Novel inhibitor of Y. pestis Dam

British Journal of Pharmacology

Volumn 168, Issue 1, 2013, Pages 172-188

  McKelvie, J C ^a   Richards, M I ^b   Harmer, J E ^a   Milne, T S ^b   Roach, P L ^a   Oyston, P C F ^b  

^a UNIVERSITY OF SOUTHAMPTON   (United Kingdom)

^b DEFENCE SCIENCE AND TECHNOLOGY LABORATORY   (United Kingdom)

Author keywords

DNA adenine methylation; siderophore; stibonic acid; type III secretion; Yersinia

Indexed keywords

4 STIBONOBENENESULFONIC ACID; ANTIBIOTIC AGENT; ARYL STIBONIC ACID DERIVATIVE; DNA; DNA ADENINE METHYLTRANSFERASE; IRON; UNCLASSIFIED DRUG; VIRULENCE FACTOR; ANTIINFECTIVE AGENT; PLAGUE VACCINE; SITE SPECIFIC DNA METHYLTRANSFERASE (ADENINE SPECIFIC);

ARTICLE; BACTERIAL VIRULENCE; BACTERIUM CULTURE; CELLULAR SECRETION; COMPETITIVE INHIBITION; CONTROLLED STUDY; DNA METHYLATION; DRUG IDENTIFICATION; ENZYME INHIBITION; GENE EXPRESSION; GENETIC ANALYSIS; HIGH THROUGHPUT SCREENING; IN VITRO STUDY; NONHUMAN; PHENOTYPE; PRIORITY JOURNAL; STRUCTURE ACTIVITY RELATION; TRANSCRIPTIONAL ANALYSIS; YERSINIA PESTIS; CHEMISTRY; DRUG ANTAGONISM; DRUG EFFECT; ENZYMOLOGY; GENE EXPRESSION PROFILING; GENETICS; HUMAN; METABOLISM; MICROBIAL SENSITIVITY TEST; PATHOGENICITY; VIRULENCE;

ANTI-BACTERIAL AGENTS; DNA METHYLATION; GENE EXPRESSION PROFILING; HUMANS; MICROBIAL SENSITIVITY TESTS; PLAGUE VACCINE; SITE-SPECIFIC DNA-METHYLTRANSFERASE (ADENINE-SPECIFIC); STRUCTURE-ACTIVITY RELATIONSHIP; VIRULENCE; VIRULENCE FACTORS; YERSINIA PESTIS;

EID: 84872870685     PISSN: 00071188     EISSN: 14765381     Source Type: Journal    
DOI: 10.1111/j.1476-5381.2012.02134.x     Document Type: Article

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