-
1
-
-
0018155445
-
Critical evaluation of the potential error in pharmacokinetic studies of using the linear trapezoidal rule method for the calculation of the area under the plasma level-time curve
-
Chiou, W. L., Critical evaluation of the potential error in pharmacokinetic studies of using the linear trapezoidal rule method for the calculation of the area under the plasma level-time curve. J. Pharmacokinet. Biopharm., 6, 539-546 (1978).
-
(1978)
J. Pharmacokinet. Biopharm.
, vol.6
, pp. 539-546
-
-
Chiou, W.L.1
-
2
-
-
53749090602
-
Effects of cyclosporin A and itraconazole on the pharmacokinetics of atorvastatin in rats
-
Dong, J., Yu, X., Wang, L., Sun, Y. B., Chen, X. J., and Wang, G. J., Effects of cyclosporin A and itraconazole on the pharmacokinetics of atorvastatin in rats. Acta Pharmacol. Sin., 29, 1247-1252 (2008).
-
(2008)
Acta Pharmacol. Sin.
, vol.29
, pp. 1247-1252
-
-
Dong, J.1
Yu, X.2
Wang, L.3
Sun, Y.B.4
Chen, X.J.5
Wang, G.J.6
-
3
-
-
33846210597
-
Determination of the active and inactive metabolites of prasugrel in human plasma by liquid chromatography/tandem mass spectrometry
-
Farid, N. A., Mcintosh, M., Garofolo, F., Wong, E., Shwajch, A., Kennedy, M., Young, M., Sarkar, P., Kawabata, K., Takahashi, M., and Pang, H., Determination of the active and inactive metabolites of prasugrel in human plasma by liquid chromatography/tandem mass spectrometry. Rapid Commun. Mass Spectrom., 21, 169-179 (2007a).
-
(2007)
Rapid Commun. Mass Spectrom.
, vol.21
, pp. 169-179
-
-
Farid, N.A.1
McIntosh, M.2
Garofolo, F.3
Wong, E.4
Shwajch, A.5
Kennedy, M.6
Young, M.7
Sarkar, P.8
Kawabata, K.9
Takahashi, M.10
Pang, H.11
-
4
-
-
34247256797
-
Cytochrome P450 3A inhibition by ketoconazole affects prasugrel and clopidogrel pharmacokinetics and pharmacodynamics differently
-
Farid, N. A., Payne, C. D., Small, D. S., Winters, K. J., Ernest, C. S., 2nd, Brandt, J. T., Darstein, C., Jakubowski, J. A., and Salazar, D. E., Cytochrome P450 3A inhibition by ketoconazole affects prasugrel and clopidogrel pharmacokinetics and pharmacodynamics differently. Clin. Pharmacol. Ther., 81, 735-741 (2007b).
-
(2007)
Clin. Pharmacol. Ther.
, vol.81
, pp. 735-741
-
-
Farid, N.A.1
Payne, C.D.2
Small, D.S.3
Winters, K.J.4
Ernest, I.I.C.S.5
Brandt, J.T.6
Darstein, C.7
Jakubowski, J.A.8
Salazar, D.E.9
-
6
-
-
78649661850
-
Importance of P-glycoprotein for drug-drug interactions
-
Glaeser, H., Importance of P-glycoprotein for drug-drug interactions. Handb. Exp. Pharmacol., 201, 285-297 (2011).
-
(2011)
Handb. Exp. Pharmacol.
, vol.201
, pp. 285-297
-
-
Glaeser, H.1
-
7
-
-
0032754284
-
The role of intestinal P-glycoprotein in the interaction of digoxin and rifampin
-
Greiner, B., Eichelbaum, M., Fritz, P., Kreichgauer, H. P., Von Richter, O., Zundler, J., and Kroemer, H. K., The role of intestinal P-glycoprotein in the interaction of digoxin and rifampin. J. Clin. Invest., 104, 147-153 (1999).
-
(1999)
J. Clin. Invest.
, vol.104
, pp. 147-153
-
-
Greiner, B.1
Eichelbaum, M.2
Fritz, P.3
Kreichgauer, H.P.4
Von Richter, O.5
Zundler, J.6
Kroemer, H.K.7
-
8
-
-
66149110785
-
Comparison of formation of thiolactones and active metabolites of prasugrel and clopidogrel in rats and dogs
-
Hagihara, K., Kazui, M., Ikenaga, H., Nanba, T., Fusegawa, K., Takahashi, M., Kurihara, A., Okazaki, O., Farid, N. A., and Ikeda, T., Comparison of formation of thiolactones and active metabolites of prasugrel and clopidogrel in rats and dogs. Xenobiotica, 39, 218-226 (2009).
