin Pharmacol. Appl. Skin Physiol. 13 2000 265 272
12. F.M. Menger, and J.S. Keiper Gemini surfactants Angew. Chem. Int. Ed. Engl. 39 2000 1906 1920
13. F.M. Menger, and C.A. Littau Gemini surfactants: a new class of self-assembling molecule J. Am. Chem. Soc. 115 1993 10083 10090
14. Y. Mine Preparation of gemini-type amphiphiles bearing cyclitol head groups and their application as high-performance modifiers for lipases Carbohydr. Res. 39 2004 493 501
15. S. Mitragotri Synergistic effect of ultrasound and sodium lauryl sulfate on transdermal drug delivery J. Pharm. Sci. 89 2000 892 900
16. S.D. Palma Potential use of ascorbic acid-based surfactants as skin penetration enhancers Drug Dev. Ind. Pharm. 32 2000 821 827
17. N. Sekiguchi Study on novel peptide-based gemini amphiphilic compound, Pellicer L-30 and application to the cosmetic Fragrance J. 36 2008 67 74
18. H. Shibayama Permeation and metabolism of a novel ascorbic acid derivative, disodium isostearyl 2-O-l-ascorbyl phosphate, in human living skin equivalent models Skin Pharmacol. Physiol. 21 2008 235 243
19. J. Shokri The effect of surfactants on the skin penetration of diazepam Int. J. Pharm. 228 2001 99 107
20. K. Tojo Design and calibration of in vitro permeation apparatus Y.W. Chien, Transdermal Controlled Systemic Medications 1987 Mercel Dekker New York 127 158
21. K.P. Wilhelm Surfactant-induced stratum corneum hydration in vivo: prediction of the irritation potential of anionic surfactants J. Invest. Dermatol. 101 1993 310 315
22. I. Yamamoto Synthesis and characterization of a series of novel monoacylated ascorbic acid derivatives, 6-O-acyl-2-O-α-d-glucopyranosyl-l- ascorbic acids, as skin antioxidants J. Med. Chem. 45 2002 462 468
23. M. Yamamoto Oil gelation utilizing a novel gemini-type peptide amphiphilie Fragrance J. 37 2009 42 45
24. A.A. Yaroslavov Conventional and gemini surfactants embedded within bilayer membrane: contrasting behavior Chemistry 7 2001 4835 4843