The hypotensive activity and alpha1-adrenoceptor antagonistic properties of some aroxyalkyl derivatives of 2-methoxyphenylpiperazine

European Journal of Pharmacology

Volumn 698, Issue 1-3, 2013, Pages 335-344

  Kubacka, Monika ^a   Mogilski, Szczepan ^a   Filipek, Barbara ^a   Marona, Henryk ^a  

^a JAGIELLONIAN UNIVERSITY   (Poland)

Author keywords

1 adrenoceptor subtype; Hypotensive activity; Phenylpiperazine derivative; Selectivity

Indexed keywords

2 METHOXYPHENYLPIPERIZINE DERIVATIVE; ADRENALIN; ALPHA 1 ADRENERGIC RECEPTOR; ALPHA 1 ADRENERGIC RECEPTOR BLOCKING AGENT; ALPHA 1B ADRENERGIC RECEPTOR; ALPHA 1D ADRENERGIC RECEPTOR; ALPHA 1L ADRENERGIC RECEPTOR; ALPHA 2 ADRENERGIC RECEPTOR; METHOXAMINE; MH 101; MH 76; MH 77; MH 79; MH 88; NORADRENALIN; RECEPTOR SUBTYPE; UNCLASSIFIED DRUG; URAPIDIL;

ANIMAL EXPERIMENT; ANIMAL TISSUE; ANTIHYPERTENSIVE ACTIVITY; ARTICLE; CONTROLLED STUDY; GUINEA PIG; MALE; NONHUMAN; PRESSOR RESPONSE; PRIORITY JOURNAL; RABBIT; RAT; SPASMOLYSIS; VASODILATATION;

ADRENERGIC ALPHA-1 RECEPTOR ANTAGONISTS; ANIMALS; AORTA; BLOOD PRESSURE; DRUG DISCOVERY; GUINEA PIGS; ILEUM; MALE; MUSCLE CONTRACTION; PIPERAZINES; POTASSIUM CHLORIDE; RABBITS; RATS; RECEPTORS, ADRENERGIC, ALPHA-1; VASOCONSTRICTION;

EID: 84871920087     PISSN: 00142999     EISSN: 18790712     Source Type: Journal    
DOI: 10.1016/j.ejphar.2012.10.025     Document Type: Article

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