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Volumn 10, Issue 46, 2012, Pages 9223-9236

Synthesis and evaluation of M. tuberculosis salicylate synthase (MbtI) inhibitors designed to probe plasticity in the active site

(11) Manos Turvey, Alexandra a Cergol, Katie M a Salam, Noeris K a Bulloch, Esther M M b Chi, Gamma b Pang, Angel c,d Britton, Warwick J c,d West, Nicholas P c,d Baker, Edward N b Lott, J Shaun b Payne, Richard J a

a UNIVERSITY OF SYDNEY (Australia)

b UNIVERSITY OF AUCKLAND (New Zealand)

c CENTENARY INSTITUTE (Australia)

d UNIVERSITY OF SYDNEY (Australia)

Author keywords

[No Author keywords available]

Indexed keywords

ACTIVE SITE; COCRYSTAL STRUCTURE; DIMETHYL ESTERS; IN-VITRO; INHIBITION CONSTANTS; INHIBITORY ACTIVITY; M. TUBERCULOSIS; MICROMOLAR RANGE; MYCOBACTERIUM TUBERCULOSIS; SALICYLATE SYNTHASE; SIDE-CHAINS; SIDEROPHORES;

BIOCHEMISTRY; ENZYME ACTIVITY; SCAFFOLDS; TUBES (COMPONENTS);

ENZYME INHIBITION;

2,3 DIHYDROXYBENZOIC ACID; 2,3-DIHYDROXYBENZOIC ACID; ACRYLIC ACID DERIVATIVE; BACTERIAL PROTEIN; ENZYME INHIBITOR; ESTER; HYDROXYBENZOIC ACID DERIVATIVE; LYASE; SALICYLATE SYNTHETASE;

ARTICLE; CHEMICAL STRUCTURE; CHEMISTRY; DRUG ANTAGONISM; DRUG DESIGN; DRUG EFFECT; ENZYME ACTIVE SITE; ENZYMOLOGY; KINETICS; METABOLISM; MICROBIAL SENSITIVITY TEST; MICROBIAL VIABILITY; MOLECULAR LIBRARY; MYCOBACTERIUM TUBERCULOSIS; NUCLEAR MAGNETIC RESONANCE SPECTROSCOPY; PROTEIN BINDING; STRUCTURE ACTIVITY RELATION; SYNTHESIS; X RAY CRYSTALLOGRAPHY;

ACRYLATES; BACTERIAL PROTEINS; CATALYTIC DOMAIN; CRYSTALLOGRAPHY, X-RAY; DRUG DESIGN; ENZYME INHIBITORS; ESTERS; HYDROXYBENZOATES; KINETICS; LYASES; MAGNETIC RESONANCE SPECTROSCOPY; MICROBIAL SENSITIVITY TESTS; MICROBIAL VIABILITY; MODELS, MOLECULAR; MYCOBACTERIUM TUBERCULOSIS; PROTEIN BINDING; SMALL MOLECULE LIBRARIES; STRUCTURE-ACTIVITY RELATIONSHIP;

MYCOBACTERIUM TUBERCULOSIS;

EID: 84868652011 PISSN: 14770520 EISSN: None Source Type: Journal
DOI: 10.1039/c2ob26736e Document Type: Article

Times cited : (24)

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