-
(2009)
Xenobiotica
, vol.39
, pp. 218-226
-
-
Hagihara, K.1
Kazui, M.2
Ikenaga, H.3
Nanba, T.4
Fusegawa, K.5
Takahashi, M.6
Kurihara, A.7
Okazaki, O.8
Farid, N.A.9
Ikeda, T.10
-
9
-
-
0036299716
-
Effects of various principles from Chinese herbal medicine on rhodamine123 accumulation in brain capillary endothelial cells
-
He, L. and Liu, G. Q., Effects of various principles from Chinese herbal medicine on rhodamine123 accumulation in brain capillary endothelial cells. Acta Pharmacol. Sin., 23, 591-596 (2002).
-
(2002)
Acta Pharmacol. Sin.
, vol.23
, pp. 591-596
-
-
He, L.1
Liu, G.Q.2
-
10
-
-
70350647476
-
Characterization of cardamonin metabolism by P450 in different species via HPLC-ESI-ion trap and UPLC-ESI-quadrupole mass spectrometry
-
He, Y. Q., Yang, L., Liu, Y., Zhang, J. W., Tang, J., Su, J., Li, Y. Y., Lu, Y. L., Wang, C. H., and Wang, Z. T., Characterization of cardamonin metabolism by P450 in different species via HPLC-ESI-ion trap and UPLC-ESI-quadrupole mass spectrometry. Acta Pharmacol. Sin., 30, 1462-1470 (2009).
-
(2009)
Acta Pharmacol. Sin.
, vol.30
, pp. 1462-1470
-
-
He, Y.Q.1
Yang, L.2
Liu, Y.3
Zhang, J.W.4
Tang, J.5
Su, J.6
Li, Y.Y.7
Lu, Y.L.8
Wang, C.H.9
Wang, Z.T.10
-
11
-
-
84872115491
-
-
Cited Aug 11.
-
IMS. Top Ten Global Products - 2007. Cited 2011 Aug 11. Available from: http://www.imshealth.com/deployedfiles/imshealth/Global/Content/StaticFile/ Top-Line-Data/Top10GlobalProducts.pdf.
-
(2011)
Top Ten Global Products - 2007
-
-
-
12
-
-
70350335772
-
Antiplatelet aggregation activity of compounds isolated from Guttiferae species in human whole blood
-
Jantan, I., Yasin, Y. H. M., Jalil, J., Murad, S., and Idris, M. S., Antiplatelet aggregation activity of compounds isolated from Guttiferae species in human whole blood. Pharm. Biol., 47, 1090-1095 (2009).
-
(2009)
Pharm. Biol.
, vol.47
, pp. 1090-1095
-
-
Jantan, I.1
Yasin, Y.H.M.2
Jalil, J.3
Murad, S.4
Idris, M.S.5
-
13
-
-
33645830172
-
A surface glycoprotein modulating drug permeability in Chinese hamster ovary cell mutants
-
Juliano, R. L. and Ling, V., A surface glycoprotein modulating drug permeability in Chinese hamster ovary cell mutants. Biochim. Biophys. Acta, 455, 152-162 (1976).
-
(1976)
Biochim. Biophys. Acta
, vol.455
, pp. 152-162
-
-
Juliano, R.L.1
Ling, V.2
-
14
-
-
42449156364
-
Modest effect of impaired P-glycoprotein on the plasma concentrations of fexofenadine, quinidine, and loperamide following oral administration in collies
-
Kitamura, Y., Koto, H., Matsuura, S., Kawabata, T., Tsuchiya, H., Kusuhara, H., Tsujimoto, H., and Sugiyama, Y., Modest effect of impaired P-glycoprotein on the plasma concentrations of fexofenadine, quinidine, and loperamide following oral administration in collies. Drug Metab. Dispos., 36, 807-810 (2008).
-
(2008)
Drug Metab. Dispos.
, vol.36
, pp. 807-810
-
-
Kitamura, Y.1
Koto, H.2
Matsuura, S.3
Kawabata, T.4
Tsuchiya, H.5
Kusuhara, H.6
Tsujimoto, H.7
Sugiyama, Y.8
-
15
-
-
55149116576
-
Intra-herb pharmacokinetics interaction between quercetin and isorhamentin
-
Lan, K., He, J. L., Tian, Y., Tan, F., Jiang, X. H., Wang, L., and Ye, L. M., Intra-herb pharmacokinetics interaction between quercetin and isorhamentin. Acta Pharmacol. Sin., 29, 1376-1382 (2008).
-
(2008)
Acta Pharmacol. Sin.
