Design and evaluation of hydrochlorothiazide gastroretentive floating drug delivery system

Asian Journal of Pharmaceutical Sciences

Volumn 6, Issue 5, 2011, Pages 208-217

  Madaka, Srinivas ^a   Sanka, Krishna ^a   Veerareddy, Prabhakar Reddy ^a  

^a ST PETER'S INSTITUTE OF PHARMACEUTICAL SCIENCES   (India)

Author keywords

Buoyancy; Floating drug delivery system; In vitro drug release profile; In vivo gastric residence time; Stability

Indexed keywords

BICARBONATE; HYDROCHLOROTHIAZIDE; HYDROXYPROPYLMETHYLCELLULOSE; LACTOSE; MACROGOL; MICROCRYSTALLINE CELLULOSE;

ADULT; ARTICLE; CONCENTRATION (PARAMETERS); DRUG DELIVERY SYSTEM; DRUG DESIGN; DRUG GRANULATION; DRUG STABILITY; GASTRORETENTIVE FLOATING DRUG DELIVERY SYSTEM; GATRIC RESIDENCE TIME; HUMAN; HUMAN EXPERIMENT; HUMIDITY; HYDROPHILICITY; IN VITRO STUDY; IN VIVO STUDY; MATRIX TABLET; MEAN RESIDENCE TIME; NORMAL HUMAN; SUSTAINED DRUG RELEASE; TABLET COMPRESSION; TABLET FRIABILITY; TABLET HARDNESS; VISCOSITY;

EID: 84866556997     PISSN: 18180876     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

References (20)

1. Brahma NS, Kwon HK. Floating drug delivery systems: an approach to oral controlled drug delivery via gastric retention J. Control Release. 2000, 63: 235-259.
2. Shweta A, Ali J, Alka A, et al. Floating drug delivery systems: a review. AAPS Pharm Sci Tech. 2005, 6: Article 47.
3. Singh BN, Kim KH. Floating drug delivery systems: an approach to oral controlled drug delivery via gastric retention. J Control Release. 2000, 63: 235-259.
4. Liu Q, Fassihi R. Zero-order delivery of a highly soluble, low dose drug alfuzosin hydrochloride via gastro-retentive system. Int J Pharm. 2008, 348: 27-34.
5. Chen J, Park K. Synthesis of fast-swelling, superporous sucrose hydrogels. Carbohydr Polym. 2000, 41: 259-268.
6. Lee JW, Park JH, Robinson JR. Bioadhesive-based dosage forms: the next generation. J Pharm Sci. 2000, 89: 850-866.
7. Bardonnet P, Faivre V, Pugh W, et al. Gastroretentive dosage forms: overview and special case of Helicobacter pylori. J Control Release. 2006, 111: 1-18.
8. Klausner EA, Eran L, Michael F, et al. Expandable gastroretentive dosage forms. J. Control Release. 2003, 90: 143-162.
9. Alexander S, Juergen S, Roland B. Drug delivery to the upper small intestine window using gastroretentive technologies. Curr Opin Pharmacol. 2006, 6: 501-508.
10. Swamy PV, Bhosale UV, Hiremath SN, et al. Formulation and optimization of gastric floating drug delivery system of atenolol using 32 full factorial design. Indian drug. 2008, [45:] 296-300.
11. James WA. Expandable gastric retention device. 2004, US Patent US2004/0219186A1.
12. Government of India ministry of health and family welfare. The Pharmacopoeia of India. Controller of publication, 2007.
13. Mahesh CH, Paras J, Sachin CH, et al. Development of sustained release gastroretentive drug delivery system for ofloxacin: In vitro and in vivo evaluation. Int J Pharm. [2005,] 304: 178-184.
14. Moore JW, Flanner HH. Mathematical comparison of curves with an emphasis on in vitro dissolution profiles. Pharm Tech. 1996, 20: 64-74.
15. Dave BS, Amin AF, Patel MM. Gastroretentive drug delivery system of ranitidine hydrochloride: formulation and in vitro evaluation. AAPS Pharm Sci Tech. 2004, 5: article 34.
16. Mortazavia SA, Jaffariazar Z, Damercheli E. Formulation and in-vitro evaluation of ocular ciprofloxacin-containing minitablets prepared with different combinations of Carbopol 974P andvarious cellulose derivatives. Iran J Pharm Res. 2010, 9: 107-114.
17. Freitas MN, Marchetti JM. Nimuesulide PLA microspheres as a potential sustained release system for the treatment of inflammatory disease. Int J Pharm. 2005, 295: 201-211.
18. Dorozynski P, Jachowicz R, Kulinowski P, et al. The polymers for the preparation of hydrodynamically balanced systems-methods of evaluation, Drug Dev Ind Pharm. [2004,] 30: 947-957.
19. Tadros MI. Controlled-release effervescent floating matrix tablets of ciprofloxacin hydrochloride: development, optimization and in vitro-in vivo evaluation in healthy human volunteers. Eur J Pharm Biopharm. 2010, 74: 332-339.
20. Jain SK, Awasthi AM, Jain NK, et al. Calcium silicate based microsheres of rapiglinide for gastroretentive floating drug delivery: preparation and in vitro characterization. J Control Release. 2005, 107: 300-309.