Chemotherapy of leishmaniasis. Part XI: Synthesis and bioevaluation of novel isoxazole containing heteroretinoid and its amide derivatives

Bioorganic and Medicinal Chemistry Letters

Volumn 22, Issue 21, 2012, Pages 6559-6562

  Suryawanshi, S N ^a   Tiwari, Avinash ^a   Chandra, Naveen ^a   Ramesh, ^a   Gupta, Suman ^a  

^a CENTRAL DRUG RESEARCH INSTITUTE   (India)

Author keywords

Hamster; Heteroretinoid; In vivo trial; Isoxazole; Leishmania donovani

Indexed keywords

AMIDE; ANTILEISHMANIAL AGENT; ISOXAZOLE; RETINOID;

ANTILEISHMANIAL ACTIVITY; ARTICLE; CHEMICAL REACTION; CHEMOTHERAPY; COMPETITIVE INHIBITION; DRUG ACTIVITY; DRUG SCREENING; DRUG STRUCTURE; DRUG SYNTHESIS; HAMSTER; LEISHMANIASIS; MICROBIAL GROWTH; MOLECULAR WEIGHT; NONHUMAN;

AMIDES; ANIMALS; ANTIPROTOZOAL AGENTS; CRICETINAE; FEMALE; ISOXAZOLES; LEISHMANIA DONOVANI; LEISHMANIASIS; MALE; MOLECULAR STRUCTURE; RETINOIDS;

CRICETINAE; LEISHMANIA DONOVANI;

EID: 84867581168     PISSN: 0960894X     EISSN: 14643405     Source Type: Journal    
DOI: 10.1016/j.bmcl.2012.09.024     Document Type: Article

References (23)

1. F. Frézard, C. Demicheli, and R.R. Ribeiro Molecules 14 2009 2317
2. E.M. Moore, and D.N. Lockwood J. Global Infect. Dis. 2 2010 151
3. H.C. Maltezou Biomed. Biotechnol. 2010 2010 617521
4. L.V. Alves, M.M. Do Canto-Cavalheiro, L. Cysne-Finkelstein, and L. Leon Biol. Pharm. Bull. 26 2003 453
5. T. Koide, M. Nose, Y. Ogihara, Y. Yabu, and N. Ohta Biol. Pharm. Bull. 25 2002 131
6. D.C.F. Gomes, L.V. Alegrio, M.E.F. Lima, L.L. Leon, and C.A.C. Aranjo Arzneim-Farsch Drug Res. 52 2002 120
7. N. Tan, M. Kaloga, O. Radtke, A.F. Kiderlen, S. Oksuz, A. Ulubelen, and H. Kolodziej Phytochemistry 61 2002 881
8. M. Sairafianpour, J. Christensen, D. Staerk, B.A. Budnik, A. Kharazmi, K. Bagherzadeh, and J.W. Jaroszewski J. Nat. Prod. 64 2001 1398
9. A.J. Valderrama, J. Benites, M. Cortes, H. Pessoa-Mahana, E. Prina, and A. Fournet Bioorg. Med. Chem. 11 2003 4713
10. M. Anzaldi, E. Sottofattori, R. Rizzetto, B. Granello di Casaleto, and A. Balbi Eur. J. Med. Chem. 34 1999 837
11. A. Rosowsky, A.T. Papoulis, and S.F. Queener J. Heterocyclic Chem. 36 1999 723
12. B.B. Aggarwal, C. Sundaram, S. Prasad, and R. Kannappan Biochem. Pharmacology 80 2010 1613
13. E. Sadikoglou, G. Magoulas, C. Theodoropoulou, C.M. Athanassopoulos, E. Giannopoulou, O. Theodorakopoulou, D. Drainas, D. Papaioannou, and E. Papadimitriou Eur. J. Med Chem. 44 2009 3175
14. D. Simoni, F.P. Invidiata, R. Rondanin, S. Grimaudo, G. Cannizzo, E. Barbusca, F. Porretto, N. D'Alessandro, and M. Tolomeo J. Med. Chem. 42 1999 4961
15. J.V. Richard, and K.A. Werbovetz Curr. Opin. Chem. Biol. 14 2010 447
16. S. Pandey, S.N. Suryawanshi, S. Gupta, and V.M.L. Srivastava Eur. J. Med. Chem. 39 2004 969
17. N. Chandra, Ramesh, Ashutosh, N. Goyal, S.N. Suryawanshi, and S. Gupta Eur. J. Med. Chem. 40 2005 552
18. N. Chandra, S. Pandey, Ramesh, S.N. Suryawanshi, and S. Gupta Eur. J. Med. Chem. 41 2006 779
19. N. Sunduru, A. Agarwal, S.B. Katiyar, Nishi, N. Goyal, S. Gupta, and P.M.S. Chauhan Bioorg. Med. Chem. 14 2006 7706
20. N. Sunduru, Nishi, S. Palne, P.M.S. Chauhan, and S. Gupta Eur. J. Med. Chem. 44 2009 2473
21. S. Beveridge, R.J. Schnitzer, and F.I. Hanoking Experimental Chemotherapy 1 1963 257
22. S. Bhatnagar, P.Y. Guru, J.C. Katiyar, R. Srivastava, A. Mukherjee, M.S. Akhtar, M. Seth, and A.P. Bhaduri J. Indian Med. Res. 89 1989 439
23. S. Gupta, S. Tiwari, A.P. Bhaduri, and G.K. Jain Acta Trop. 84 2002 165