, vol.29
, pp. 1376-1382
-
-
Lan, K.1
He, J.L.2
Tian, Y.3
Tan, F.4
Jiang, X.H.5
Wang, L.6
Ye, L.M.7
-
16
-
-
84859101513
-
Absorption enhancement studies of clopidogrel hydrogen sulphate in rat everted gut sacs
-
Lassoued, M. A., Sfar, S., Bouraoui, A., and Khemiss, F., Absorption enhancement studies of clopidogrel hydrogen sulphate in rat everted gut sacs. J. Pharm. Pharmacol., 64, 541-552 (2012).
-
(2012)
J. Pharm. Pharmacol.
, vol.64
, pp. 541-552
-
-
Lassoued, M.A.1
Sfar, S.2
Bouraoui, A.3
Khemiss, F.4
-
17
-
-
77149136766
-
Pharmacokinetic Interaction between Telithromycin and Metformin in Diabetes Mellitus Rats
-
Lee, J. H., Kang, H. E., and Lee, M. G., Pharmacokinetic interaction between telithromycin and metformin in diabetes mellitus rats. Xenobiotica, 40, 217-224 (2010).
-
(2010)
Xenobiotica
, vol.40
, pp. 217-224
-
-
Lee, J.H.1
Kang, H.E.2
Lee, M.G.3
-
18
-
-
34250704230
-
Esterase inhibition by grapefruit juice flavonoids leading to a new drug interaction
-
Li, P., Callery, P. S., Gan, L. S., and Balani, S. K., Esterase inhibition by grapefruit juice flavonoids leading to a new drug interaction. Drug Metab. Dispos., 35, 1203-1208 (2007).
-
(2007)
Drug Metab. Dispos.
, vol.35
, pp. 1203-1208
-
-
Li, P.1
Callery, P.S.2
Gan, L.S.3
Balani, S.K.4
-
19
-
-
78649914959
-
Characterization of nuciferine metabolism by P450 enzymes and uridine diphosphate glucuronosyltransferases in liver microsomes from humans and animals
-
Lu, Y. L., He, Y. Q., Wang, M., Zhang, L., Yang, L., Wang, Z. T., and Ji, G., Characterization of nuciferine metabolism by P450 enzymes and uridine diphosphate glucuronosyltransferases in liver microsomes from humans and animals. Acta Pharmacol. Sin., 31, 1635-1642 (2010).
-
(2010)
Acta Pharmacol. Sin.
, vol.31
, pp. 1635-1642
-
-
Lu, Y.L.1
He, Y.Q.2
Wang, M.3
Zhang, L.4
Yang, L.5
Wang, Z.T.6
Ji, G.7
-
20
-
-
33845473315
-
Species differences between mouse, rat, dog, monkey and human CYP-mediated drug metabolism, inhibition and induction
-
Martignoni, M., Groothuis, G. M., and De Kanter, R., Species differences between mouse, rat, dog, monkey and human CYP-mediated drug metabolism, inhibition and induction. Expert Opin. Drug Metab. Toxicol., 2, 875-894 (2006).
-
(2006)
Expert Opin. Drug Metab. Toxicol.
, vol.2
, pp. 875-894
-
-
Martignoni, M.1
Groothuis, G.M.2
De Kanter, R.3
-
21
-
-
73949094806
-
Immunosuppressors as multidrug resistance reversal agents
-
Morjani, H. and Madoulet, C., Immunosuppressors as multidrug resistance reversal agents. Methods Mol. Biol., 596, 433-446 (2010).
-
(2010)
Methods Mol. Biol.
, vol.596
, pp. 433-446
-
-
Morjani, H.1
Madoulet, C.2
-
22
-
-
18044378766
-
Clopidogrel and ticlopidine: P2Y12 adenosine diphosphate-receptor antagonists for the prevention of atherothrombosis
-
Savi, P. and Herbert, J. M., Clopidogrel and ticlopidine: P2Y12 adenosine diphosphate-receptor antagonists for the prevention of atherothrombosis. Semin. Thromb. Hemost., 31, 174-183 (2005).
-
(2005)
Semin. Thromb. Hemost.
, vol.31
, pp. 174-183
-
-
Savi, P.1
Herbert, J.M.2
-
23
-
-
0027981909
-
Quercetin potentiates the effect of adriamycin in a multidrug-resistant MCF-7 human breast-cancer cell line: P-glycoprotein as a possible target
-
Scambia, G., Ranelletti, F. O., Panici, P. B., De Vincenzo, R., Bonanno, G., Ferrandina, G., Piantelli, M., Bussa, S., Rumi, C., Cianfriglia, M., and Mancuso, S., Quercetin potentiates the effect of adriamycin in a multidrug-resistant MCF-7 human breast-cancer cell line: P-glycoprotein as a possible target. Cancer Chemother. Pharmacol., 34, 459-464 (1994).
-
(1994)
Cancer Chemother. Pharmacol.
, vol.34
, pp. 459-464
-
-
Scambia, G.1
Ranelletti, F.O.2
Panici, P.B.3
De Vincenzo, R.4
Bonanno, G.5
Ferrandina, G.6
Piantelli, M.7
Bussa, S.8
Rumi, C.9
Cianfriglia, M.10
Mancuso, S.11
-
24
-
-
58749090547
-
Genetic determinants of response to clopidogrel and cardiovascular events
-
Simon, T., Verstuyft, C., Mary-Krause, M., Quteineh, L., Drouet, E., Méneveau, N., Steg, P. G., Ferrières, J., Danchin, N., and Becquemont, L., Genetic determinants of response to clopidogrel and cardiovascular events. N. Engl. J. Med., 360, 363-375 (2009).
-
(2009)
N. Engl. J. Med.
, vol.360
, pp. 363-375
-
-
Simon, T.1
Verstuyft, C.2
Mary-Krause, M.3
Quteineh, L.4
Drouet, E.5
Méneveau, N.6
Steg, P.G.7
Ferrières, J.8
Danchin, N.9
Becquemont, L.10
-
25
-
-
0033748479
-
The effect of telmisartan on the steady-state pharmacokinetics of digoxin in healthy male volunteers
-
Stangier, J., Su, C. A., Hendriks, M. G., Van Lier, J. J., Sollie, F. A., Oosterhuis, B., and Jonkman, J. H., The effect of telmisartan on the steady-state pharmacokinetics of digoxin in healthy male volunteers. J. Clin. Pharmacol., 40, 1373- 1379 (2000).
-
(2000)
J. Clin. Pharmacol.
, vol.40
, pp. 1373-1379
-
-
Stangier, J.1
Su, C.A.2
Hendriks, M.G.3
Van Lier, J.J.4
Sollie, F.A.5
Oosterhuis, B.6
Jonkman, J.H.7
-
26
-
-
34250763702
-
Species differences of inhibitory effects on P-glycoprotein-mediated drug transport
-
Suzuyama, N., Katoh, M., Takeuchi, T., Yoshitomi, S., Higuchi, T., Asashi, S., and Yokoi, T., Species differences of inhibitory effects on P-glycoprotein-mediated drug transport. J. Pharm. Sci., 96, 1609-1618 (2007).
-
(2007)
J. Pharm. Sci.
, vol.96
, pp. 1609-1618
-
-
Suzuyama, N.1
Katoh, M.2
Takeuchi, T.3
Yoshitomi, S.4
Higuchi, T.5
Asashi, S.6
Yokoi, T.7
-
27
-
-
22344436690
-
P-glycoprotein plays a major role in the efflux of fexofenadine in the small intestine and blood-brain barrier, but only a limited role in its biliary excretion
-
Tahara, H., Kusuhara, H., Fuse, E., and Sugiyama, Y., P-glycoprotein plays a major role in the efflux of fexofenadine in the small intestine and blood-brain barrier, but only a limited role in its biliary excretion. Drug Metab. Dispos., 33, 963-968 (2005).
-
(2005)
Drug Metab. Dispos.
, vol.33
, pp. 963-968
-
-
Tahara, H.1
Kusuhara, H.2
Fuse, E.3
Sugiyama, Y.4
-
28
-
-
34548498086
-
Carboxylesterase in the liver and small intestine of experimental animals and human
-
Taketani, M., Shii, M., Ohura, K., Ninomiya, S., and Imai, T., Carboxylesterase in the liver and small intestine of experimental animals and human. Life Sci., 81, 924-932 (2007).
-
(2007)
Life Sci.
, vol.81
, pp. 924-932
-
-
Taketani, M.1
Shii, M.2
Ohura, K.3
Ninomiya, S.4
Imai, T.5
-
29
-
-
33751171573
-
Antiplatelet agents aspirin and clopidogrel are hydrolyzed by distinct carboxylesterases, and clopidogrel is transesterificated in the presence of ethyl alcohol
-
Tang, M., Mukundan, M., Yang, J., Charpentier, N., Lecluyse, E. L., Black, C., Yang, D., Shi, D., and Yan, B., Antiplatelet agents aspirin and clopidogrel are hydrolyzed by distinct carboxylesterases, and clopidogrel is transesterificated in the presence of ethyl alcohol. J. Pharmacol. Exp. Ther., 319, 1467-1476 (2006).
-
(2006)
J. Pharmacol. Exp. Ther.
, vol.319
, pp. 1467-1476
-
-
Tang, M.1
Mukundan, M.2
Yang, J.3
Charpentier, N.4
Lecluyse, E.L.5
Black, C.6
Yang, D.7
Shi, D.8
Yan, B.9
-
30
-
-
33751080762
-
Impact of P-glycoprotein on clopidogrel absorption
-
Taubert, D., Von Beckerath, N., Grimberg, G., Lazar, A., Jung, N., Goeser, T., Kastrati, A., Schomig, A., and Schomig, E., Impact of P-glycoprotein on clopidogrel absorption. Clin. Pharmacol. Ther., 80, 486-501 (2006).
-
(2006)
Clin. Pharmacol. Ther.
, vol.80
, pp. 486-501
-
-
Taubert, D.1
Von Beckerath, N.2
Grimberg, G.3
Lazar, A.4
Jung, N.5
Goeser, T.6
Kastrati, A.7
Schomig, A.8
Schomig, E.9
-
31
-
-
0031811031
-
Three important subgroups of hypertensive persons at greater risk of intracerebral hemorrhage. Melbourne Risk Factor Study Group
-
Thrift, A. G., Mcneil, J. J., Forbes, A., and Donnan, G. A., Three important subgroups of hypertensive persons at greater risk of intracerebral hemorrhage. Melbourne Risk Factor Study Group. Hypertension, 31, 1223-1229 (1998).
-
(1998)
Hypertension
, vol.31
, pp. 1223-1229
-
-
Thrift, A.G.1
McNeil, J.J.2
Forbes, A.3
Donnan, G.A.4
-
32
-
-
40949088898
-
Quercetin pretreatment increases the bioavailability of pioglitazone in rats: Involvement of CYP3A inhibition
-
Umathe, S. N., Dixit, P. V., Kumar, V., Bansod, K. U., and Wanjari, M. M., Quercetin pretreatment increases the bioavailability of pioglitazone in rats: involvement of CYP3A inhibition. Biochem. Pharmacol., 75, 1670-1676 (2008).
-
(2008)
Biochem. Pharmacol.
, vol.75
, pp. 1670-1676
-
-
Umathe, S.N.1
Dixit, P.V.2
Kumar, V.3
Bansod, K.U.4
Wanjari, M.M.5
-
33
-
-
0347510572
-
Lethal quercetin-digoxin interaction in pigs
-
Wang, Y. H., Chao, P. D., Hsiu, S. L., Wen, K. C., and Hou, Y. C., Lethal quercetin-digoxin interaction in pigs. Life Sci., 74, 1191-1197 (2004).
-
(2004)
Life Sci.
, vol.74
, pp. 1191-1197
-
-
Wang, Y.H.1
Chao, P.D.2
Hsiu, S.L.3
Wen, K.C.4
Hou, Y.C.5
-
34
-
-
77951031222
-
Interaction of angiotensin receptor type 1 blockers with ATPbinding cassette transporters
-
Weiss, J., Sauer, A., Divac, N., Herzog, M., Schwedhelm, E., Boger, R. H., Haefeli, W. E., and Benndorf, R. A., Interaction of angiotensin receptor type 1 blockers with ATPbinding cassette transporters. Biopharm. Drug Dispos., 31, 150-161 (2010).
-
(2010)
Biopharm. Drug Dispos.
, vol.31
, pp. 150-161
-
-
Weiss, J.1
Sauer, A.2
Divac, N.3
Herzog, M.4
Schwedhelm, E.5
Boger, R.H.6
Haefeli, W.E.7
Benndorf, R.A.8
-
35
-
-
46449103184
-
The biotransformation of prasugrel, a new thienopyridine prodrug, by the human carboxylesterases 1 and 2
-
Williams, E. T., Jones, K. O., Ponsler, G. D., Lowery, S. M., Perkins, E. J., Wrighton, S. A., Ruterbories, K. J., Kazui, M., and Farid, N. A., The biotransformation of prasugrel, a new thienopyridine prodrug, by the human carboxylesterases 1 and 2. Drug Metab. Dispos., 36, 1227-1232 (2008).
-
(2008)
Drug Metab. Dispos.
, vol.36
, pp. 1227-1232
-
-
Williams, E.T.1
Jones, K.O.2
Ponsler, G.D.3
Lowery, S.M.4
Perkins, E.J.5
Wrighton, S.A.6
Ruterbories, K.J.7
Kazui, M.8
Farid, N.A.9
|